CH479595A - Verfahren zur Herstellung von 1-Peracylglycosyl-5-azacytosinen - Google Patents
Verfahren zur Herstellung von 1-Peracylglycosyl-5-azacytosinenInfo
- Publication number
- CH479595A CH479595A CH1590864A CH1590864A CH479595A CH 479595 A CH479595 A CH 479595A CH 1590864 A CH1590864 A CH 1590864A CH 1590864 A CH1590864 A CH 1590864A CH 479595 A CH479595 A CH 479595A
- Authority
- CH
- Switzerland
- Prior art keywords
- peracylglycosyl
- azacytosines
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/12—Triazine radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS709363 | 1963-12-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH479595A true CH479595A (de) | 1969-10-15 |
Family
ID=5419399
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH1590864A CH479595A (de) | 1963-12-22 | 1964-12-09 | Verfahren zur Herstellung von 1-Peracylglycosyl-5-azacytosinen |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US3350388A (de) |
| AT (1) | AT252458B (de) |
| BE (1) | BE657451A (de) |
| BR (1) | BR6465569D0 (de) |
| CH (1) | CH479595A (de) |
| DE (1) | DE1245384B (de) |
| DK (1) | DK108500C (de) |
| ES (1) | ES307376A1 (de) |
| FI (1) | FI46389C (de) |
| FR (1) | FR1450440A (de) |
| GB (1) | GB1050899A (de) |
| IT (1) | IT1043755B (de) |
| NL (1) | NL6414959A (de) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1030970A (en) * | 1964-05-15 | 1966-05-25 | Inst Mikrobiologii Im Akad D K | Method for the preparation of 2', 3', 5'-tri-o-acyl-6-azacytidines |
| DE2012888C3 (de) * | 1970-03-14 | 1981-04-02 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden |
| US6887855B2 (en) | 2003-03-17 | 2005-05-03 | Pharmion Corporation | Forms of 5-azacytidine |
| US7038038B2 (en) * | 2003-03-17 | 2006-05-02 | Pharmion Corporation | Synthesis of 5-azacytidine |
| US6943249B2 (en) * | 2003-03-17 | 2005-09-13 | Ash Stevens, Inc. | Methods for isolating crystalline Form I of 5-azacytidine |
| US20060014949A1 (en) * | 2004-07-13 | 2006-01-19 | Supergen Inc. | Compositions and formulations of decitabine polymorphs and methods of use thereof |
| US8741858B2 (en) | 2007-09-21 | 2014-06-03 | Zhongxu Ren | Oligomer-nucleoside phosphate conjugates |
| UA99308C2 (ru) * | 2007-09-26 | 2012-08-10 | Маунт Синай Скул Оф Медсин | Аналог азацитидина и его применение |
| ES2774226T3 (es) | 2008-05-15 | 2020-07-17 | Celgene Corp | Formulaciones orales de análogos de citidina y métodos de uso de los mismos |
| EP2321302B1 (de) | 2008-08-01 | 2014-10-29 | Dr. Reddy's Laboratories Ltd. | Herstellungsverfahren für azacitidin und polymorphen davon |
| AR073003A1 (es) * | 2008-08-08 | 2010-10-06 | Scinopharm Taiwan Ltd | Proceso para preparar 5-azacitosina nucleosidos y sus derivados |
| CA2755976C (en) * | 2009-03-23 | 2020-04-07 | Ambit Biosciences Corporation | Methods of treatment using combination therapy |
| IT1399195B1 (it) | 2010-03-30 | 2013-04-11 | Chemi Spa | Processo per la sintesi di azacitidina e decitabina |
| US9951098B2 (en) | 2011-03-31 | 2018-04-24 | Pharmion Llc | Synthesis of 5-azacytidine |
| US9913822B2 (en) | 2012-04-04 | 2018-03-13 | Halozyme, Inc. | Combination therapy with an anti-hyaluronan agent and therapeutic agent |
| CN108239128B (zh) | 2016-12-23 | 2019-03-29 | 江苏奥赛康药业股份有限公司 | β-核苷类化合物的制备方法 |
| US20190351031A1 (en) | 2018-05-16 | 2019-11-21 | Halozyme, Inc. | Methods of selecting subjects for combination cancer therapy with a polymer-conjugated soluble ph20 |
