CL2007003389A1 - Formas cristalinas de sales de acido zoledronico; composicion farmaceutica; y uso en el tratamiento del cancer. - Google Patents
Formas cristalinas de sales de acido zoledronico; composicion farmaceutica; y uso en el tratamiento del cancer.Info
- Publication number
- CL2007003389A1 CL2007003389A1 CL200703389A CL2007003389A CL2007003389A1 CL 2007003389 A1 CL2007003389 A1 CL 2007003389A1 CL 200703389 A CL200703389 A CL 200703389A CL 2007003389 A CL2007003389 A CL 2007003389A CL 2007003389 A1 CL2007003389 A1 CL 2007003389A1
- Authority
- CL
- Chile
- Prior art keywords
- cancer
- salts
- treatment
- pharmaceutical composition
- zoledronic acid
- Prior art date
Links
- 206010028980 Neoplasm Diseases 0.000 title 1
- 201000011510 cancer Diseases 0.000 title 1
- 239000013078 crystal Substances 0.000 title 1
- 239000008194 pharmaceutical composition Chemical class 0.000 title 1
- XRASPMIURGNCCH-UHFFFAOYSA-N zoledronic acid Chemical class OP(=O)(O)C(P(O)(O)=O)(O)CN1C=CN=C1 XRASPMIURGNCCH-UHFFFAOYSA-N 0.000 title 1
- 229960004276 zoledronic acid Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6503—Five-membered rings
- C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Physical Education & Sports Medicine (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Rheumatology (AREA)
- General Chemical & Material Sciences (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06124850A EP1925621A1 (en) | 2006-11-27 | 2006-11-27 | Crystalline forms of zoledronic acid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2007003389A1 true CL2007003389A1 (es) | 2008-06-27 |
Family
ID=37909616
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL200703389A CL2007003389A1 (es) | 2006-11-27 | 2007-11-26 | Formas cristalinas de sales de acido zoledronico; composicion farmaceutica; y uso en el tratamiento del cancer. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20100056481A1 (es) |
| EP (2) | EP1925621A1 (es) |
| JP (1) | JP2010510970A (es) |
| KR (1) | KR20090083407A (es) |
| CN (1) | CN101535323A (es) |
| AR (1) | AR063923A1 (es) |
| AU (1) | AU2007324833A1 (es) |
| BR (1) | BRPI0719567A2 (es) |
| CA (1) | CA2670638A1 (es) |
| CL (1) | CL2007003389A1 (es) |
| MX (1) | MX2009005413A (es) |
| PE (1) | PE20081391A1 (es) |
| RU (1) | RU2009123936A (es) |
| TW (1) | TW200829598A (es) |
| WO (1) | WO2008064849A1 (es) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2407746C2 (ru) * | 2008-09-29 | 2010-12-27 | ЗАО "Фарм-Синтез" | Радиофармацевтическое средство для диагностики и лечения (терапии) костных поражений скелета и способ его получения |
| US9169279B2 (en) | 2009-07-31 | 2015-10-27 | Thar Pharmaceuticals, Inc. | Crystallization method and bioavailability |
| US8980868B2 (en) | 2009-07-31 | 2015-03-17 | Thar Pharmaceuticals, Inc. | Oral forms of a phosphonic acid derivative |
| US20160016982A1 (en) | 2009-07-31 | 2016-01-21 | Thar Pharmaceuticals, Inc. | Crystallization method and bioavailability |
| DK2459176T3 (en) | 2009-07-31 | 2017-12-04 | Gruenenthal Gmbh | Crystallization process and bioavailability |
| CN105920023A (zh) * | 2009-09-01 | 2016-09-07 | 杜克大学 | 双膦酸类组合物及其治疗心力衰竭的方法 |
| AU2011239935A1 (en) | 2010-04-16 | 2012-11-08 | Novartis Ag | Methods and compositions for improving implant osseointegration |
| US9340565B2 (en) | 2010-11-24 | 2016-05-17 | Thar Pharmaceuticals, Inc. | Crystalline forms |
| JP6492321B2 (ja) * | 2015-03-23 | 2019-04-03 | 株式会社大阪合成有機化学研究所 | [1−ヒドロキシ−2−(イミダゾ[1,2−a]ピリジン−3−イル)エチリデン]ビスホスホン酸一水和物の製造方法 |
| EP3455229B1 (en) | 2016-05-13 | 2021-03-24 | Thar Pharma LLC | Novel crystalline forms |
| US10195218B2 (en) | 2016-05-31 | 2019-02-05 | Grunenthal Gmbh | Crystallization method and bioavailability |
| CN106749405B (zh) * | 2016-12-29 | 2019-07-16 | 江苏省原子医学研究所 | 一种咪唑杂环类双膦酸化合物及其制备方法、应用 |
| EP3713575A4 (en) | 2017-11-21 | 2021-08-25 | Rgenix, Inc. | POLYMORPHS AND THEIR USES |
| CN110551152A (zh) * | 2018-05-31 | 2019-12-10 | 四川科伦药物研究院有限公司 | 唑来膦酸一水合物及无水物晶型制备方法 |
