CL2008002060A1 - Compuestos derivados de sulfonamida, inhibidores de la produccion de beta amiloide; metodo de preparacion; composicion farmaceutica; kit farmaceutico; y uso en el tratamiento de enfermedades tales como alzheimer, angiopatia amiloide, sindrome de down, entre otras. - Google Patents
Compuestos derivados de sulfonamida, inhibidores de la produccion de beta amiloide; metodo de preparacion; composicion farmaceutica; kit farmaceutico; y uso en el tratamiento de enfermedades tales como alzheimer, angiopatia amiloide, sindrome de down, entre otras.Info
- Publication number
- CL2008002060A1 CL2008002060A1 CL2008002060A CL2008002060A CL2008002060A1 CL 2008002060 A1 CL2008002060 A1 CL 2008002060A1 CL 2008002060 A CL2008002060 A CL 2008002060A CL 2008002060 A CL2008002060 A CL 2008002060A CL 2008002060 A1 CL2008002060 A1 CL 2008002060A1
- Authority
- CL
- Chile
- Prior art keywords
- alzheimer
- inhibitors
- diseases
- preparation
- treatment
- Prior art date
Links
- 102000013455 Amyloid beta-Peptides Human genes 0.000 title abstract 2
- 108010090849 Amyloid beta-Peptides Proteins 0.000 title abstract 2
- 206010059245 Angiopathy Diseases 0.000 title abstract 2
- 201000010374 Down Syndrome Diseases 0.000 title abstract 2
- 201000010099 disease Diseases 0.000 title abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- 229940124530 sulfonamide Drugs 0.000 title abstract 2
- 150000003456 sulfonamides Chemical class 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
- C07C311/16—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
- C07C311/17—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Compuestos derivados de sulfonamida, inhibidores de la producción de beta amiloide; método de preparación; composición farmacéutica; kit farmacéutico; y uso en el tratamiento de enfermedades, tales como, Alzheimer, angiopatía amiloide, Síndrome de Down, entre otras.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US95967507P | 2007-07-16 | 2007-07-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2008002060A1 true CL2008002060A1 (es) | 2008-11-21 |
Family
ID=39769171
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2008002060A CL2008002060A1 (es) | 2007-07-16 | 2008-07-14 | Compuestos derivados de sulfonamida, inhibidores de la produccion de beta amiloide; metodo de preparacion; composicion farmaceutica; kit farmaceutico; y uso en el tratamiento de enfermedades tales como alzheimer, angiopatia amiloide, sindrome de down, entre otras. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20090023801A1 (es) |
| EP (1) | EP2193117A1 (es) |
| JP (1) | JP2010533723A (es) |
| CA (1) | CA2693959A1 (es) |
| CL (1) | CL2008002060A1 (es) |
| PA (1) | PA8789701A1 (es) |
| PE (1) | PE20090445A1 (es) |
| TW (1) | TW200911779A (es) |
| WO (1) | WO2009012205A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA82093C2 (uk) * | 2003-03-31 | 2008-03-11 | Уайт | Фтор- та трифторалкіловмісні гетероциклічні сульфонамідні інгібітори утворення бета-амілоїду та їх похідні |
| WO2009089237A1 (en) * | 2008-01-11 | 2009-07-16 | Wyeth | Compositions containing o-sulfate and o-phosphate containing aryl sulfonamide derivatives useful as beta-amyloid inhibitors |
| AU2010232923A1 (en) * | 2009-04-03 | 2011-11-03 | Medisyn Technologies, Inc. | Compositions for treatment of Alzheimer's disease |
| US9156814B2 (en) * | 2011-04-21 | 2015-10-13 | Hong Kong Baptist University | Imaging beta-amyloid peptides and inhibition of beta-amyloid peptide aggregation |
| CN104649857B (zh) * | 2013-11-19 | 2017-05-17 | 中国科学院上海有机化学研究所 | 三氟甲基取代的叠氮、胺及杂环类化合物及制备方法 |
| TW202126617A (zh) | 2019-09-20 | 2021-07-16 | 美商富曼西公司 | 間二醯胺類殺蟲劑 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030104559A1 (en) * | 1998-03-27 | 2003-06-05 | Genentech, Inc. | Secreted and transmembrane polypeptides and nucleic acids encoding the same |
| UA74849C2 (en) * | 2000-11-17 | 2006-02-15 | Lilly Co Eli | Lactam |
| ES2267853T3 (es) * | 2000-12-13 | 2007-03-16 | Wyeth | Inhibidroes de sulfonamida heteriociclicos de la produccion de beta amiloides. |
| KR20050010882A (ko) * | 2002-06-11 | 2005-01-28 | 와이어쓰 | 베타 아밀로이드 생산의 치환 페닐술폰아미드 저해제 |
| UA82093C2 (uk) * | 2003-03-31 | 2008-03-11 | Уайт | Фтор- та трифторалкіловмісні гетероциклічні сульфонамідні інгібітори утворення бета-амілоїду та їх похідні |
| CA2552558A1 (en) * | 2004-01-16 | 2005-08-11 | Wyeth | Heterocyclic sulfonamide inhibitors of beta amyloid production containing an azole |
| AR059518A1 (es) * | 2006-02-17 | 2008-04-09 | Wyeth Corp | Metodos para preparar alcoholes sustituidos con sulfonamidas y sus compuestos intermedios |
| EP1984347A1 (en) * | 2006-02-17 | 2008-10-29 | Wyeth a Corporation of the State of Delaware | Selective n-sulfonylation of 2-amino trifluoroalkyl substituted alcohols |
| US7476762B2 (en) * | 2006-04-21 | 2009-01-13 | Wyeth | Methods for preparing sulfonamide compounds |
| US7550629B2 (en) * | 2006-04-21 | 2009-06-23 | Wyeth | Trifluoromethyl-containing phenylsulfonamide beta amyloid inhibitors |
-
2008
- 2008-07-14 WO PCT/US2008/069942 patent/WO2009012205A1/en not_active Ceased
- 2008-07-14 US US12/172,505 patent/US20090023801A1/en not_active Abandoned
- 2008-07-14 CA CA2693959A patent/CA2693959A1/en not_active Abandoned
- 2008-07-14 JP JP2010517095A patent/JP2010533723A/ja not_active Withdrawn
- 2008-07-14 PA PA20088789701A patent/PA8789701A1/es unknown
- 2008-07-14 EP EP08781785A patent/EP2193117A1/en not_active Withdrawn
- 2008-07-14 CL CL2008002060A patent/CL2008002060A1/es unknown
- 2008-07-14 PE PE2008001176A patent/PE20090445A1/es not_active Application Discontinuation
- 2008-07-14 TW TW097126640A patent/TW200911779A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW200911779A (en) | 2009-03-16 |
| EP2193117A1 (en) | 2010-06-09 |
| US20090023801A1 (en) | 2009-01-22 |
| PE20090445A1 (es) | 2009-05-18 |
| CA2693959A1 (en) | 2009-01-22 |
| WO2009012205A1 (en) | 2009-01-22 |
| PA8789701A1 (es) | 2009-04-23 |
| JP2010533723A (ja) | 2010-10-28 |
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