CL2017002255A1 - Procesos para preparar fluorocetólidos. - Google Patents

Procesos para preparar fluorocetólidos.

Info

Publication number
CL2017002255A1
CL2017002255A1 CL2017002255A CL2017002255A CL2017002255A1 CL 2017002255 A1 CL2017002255 A1 CL 2017002255A1 CL 2017002255 A CL2017002255 A CL 2017002255A CL 2017002255 A CL2017002255 A CL 2017002255A CL 2017002255 A1 CL2017002255 A1 CL 2017002255A1
Authority
CL
Chile
Prior art keywords
processes
fluorocetolides
prepare
fluorocetolide
intermediates
Prior art date
Application number
CL2017002255A
Other languages
English (en)
Inventor
David Eugene Pereira
Stephen E Schneider
Keshav Deo
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of CL2017002255A1 publication Critical patent/CL2017002255A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)

Abstract

<p>En la presente, se describen procesos e intermediarios para preparar compuestos de fluorocetólido.</p>
CL2017002255A 2015-03-06 2017-09-06 Procesos para preparar fluorocetólidos. CL2017002255A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06

Publications (1)

Publication Number Publication Date
CL2017002255A1 true CL2017002255A1 (es) 2018-05-11

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2017002255A CL2017002255A1 (es) 2015-03-06 2017-09-06 Procesos para preparar fluorocetólidos.

Country Status (19)

Country Link
US (2) US20180044365A1 (es)
EP (1) EP3265100A4 (es)
JP (1) JP6773672B2 (es)
KR (1) KR20170133377A (es)
CN (1) CN107405355A (es)
AU (1) AU2016230027A1 (es)
BR (1) BR112017019176A2 (es)
CA (1) CA2978731A1 (es)
CL (1) CL2017002255A1 (es)
CO (1) CO2017010143A2 (es)
HK (1) HK1247097A1 (es)
IL (1) IL254306A0 (es)
MX (2) MX2017011454A (es)
PE (1) PE20180219A1 (es)
RU (1) RU2017131253A (es)
SG (2) SG10201908248PA (es)
TW (1) TW201638102A (es)
WO (1) WO2016144833A1 (es)
ZA (1) ZA201706505B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2008316830B2 (en) 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
CN107854477A (zh) 2008-10-24 2018-03-30 森普拉制药公司 使用含三唑的大环内酯治疗抗性疾病的方法
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
WO2013148891A1 (en) 2012-03-27 2013-10-03 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
WO2014152326A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
US7601695B2 (en) * 2003-03-10 2009-10-13 Optimer Pharmaceuticals, Inc. Antibacterial agents
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
AU2008316830B2 (en) * 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
US8376805B2 (en) * 2008-07-24 2013-02-19 Ideo Llc Printable pre-sewn stuffed toy composite sheets
CN103619849B (zh) * 2011-03-01 2016-05-25 沃克哈特有限公司 酮内酯中间体的制备方法
WO2014152326A1 (en) * 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
AU2014233240B2 (en) * 2013-03-15 2018-08-09 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
EP4095146A1 (en) * 2013-04-04 2022-11-30 President And Fellows Of Harvard College Macrolides and methods of their preparation and use

Also Published As

Publication number Publication date
CA2978731A1 (en) 2016-09-15
KR20170133377A (ko) 2017-12-05
JP6773672B2 (ja) 2020-10-21
WO2016144833A1 (en) 2016-09-15
CN107405355A (zh) 2017-11-28
CO2017010143A2 (es) 2018-02-28
US20210070797A1 (en) 2021-03-11
HK1247097A1 (zh) 2018-09-21
BR112017019176A2 (pt) 2018-04-24
TW201638102A (zh) 2016-11-01
US20180044365A1 (en) 2018-02-15
AU2016230027A1 (en) 2017-09-28
EP3265100A4 (en) 2019-01-09
EP3265100A1 (en) 2018-01-10
MX2017011454A (es) 2018-01-23
SG11201707215XA (en) 2017-10-30
JP2018508537A (ja) 2018-03-29
IL254306A0 (en) 2017-11-30
PE20180219A1 (es) 2018-01-31
MX2020007742A (es) 2020-09-25
SG10201908248PA (en) 2019-10-30
ZA201706505B (en) 2021-04-28
RU2017131253A (ru) 2019-04-08

Similar Documents

Publication Publication Date Title
CL2016002455A1 (es) Anticuerpos multiespecíficos.
CU20180001A7 (es) Derivados de oxopiridina sustituidos y procesos para su preparación
EA201891211A1 (ru) Ингибиторы cxcr2
CL2016001871A1 (es) Anticuerpos humanos para pd-1
MX2021008376A (es) Cultivo, produccion, procesamiento y uso de cannabis de especialidad.
LT3190113T (lt) Pirolopirimidino junginiai, naudotini kaip tlr7 agonistai
MX384024B (es) Peptidos macrociclicos utiles como inmunomoduladores.
LT3149032T (lt) Naujas bispecifinis formatas, tinkamas naudoti didelio našumo atrankoje
LT3126499T (lt) Kompozicijos, skirtos sod-1 ekspresijos moduliavimui
AR095075A1 (es) Acoplamiento electroquímico de anilinas
IT201600117287A1 (it) Metodo di trasfezione transiente per produzione retrovirale.
UY36737A (es) 3-amino-1,5,6,7-tetrahidro-4h-indol-4-onas
BR112016029510A2 (pt) métodos para a preparação de um composto, e, composto intermediário.
MX2017005578A (es) Métodos de administración de composiciones de amantadina.
CO2017010143A2 (es) Procesos para preparar fluorocetólidos
MX384794B (es) Proceso para la preparacion de 5-fluoro-1h-pirazoles a partir de hexafluoropropeno.
MX389099B (es) Proceso para la preparación de 3-cloro-2-vinilfenilsulfonatos.
BR112017002139A2 (pt) ?método para preparar um composto?
CL2017002653A1 (es) Procedimiento y reactor para fijar arsénico.
MX382631B (es) Proceso para la preparacion de derivados dihidroisoxazol.
MX2015011881A (es) Proceso para la preparacion de 3,7-dimetilnonan-1-ol.
LT3493849T (lt) N,n-bis-2-merkaptoetilizoftalamido naujas panaudojimas
CL2016002256A1 (es) Un proceso mejorado para la preparación de exametazima
MX380241B (es) Proceso para preparar 3-cloro-2-vinilfenol.
MX380240B (es) Preparación de piperidin-4-carbotioamida.