CL2017002813A1 - Proceso para preparar 4-amino-piridazinas - Google Patents
Proceso para preparar 4-amino-piridazinasInfo
- Publication number
- CL2017002813A1 CL2017002813A1 CL2017002813A CL2017002813A CL2017002813A1 CL 2017002813 A1 CL2017002813 A1 CL 2017002813A1 CL 2017002813 A CL2017002813 A CL 2017002813A CL 2017002813 A CL2017002813 A CL 2017002813A CL 2017002813 A1 CL2017002813 A1 CL 2017002813A1
- Authority
- CL
- Chile
- Prior art keywords
- prepare
- formula
- amino
- pyridazines
- dicloropiridazinamine
- Prior art date
Links
- LUCGBEPEAUHERV-UHFFFAOYSA-N pyridazin-4-amine Chemical class NC1=CC=NN=C1 LUCGBEPEAUHERV-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- -1 AMINO GROUP Chemical group 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/20—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B31/00—Reduction in general
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B39/00—Halogenation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B43/00—Formation or introduction of functional groups containing nitrogen
- C07B43/04—Formation or introduction of functional groups containing nitrogen of amino groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/12—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Health & Medical Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
<p>LA PRESENTE INVENCIÓN SE REFIERE A UN PROCESO PARA PREPARAR UN COMPUESTO DE PIRIDAZINAMINA DE FÓRMULA V, Y A PROCESOS PARA PREPARAR COMPUESTOS DE DICLOROPIRIDAZINAMINA DE FÓRMULA IVA, LVB, O MEZCLAS DE LAS MISMAS. ADEMÁS, LA PRESENTE INVENCIÓN SE REFIERE A LOS NUEVOS COMPUESTOS DE DICLOROPIRIDAZINAMINA DE FÓRMULA IVA, LVB, O MEZCLAS CE LAS MISMAS, EN DONDE EL GRUPO AMINO ES UN GRUPO ETILAMINO.</p>
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562159392P | 2015-05-11 | 2015-05-11 | |
| EP15169166 | 2015-05-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2017002813A1 true CL2017002813A1 (es) | 2018-05-04 |
Family
ID=53274420
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2017002813A CL2017002813A1 (es) | 2015-05-11 | 2017-11-07 | Proceso para preparar 4-amino-piridazinas |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US10584102B2 (es) |
| EP (2) | EP3872073A1 (es) |
| JP (1) | JP6833718B2 (es) |
| KR (3) | KR102919476B1 (es) |
| CN (1) | CN107592859A (es) |
| AU (1) | AU2016260784B2 (es) |
| BR (1) | BR112017023935B1 (es) |
| CA (2) | CA3187499A1 (es) |
| CL (1) | CL2017002813A1 (es) |
| CO (1) | CO2017012403A2 (es) |
| ES (1) | ES2882543T3 (es) |
| IL (1) | IL255302B (es) |
| MX (2) | MX390421B (es) |
| PE (1) | PE20180327A1 (es) |
| RU (1) | RU2742663C2 (es) |
| WO (1) | WO2016180833A1 (es) |
| ZA (1) | ZA201708142B (es) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN106573893B (zh) | 2014-07-31 | 2020-06-09 | 巴斯夫欧洲公司 | 制备吡唑的方法 |
| DK3294720T3 (da) | 2015-05-08 | 2021-02-15 | Basf Agro Bv | Fremgangsmåde til fremstilling af terpinolenepoxid |
| EP3294700B1 (en) | 2015-05-08 | 2020-01-29 | BASF Agro B.V. | A process for the preparation of limonene-4-ol |
| CA3187499A1 (en) | 2015-05-11 | 2016-11-17 | Eric George KLAUBER | Process for preparing 4-amino-pyridazines |
