CH558374A - PROCESS FOR THE PRODUCTION OF ARYL-SUBSTITUTED PIPERAZINYL ALKYL- OR. ALKENYL CHINAZOLONE (4) DERIVATIVES. - Google Patents

PROCESS FOR THE PRODUCTION OF ARYL-SUBSTITUTED PIPERAZINYL ALKYL- OR. ALKENYL CHINAZOLONE (4) DERIVATIVES.

Info

Publication number
CH558374A
CH558374A CH450074A CH450074A CH558374A CH 558374 A CH558374 A CH 558374A CH 450074 A CH450074 A CH 450074A CH 450074 A CH450074 A CH 450074A CH 558374 A CH558374 A CH 558374A
Authority
CH
Switzerland
Prior art keywords
chinazolone
alkenyl
aryl
derivatives
production
Prior art date
Application number
CH450074A
Other languages
German (de)
Original Assignee
Byk Gulden Lomberg Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Byk Gulden Lomberg Chem Fab filed Critical Byk Gulden Lomberg Chem Fab
Publication of CH558374A publication Critical patent/CH558374A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH450074A 1970-06-05 1971-06-02 PROCESS FOR THE PRODUCTION OF ARYL-SUBSTITUTED PIPERAZINYL ALKYL- OR. ALKENYL CHINAZOLONE (4) DERIVATIVES. CH558374A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19702027645 DE2027645A1 (en) 1970-06-05 1970-06-05 Piperazinylalkyl quinazolone (4) den vate, process for their preparation and medicinal products containing them

Publications (1)

Publication Number Publication Date
CH558374A true CH558374A (en) 1975-01-31

Family

ID=5773104

Family Applications (3)

Application Number Title Priority Date Filing Date
CH450074A CH558374A (en) 1970-06-05 1971-06-02 PROCESS FOR THE PRODUCTION OF ARYL-SUBSTITUTED PIPERAZINYL ALKYL- OR. ALKENYL CHINAZOLONE (4) DERIVATIVES.
CH450174A CH569732A5 (en) 1970-06-05 1971-06-02
CH802071A CH557829A (en) 1970-06-05 1971-06-02 PROCESS FOR THE PRODUCTION OF ARYL-SUBSTITUTED PIPERAZINYL-ALKYL- OR. ALKENYL CHINAZOLONE (4) DERIVATIVES.

Family Applications After (2)

Application Number Title Priority Date Filing Date
CH450174A CH569732A5 (en) 1970-06-05 1971-06-02
CH802071A CH557829A (en) 1970-06-05 1971-06-02 PROCESS FOR THE PRODUCTION OF ARYL-SUBSTITUTED PIPERAZINYL-ALKYL- OR. ALKENYL CHINAZOLONE (4) DERIVATIVES.

Country Status (10)