| JP7644933B2 (ja) * | 2019-04-11 | 2025-03-13 | シァメン・イノヴァックス・バイオテック・カンパニー・リミテッド | ゾレドロン酸亜鉛マイクロ/ナノ粒子アジュバントの作製及びワクチンアジュバントとしてのその使用 |
| HUE067466T2 (hu) | 2019-12-13 | 2024-10-28 | Inspirna Inc | Fémsók és alkalmazásuk |
| CN112724174A (zh) * | 2020-12-30 | 2021-04-30 | 华南理工大学 | 一种薄片状双膦酸钙配合物及其制备方法 |
| CN112646193A (zh) * | 2020-12-30 | 2021-04-13 | 华南理工大学 | 一种块状双膦酸钙配合物及其制备方法 |
| CN112778365A (zh) * | 2020-12-30 | 2021-05-11 | 华南理工大学 | 一种唑来膦酸钙配合物及其制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4244422A1 (de) * | 1992-12-29 | 1994-06-30 | Boehringer Mannheim Gmbh | Schwerlösliche Zink- und Magnesiumsalze von 1,1-Bisphosphonsäuren, ihre Herstellung und Verwendung als Arzneimittel |
| US20040097468A1 (en) * | 2002-11-20 | 2004-05-20 | Wimalawansa Sunil J. | Method of treating osteoporosis and other bone disorders with upfront loading of bisphosphonates, and kits for such treatment |
| EP1612212A1 (en) * | 2003-07-03 | 2006-01-04 | Teva Pharmaceutical Industries Ltd | Zoledronic acid crystal forms, zoledronate sodium salt crystal forms, amorphous zoledronate sodium salt, and processes for their preparation |
| US20060178439A1 (en) * | 2005-01-04 | 2006-08-10 | Mohakhud Pradeep K | Crystalline form of zoledronic acid |
| AR054673A1 (es) * | 2005-07-28 | 2007-07-11 | Gador Sa | Una forma cristalina del acido zoledronico, un proceso para su obtencion y la composicion farmaceutica que la comprende |
| US20080255366A1 (en) * | 2005-09-12 | 2008-10-16 | Dr. Reddy's Laboratories Limited | Crystalline Trihydrate of Zoledronic Acid |
| WO2007125521A2 (en) * | 2006-05-02 | 2007-11-08 | Ranbaxy Laboratories Limited | Polymorphic form of zoledronic acid and processes for their preparation |
-
2006
- 2006-11-27 EP EP06124850A patent/EP1925621A1/en not_active Ceased
-
2007
- 2007-11-23 AR ARP070105215A patent/AR063923A1/es unknown
- 2007-11-23 PE PE2007001630A patent/PE20081391A1/es not_active Application Discontinuation
- 2007-11-26 AU AU2007324833A patent/AU2007324833A1/en not_active Abandoned
- 2007-11-26 JP JP2009537559A patent/JP2010510970A/ja active Pending
- 2007-11-26 CA CA002670638A patent/CA2670638A1/en not_active Abandoned
- 2007-11-26 WO PCT/EP2007/010255 patent/WO2008064849A1/en not_active Ceased
- 2007-11-26 BR BRPI0719567-2A patent/BRPI0719567A2/pt not_active Application Discontinuation
- 2007-11-26 CL CL200703389A patent/CL2007003389A1/es unknown
- 2007-11-26 RU RU2009123936/04A patent/RU2009123936A/ru not_active Application Discontinuation
- 2007-11-26 MX MX2009005413A patent/MX2009005413A/es not_active Application Discontinuation
- 2007-11-26 CN CNA2007800419850A patent/CN101535323A/zh active Pending
- 2007-11-26 US US12/515,742 patent/US20100056481A1/en not_active Abandoned
- 2007-11-26 KR KR1020097010727A patent/KR20090083407A/ko not_active Withdrawn
- 2007-11-26 EP EP07846821A patent/EP2089404A1/en not_active Withdrawn
- 2007-11-26 TW TW096144824A patent/TW200829598A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PE20081391A1 (es) | 2008-11-14 |
| EP2089404A1 (en) | 2009-08-19 |
| TW200829598A (en) | 2008-07-16 |
| BRPI0719567A2 (pt) | 2013-12-10 |
| MX2009005413A (es) | 2009-06-01 |
| WO2008064849A1 (en) | 2008-06-05 |
| CA2670638A1 (en) | 2008-06-05 |
| RU2009123936A (ru) | 2011-01-10 |
| CN101535323A (zh) | 2009-09-16 |
| AU2007324833A1 (en) | 2008-06-05 |
| KR20090083407A (ko) | 2009-08-03 |
| AR063923A1 (es) | 2009-02-25 |
| JP2010510970A (ja) | 2010-04-08 |
| US20100056481A1 (en) | 2010-03-04 |
| EP1925621A1 (en) | 2008-05-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CL2007003389A1 (es) | Formas cristalinas de sales de acido zoledronico; composicion farmaceutica; y uso en el tratamiento del cancer. | |
| CL2008001076A1 (es) | Compuestos derivados de sulfonamida; composicion farmaceutica; y uso en el tratamiento del cancer. | |
| CL2007000806A1 (es) | Compuestos derivados de heteropentaciclos sustituidos; proceso de preparacion; compuestos intermediarios; composicion farmaceutica; y uso en el tratamiento del cancer. | |