| CA3010561C (en) | 2016-02-02 | 2024-04-16 | Basf Se | Catalytic hydrogenation process for preparing pyrazoles |
| US10640477B2 (en) | 2016-06-15 | 2020-05-05 | BASF Agro B.V. | Process for the epoxidation of a tetrasubstituted alkene |
| MX2018015764A (es) | 2016-06-15 | 2019-08-29 | Basf Agro Bv | Proceso para la epoxidacion de un alqueno tetrasustituido. |
| EP3481795A1 (en) | 2016-07-07 | 2019-05-15 | Basf Se | Oxy-cope rearrangement for the manufacture of insecticidal cyclopentene compounds |
| US10961226B2 (en) | 2016-11-04 | 2021-03-30 | Basf Se | Process for purification of pyrazolpyridazines |
| WO2018082964A1 (en) | 2016-11-04 | 2018-05-11 | Basf Se | Process for the production of pyridazinyl-amides in a one-pot synthesis |
| EP3541788B1 (en) | 2016-11-17 | 2020-09-02 | Basf Se | Process for the purification of 1-(4-chlorophenyl)pyrazol-3-ol |
| CN110290704B (zh) | 2017-02-14 | 2022-12-06 | 巴斯夫欧洲公司 | 灭害的哒嗪吡唑酰胺类的稳定配制剂 |
| CN110431126B (zh) | 2017-03-20 | 2022-12-02 | 巴斯夫欧洲公司 | 制备一溴三氯甲烷的方法 |
| CA3122208A1 (en) * | 2019-01-11 | 2020-07-16 | Basf Se | Crystalline forms of 1-(1,2-dimethylpropyl)-n-ethyl-5-methyl-n-pyridazin-4-yl-pyrazole-4-carboxamide |
| KR20220004658A (ko) | 2019-05-03 | 2022-01-11 | 바스프 에스이 | 고도로 술폰화된 리그노술포네이트에 의한 현탁액 농축물의 안정화 |
| EP3962270B1 (en) | 2019-05-03 | 2025-07-23 | Basf Se | Stabilization of suspension concentrates by hydrophobic fumed silica |
| EP3962269B1 (en) | 2019-05-03 | 2025-07-23 | Basf Se | Stabilization of suspension concentrates by ethoxylated ricinolein |
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| US4A (en) * | 1836-08-10 | Thomas Blanchard | Stock shaving or rounding machine for edges ends etc of ships' tackle-blocks | |
| US4728355A (en) * | 1985-10-10 | 1988-03-01 | Fmc Corporation | Pyridazinylurea plant regulators |
| RU2069660C1 (ru) * | 1994-08-23 | 1996-11-27 | Акционерное общество открытого типа "Научно-исследовательский и проектный институт азотной промышленности и продуктов органического синтеза" | Способ получения производных 4-аминопиридина |
| DE4430757A1 (de) | 1994-08-30 | 1996-03-07 | Boehringer Mannheim Gmbh | Neue 4-Aminopyridazine, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel |
| TW406075B (en) * | 1994-12-13 | 2000-09-21 | Upjohn Co | Alkyl substituted piperidinyl and piperazinyl anti-AIDS compounds |
| SI9620103A (sl) * | 1995-07-06 | 1998-10-31 | Novartis Ag | Pirolopirimidini in postopki za njihovo pripravo |
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| ATE474833T1 (de) * | 2004-09-22 | 2010-08-15 | Janssen Pharmaceutica Nv | Inhibitoren der wechselwirkung zwischen mdm2 und p53 |
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| EP2346335B1 (en) | 2008-09-24 | 2018-11-14 | Basf Se | Pyrazole compounds for controlling invertebrate pests |
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| JO3407B1 (ar) | 2012-05-31 | 2019-10-20 | Eisai R&D Man Co Ltd | مركبات رباعي هيدرو بيرازولو بيريميدين |
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| EP3646731A1 (en) | 2012-06-20 | 2020-05-06 | Basf Se | Pesticidal mixtures comprising a pyrazole compound |
| WO2014063929A1 (en) * | 2012-10-23 | 2014-05-01 | Basf Se | Substituted pesticidal pyrazole compounds |
