CL2011002500A1 - Compuestos derivados 1-alquil-cinolin-4(1h)-ona, moduladores de cb2; procedimiento de preparacion; composicion farmaceutica; y uso para tratar y prevenir el dolor, enfermedades inflamatorias, autoinmunes, entre otras. - Google Patents

Compuestos derivados 1-alquil-cinolin-4(1h)-ona, moduladores de cb2; procedimiento de preparacion; composicion farmaceutica; y uso para tratar y prevenir el dolor, enfermedades inflamatorias, autoinmunes, entre otras.

Info

Publication number
CL2011002500A1
CL2011002500A1 CL2011002500A CL2011002500A CL2011002500A1 CL 2011002500 A1 CL2011002500 A1 CL 2011002500A1 CL 2011002500 A CL2011002500 A CL 2011002500A CL 2011002500 A CL2011002500 A CL 2011002500A CL 2011002500 A1 CL2011002500 A1 CL 2011002500A1
Authority
CL
Chile
Prior art keywords
cinolin
modulators
autoimmune
treat
alkyl
Prior art date
Application number
CL2011002500A
Other languages
English (en)
Inventor
Elodie Barbagallo
Murielle Rinaldi-Carmona
Pascale Roux
Claude Vernhet
Carole Legeay
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41051781&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2011002500(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of CL2011002500A1 publication Critical patent/CL2011002500A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/28—Cinnolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/502—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with carbocyclic ring systems, e.g. cinnoline, phthalazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CL2011002500A 2009-04-07 2011-10-07 Compuestos derivados 1-alquil-cinolin-4(1h)-ona, moduladores de cb2; procedimiento de preparacion; composicion farmaceutica; y uso para tratar y prevenir el dolor, enfermedades inflamatorias, autoinmunes, entre otras. CL2011002500A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0901696A FR2944013B1 (fr) 2009-04-07 2009-04-07 Derives de 1-alkyl-cinnolin-4(1h)-one substitues,leur preparation et leur application en therapeutique.

Publications (1)

Publication Number Publication Date
CL2011002500A1 true CL2011002500A1 (es) 2012-03-23

Family

ID=41051781

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2011002500A CL2011002500A1 (es) 2009-04-07 2011-10-07 Compuestos derivados 1-alquil-cinolin-4(1h)-ona, moduladores de cb2; procedimiento de preparacion; composicion farmaceutica; y uso para tratar y prevenir el dolor, enfermedades inflamatorias, autoinmunes, entre otras.

Country Status (20)

Country Link
US (1) US8420651B2 (es)
EP (1) EP2417111B1 (es)
JP (1) JP5651683B2 (es)
KR (1) KR20120027212A (es)
CN (1) CN102459195A (es)
AR (1) AR076205A1 (es)
AU (1) AU2010233590A1 (es)
BR (1) BRPI1015951A2 (es)
CA (1) CA2757859A1 (es)
CL (1) CL2011002500A1 (es)
CO (1) CO6440578A2 (es)
EA (1) EA201171212A1 (es)
FR (1) FR2944013B1 (es)
IL (1) IL215512A0 (es)
MA (1) MA33250B1 (es)
MX (1) MX2011010650A (es)
SG (1) SG175128A1 (es)
TW (1) TW201040147A (es)
UY (1) UY32548A (es)
WO (1) WO2010116084A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021233861A1 (en) 2020-05-19 2021-11-25 Bayer Aktiengesellschaft Azabicyclic(thio)amides as fungicidal compounds
UY39214A (es) * 2020-05-19 2021-12-31 Syngenta Crop Protection Ag Compuestos herbicidas sustituídos con azufre
BR112022024413A2 (pt) 2020-06-10 2023-02-07 Bayer Ag Heterociclos substituídos com azabiciclila como fungicidas inovadores

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200306839A (en) * 2002-02-06 2003-12-01 Novartis Ag Quinazolinone derivatives and their use as CB agonists
WO2009053799A1 (en) * 2007-10-24 2009-04-30 Glenmark Pharmaceuticals, S.A. Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation
FR2933697B1 (fr) * 2008-07-11 2010-08-13 Sanofi Aventis Derives de 1-benzyl-cinnolin-4-(1h)-one substitues, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
TW201040147A (en) 2010-11-16
MX2011010650A (es) 2012-01-20
JP5651683B2 (ja) 2015-01-14
CO6440578A2 (es) 2012-05-15
EA201171212A1 (ru) 2012-04-30
JP2012522829A (ja) 2012-09-27
US8420651B2 (en) 2013-04-16
MA33250B1 (fr) 2012-05-02
CN102459195A (zh) 2012-05-16
EP2417111B1 (fr) 2014-06-04
UY32548A (es) 2010-11-30
AR076205A1 (es) 2011-05-26
WO2010116084A1 (fr) 2010-10-14
CA2757859A1 (fr) 2010-10-14
FR2944013B1 (fr) 2011-07-15
US20120129864A1 (en) 2012-05-24
EP2417111A1 (fr) 2012-02-15
KR20120027212A (ko) 2012-03-21
BRPI1015951A2 (pt) 2016-04-26
AU2010233590A1 (en) 2011-11-03
SG175128A1 (en) 2011-11-28
FR2944013A1 (fr) 2010-10-08
IL215512A0 (en) 2011-12-29

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