-
0
- GB GB1050899D patent/GB1050899A/en active Active
-
1964
- 1964-12-08 DE DEC34587A patent/DE1245384B/de active Pending
- 1964-12-09 CH CH1590864A patent/CH479595A/de not_active IP Right Cessation
- 1964-12-10 AT AT1047164A patent/AT252458B/de active
- 1964-12-12 FI FI642632A patent/FI46389C/fi active
- 1964-12-14 US US418273A patent/US3350388A/en not_active Expired - Lifetime
- 1964-12-18 DK DK620664AA patent/DK108500C/da active
- 1964-12-19 IT IT27006/64A patent/IT1043755B/it active
- 1964-12-21 ES ES0307376A patent/ES307376A1/es not_active Expired
- 1964-12-22 NL NL6414959A patent/NL6414959A/xx unknown
- 1964-12-22 BE BE657451D patent/BE657451A/xx unknown
- 1964-12-22 FR FR999626A patent/FR1450440A/fr not_active Expired
- 1964-12-22 BR BR165569/64A patent/BR6465569D0/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NL6414959A (de) | 1965-06-23 |
| FI46389C (fi) | 1973-03-12 |
| DK108500C (da) | 1967-12-27 |
| DE1245384B (de) | 1967-07-27 |
| FI46389B (de) | 1972-11-30 |
| BR6465569D0 (pt) | 1973-08-02 |
| IT1043755B (it) | 1980-02-29 |
| US3350388A (en) | 1967-10-31 |
| ES307376A1 (es) | 1965-05-01 |
| GB1050899A (de) | |
| AT252458B (de) | 1967-02-27 |
| FR1450440A (fr) | 1966-06-24 |
| BE657451A (de) | 1965-04-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CH463787A (de) | Verfahren zur Herstellung von Polyiminolactonen | |
| CH479595A (de) | Verfahren zur Herstellung von 1-Peracylglycosyl-5-azacytosinen | |
| CH444868A (de) | Verfahren zur Herstellung von Fluoracylaziridinen | |
| CH471134A (de) | Verfahren zur Herstellung von Pyrazinoylbenzamidinen | |
| CH466300A (de) | Verfahren zur Herstellung von Dihydrotriazinen | |
| CH469696A (de) | Verfahren zur Herstellung von 2-Guanidino-alkylchromanen | |
| CH449623A (de) | Verfahren zur Herstellung von 4-Alkyl-5-cyan-oxazolen | |
| CH438286A (de) | Verfahren zur Herstellung von Dibenzocycloheptadien-ketoxim-O-äthern | |
| AT244338B (de) | Verfahren zur Herstellung von 3-Amino-isoxazolen | |
| CH466272A (de) | Verfahren zur Herstellung von Cycloalkylmethylaminobenzophenonen | |
| CH440240A (de) | Verfahren zur Herstellung von Fluorjodalkanen | |
| CH456579A (de) | Verfahren zur Herstellung von Diphenylbenzocycloalkenen | |
| CH426836A (de) | Verfahren zur Herstellung von Naphthindolizinchinonen | |
| CH430716A (de) | Verfahren zur Herstellung von trans-2-Phenyl-3-methylmorpholin | |
| CH432536A (de) | Verfahren zur Herstellung von Diamino-monoazidotriazinen | |
| CH470376A (de) | Verfahren zur Herstellung von 17a-Äthinyl-19-nor-testosteron | |
| CH447211A (de) | Verfahren zur Herstellung von Diaminodihydroxy-anthrachinonen | |
| CH425809A (de) | Verfahren zur Herstellung von Pyridazoniminen | |
| CH416106A (de) | Verfahren zur Herstellung von Polydodecalactam | |
| CH459973A (de) | Verfahren zur Herstellung von Acetylacetamiden | |
| CH450378A (de) | Verfahren zur Herstellung von B-Hydroxyäthylthiocelestosaminid | |
| CH479570A (de) | Verfahren zur Herstellung von 7a-Alkyl-19-nor-steroiden | |
| CH436342A (de) | Verfahren zur Herstellung von substituierten 1-Hydroxy-2-amino-1-phenylalkanen | |
| CH442340A (de) | Verfahren zur Herstellung von Aminoalkyl-1-naphthylacetamiden | |
| CH482664A (de) | Verfahren zur Herstellung von 6-Methyl- 14-pregnenen |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PL | Patent ceased |