Country Link
US (1) US3984555A (en)
AT (3) AT318628B (en)
BE (1) BE768137A (en)
CA (1) CA951319A (en)
CH (3) CH558374A (en)
DE (1) DE2027645A1 (en)
FR (1) FR2100726B1 (en)
GB (1) GB1331522A (en)
LU (1) LU63267A1 (en)
NL (1) NL7107695A (en)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US6723727B1 (en) * 1996-12-20 2004-04-20 Hoechst Aktiengesellschaft Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them
EP0903344B1 (en) * 1997-08-21 2011-01-26 Shiseido Co., Ltd. Quinazolin-4-one derivatives, their preparation and their use as hair growth promoters or in external compositions for skin
AU7734700A (en) 1999-10-01 2001-05-10 Advanced Medicine, Inc. Macrocyclic quinazolinones and their use as local anesthetics
DK2223922T3 (en) * 2000-04-25 2016-06-06 Icos Corp Inhibitors of HUMANPHOSPHATIDYL-inositol 3-KINASEDELTA
US6667300B2 (en) 2000-04-25 2003-12-23 Icos Corporation Inhibitors of human phosphatidylinositol 3-kinase delta
AUPR201600A0 (en) * 2000-12-11 2001-01-11 Fujisawa Pharmaceutical Co., Ltd. Quinazolinone derivative
CA2459583A1 (en) 2001-09-05 2003-03-13 Minerva Biotechnologies Corporation Compositions and methods of treatment of cancer
JP2005501887A (en) * 2001-09-05 2005-01-20 ミナーヴァ・バイオテクノロジーズ・コーポレーション Compositions and uses thereof in the treatment of cancer
AU2002363429B2 (en) * 2001-11-07 2008-05-08 Merck & Co., Inc. Mitotic kinesin inhibitors
AUPS019702A0 (en) * 2002-01-29 2002-02-21 Fujisawa Pharmaceutical Co., Ltd. Condensed heterocyclic compounds
AU2003262747A1 (en) * 2002-08-21 2004-03-11 Cytokinetics, Inc. Compounds, compositions, and methods
US20060052345A1 (en) * 2002-11-04 2006-03-09 Nps Pharmaceuticals, Inc. Quinazolinone compounds as calcilytics
ATE440825T1 (en) * 2003-06-06 2009-09-15 Vertex Pharma PYRIMIDINE DERIVATIVES FOR USE AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS
US20050043239A1 (en) * 2003-08-14 2005-02-24 Jason Douangpanya Methods of inhibiting immune responses stimulated by an endogenous factor
US20050054614A1 (en) * 2003-08-14 2005-03-10 Diacovo Thomas G. Methods of inhibiting leukocyte accumulation
EP1761540B1 (en) 2004-05-13 2016-09-28 Icos Corporation Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta
CA2567883A1 (en) * 2004-05-25 2005-12-15 Icos Corporation Methods for treating and/or preventing aberrant proliferation of hematopoietic cells
WO2006089106A2 (en) * 2005-02-17 2006-08-24 Icos Corporation Phosphoinositide 3-kinase inhibitors for inhibiting leukocyte accumulation
US8349850B2 (en) 2006-03-28 2013-01-08 Atir Holding S.A. Heterocyclic compounds and uses thereof in the treatment of sexual disorders
US9492449B2 (en) 2008-11-13 2016-11-15 Gilead Calistoga Llc Therapies for hematologic malignancies
KR20160091440A (en) 2008-11-13 2016-08-02 길리아드 칼리스토가 엘엘씨 Therapies for hematologic malignancies
CA2756347A1 (en) 2009-03-24 2010-09-30 Gilead Calistoga Llc Atropisomers of 2-purinyl-3-tolyl-quinazolinone derivatives and methods of use
SG175259A1 (en) * 2009-04-20 2011-11-28 Gilead Calistoga Llc Methods of treatment for solid tumors
AU2010276160A1 (en) 2009-07-21 2012-02-09 Gilead Calistoga Llc Treatment of liver disorders with PI3K inhibitors
BRPI1003506B1 (en) 2010-09-24 2019-12-03 Ache Int Bvi Ltd alkyl-piperazine-phenyl-4 (3h) quinazolinone compound and use of the alkyl-piperazine-phenyl-4 (3h) quinazolinone compound associated with 5-ht1a and 5-ht2a serotonergic receptors
WO2012140642A1 (en) 2011-04-10 2012-10-18 Atir Holding S.A. Heterocyclic compounds and uses thereof in the treatment of sexual disorders
EA025407B1 (en) 2012-03-05 2016-12-30 Джилид Калистога Ллс Polymorphic form i of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-one
IN2015MN00002A (en) 2012-07-09 2015-10-16 Lupin Ltd
NZ720867A (en) 2013-12-20 2018-01-26 Gilead Calistoga Llc Process methods for phosphatidylinositol 3-kinase inhibitors
WO2015095605A1 (en) 2013-12-20 2015-06-25 Gilead Calistoga Llc Polymorphic forms of a hydrochloride salt of (s) -2-(9h-purin-6-ylamino) propyl) -5-fluoro-3-phenylquinazolin-4 (3h) -one
JP6455995B2 (en) 2014-06-13 2019-01-23 ギリアード サイエンシーズ, インコーポレイテッド Phosphatidylinositol 3-kinase inhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1249281B (en) * 1963-05-18

Also Published As

Publication number Publication date
DE2027645A1 (en) 1971-12-09
FR2100726A1 (en) 1972-03-24
US3984555A (en) 1976-10-05
CH569732A5 (en) 1975-11-28
GB1331522A (en) 1973-09-26
LU63267A1 (en) 1972-08-23
CA951319A (en) 1974-07-16
BE768137A (en) 1971-12-06
NL7107695A (en) 1971-12-07
AT318615B (en) 1974-11-11
AT318628B (en) 1974-11-11
AT317899B (en) 1974-09-25
FR2100726B1 (en) 1975-10-10
CH557829A (en) 1975-01-15

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Legal Events

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