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| UA112028C2 (uk) | 2012-12-14 | 2016-07-11 | Пфайзер Лімітед | Похідні імідазопіридазину як модулятори гамка-рецептора |
| WO2015055497A1 (en) * | 2013-10-16 | 2015-04-23 | Basf Se | Substituted pesticidal pyrazole compounds |
| JP2017510550A (ja) | 2014-01-31 | 2017-04-13 | ビーエーエスエフ ソシエタス・ヨーロピアBasf Se | 無脊椎有害生物防除用ピラゾール |
| WO2015162133A1 (en) | 2014-04-22 | 2015-10-29 | Basf Se | C3-c4-cycloalkenyl-comprising pyrazoles for controlling invertebrate pests |
| WO2015169734A1 (en) | 2014-05-05 | 2015-11-12 | Basf Se | Pyrazoles for controlling invertebrate pests |
| WO2015189080A1 (en) | 2014-06-12 | 2015-12-17 | Basf Se | Pesticidally active mixtures |
| CN106573893B (zh) | 2014-07-31 | 2020-06-09 | 巴斯夫欧洲公司 | 制备吡唑的方法 |
| WO2016128239A1 (en) | 2015-02-11 | 2016-08-18 | Basf Se | Pesticidal mixture comprising a pyrazole compound and a biopesticide |
| WO2016128240A1 (en) | 2015-02-11 | 2016-08-18 | Basf Se | Pesticidal mixture comprising a pyrazole compound and two fungicides |
| WO2016128261A2 (en) | 2015-02-11 | 2016-08-18 | Basf Se | Pesticidal mixture comprising a pyrazole compound, an insecticide and a fungicide |
| CA3187499A1 (en) | 2015-05-11 | 2016-11-17 | Eric George KLAUBER | Process for preparing 4-amino-pyridazines |
| CA3010561C (en) | 2016-02-02 | 2024-04-16 | Basf Se | Catalytic hydrogenation process for preparing pyrazoles |
-
2016
- 2016-05-10 CA CA3187499A patent/CA3187499A1/en active Pending
- 2016-05-10 KR KR1020247006943A patent/KR102919476B1/ko active Active
- 2016-05-10 RU RU2017142621A patent/RU2742663C2/ru active
- 2016-05-10 KR KR1020177035243A patent/KR102585412B1/ko active Active
- 2016-05-10 EP EP21163074.4A patent/EP3872073A1/en active Pending
- 2016-05-10 WO PCT/EP2016/060461 patent/WO2016180833A1/en not_active Ceased
- 2016-05-10 US US15/572,303 patent/US10584102B2/en active Active
- 2016-05-10 CA CA2984703A patent/CA2984703C/en active Active
- 2016-05-10 PE PE2017002379A patent/PE20180327A1/es not_active Application Discontinuation
- 2016-05-10 JP JP2017557929A patent/JP6833718B2/ja active Active
- 2016-05-10 CN CN201680026456.2A patent/CN107592859A/zh active Pending
- 2016-05-10 ES ES16724331T patent/ES2882543T3/es active Active
- 2016-05-10 AU AU2016260784A patent/AU2016260784B2/en active Active
- 2016-05-10 EP EP16724331.0A patent/EP3294725B1/en active Active
- 2016-05-10 KR KR1020237033245A patent/KR102800555B1/ko active Active
- 2016-05-10 BR BR112017023935-3A patent/BR112017023935B1/pt active IP Right Grant
- 2016-05-10 MX MX2017014287A patent/MX390421B/es unknown
-
2017
- 2017-10-29 IL IL255302A patent/IL255302B/en active IP Right Grant
- 2017-11-07 CL CL2017002813A patent/CL2017002813A1/es unknown
- 2017-11-07 MX MX2021015546A patent/MX2021015546A/es unknown
- 2017-11-30 CO CONC2017/0012403A patent/CO2017012403A2/es unknown
- 2017-11-30 ZA ZA2017/08142A patent/ZA201708142B/en unknown
-
2019
- 2019-12-31 US US16/731,289 patent/US11046656B2/en active Active
-
2021
- 2021-05-18 US US17/323,337 patent/US12162841B2/en active Active
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