| SMT201600398B (it) | Inibitori di proteina chinasi (varianti), uso di questi nel trattamento di malattie oncologiche e composizione farmaceutica basata su questi | |
| CL2012003026A1 (es) | Composicion farmaceutica que comprende pioglitazona y linagliptina; procedimiento de preparacion; uso en el tratamiento de la diabetes tipo 2 o la obesidad. | |
| IL249838A0 (en) | Telomerase activating compounds for use in treating diseases related thereto | |
| CL2008001123A1 (es) | Compuestos derivados de acido lipoico; formulacion farmaceutica que lo comprende; y uso en el tratamiento del cancer. | |
| CL2007003635A1 (es) | Compuestos derivados de 6-amino-purin-8-ona; proceso de preparacion; composicion farmaceutica; proceso para preparar la composicion farmaceutica; y uso en el tratamiento de enfermedades alergicas, virales o cancer. | |
| CL2007000161A1 (es) | Compuestos derivados de 2,4-dioxoimidazolidina sustituida, inhibidores de proteinas cinasas; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer. | |
| BRPI0922233A2 (pt) | compostos, composições farmacêiticas e métodos para uso no tratamento de síndromes metabólicas. | |
| CL2008001234A1 (es) | Compuestos derivados de heterociclos nitrogenados, inhibidores de las proteinas de apoptosis; y uso en el tratamiento del cancer. | |
| CL2007002967A1 (es) | Forma cristalina a del compuesto 4-[3-(4-ciclopropancarbonil-piperazin-1-carbonil)-4-fluoro-bencil]-2h-ftalazin-1-ona; procedimiento de preparacion; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento de un | |
| CL2007002207A1 (es) | Compuestos derivados de sulfonilaminas; composicion farmaceutica; y uso de los compuestos en el tratamiento del glaucoma. | |
| CL2007001902A1 (es) | Compuestos derivados de piridina sustituidas; composicion farmaceutica; y uso en el tratamiento de un trastorno de agregacion de plaquetas. | |
| CL2013001654A1 (es) | Compuestos derivados de 6-amino-2-fenilamino-1h-bencimidazol-5-carboxamida; composicion farmaceutica; y su uso en el tratamiento y/o prevencion de las enfermedades inflamatorias y/o afecciones asociadas, en particular el dolor. | |
| EA201200550A1 (ru) | Фармацевтические композиции, включающие bi-1356 и метформин | |
| IL199151A (en) | Pyrimidine derivatives, their pharmaceutical preparations, their use in cancer treatment and their kits | |
| CL2007003774A1 (es) | Compuestos derivados de quinazolina sustituidos, inhibidores de quinasa; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, aterosclerosis y artritis. | |
| CL2008001633A1 (es) | Compuestos derivados de pirrolidin-3-carboxamida; composición farmacéutica; y uso comominhibidores de erk para el tratamiento del cancer. | |
| CL2013003372A1 (es) | Compuestos derivados de espiro-[1,3]-oxacinas y espiro-[1,4]-oxacepinas, inhibidores de bace1 y/o bace2; composicion farmaceutica; procedimiento para prepararlos; y su uso en el tratamiento y/o la profilaxis de la enfermedad de alzheimer y diabetes. | |
| CL2007003805A1 (es) | Forma cristalina del compuesto 3-{[5-(acetidin-1-ilcarbonil)piracin-2-il]oxi}-5-[(1-metiletil)oxi]-n-1h-pirazol-3-ilbenzamida; procedimiento de preparacion; composicion farmaceutica que comprende a dicha forma; y uso para el tratamiento de la diabete | |
| CL2014000849A1 (es) | Compuestos derivados de benzilindazoles sustituido, inhibidores de la quinasa bub1; procedimiento de fabricacion; composicion farmaceutica; combinacion farmaceutica; y su uso en el tratamiento de enfermedades hiperproliferativas. | |
| CL2007003038A1 (es) | Compuestos derivados de 2-fenil-6-aminocarbonil-pirimidina; composicion farmaceutica; y uso en el tratamiento de trastornos vasculares oclusivos. | |
| CL2007003672A1 (es) | Compuestos derivados de heteroaril-pirrolidinil-cetona y heteroaril-piperidinil-cetona; composicion farmaceutica; y uso en el tratamiento de la depresion y ansiedad. | |
| CL2012003322A1 (es) | Compuestos derivados de benzamida sustituidas; composicion farmacéutica; y uso en el tratamiento del cancer. |