CL2021002911A1 - Composiciones farmacéuticas de combinación a dosis fijas de liberación inmediata, métodos y usos de las mismas - Google Patents

Composiciones farmacéuticas de combinación a dosis fijas de liberación inmediata, métodos y usos de las mismas

Info

Publication number
CL2021002911A1
CL2021002911A1 CL2021002911A CL2021002911A CL2021002911A1 CL 2021002911 A1 CL2021002911 A1 CL 2021002911A1 CL 2021002911 A CL2021002911 A CL 2021002911A CL 2021002911 A CL2021002911 A CL 2021002911A CL 2021002911 A1 CL2021002911 A1 CL 2021002911A1
Authority
CL
Chile
Prior art keywords
dose combination
methods
pharmaceutical compositions
immediate release
fixed dose
Prior art date
Application number
CL2021002911A
Other languages
English (en)
Inventor
Serra João Pedro Silva
Machuco Estevens Maria Catarina Oliveira
Marques Da Costa Ricardo Manuel Silva
Filipe Augusto Eugénio Pardal
Original Assignee
Tecnimede Sociedade Tecnico Medicinal Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=71092565&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2021002911(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tecnimede Sociedade Tecnico Medicinal Sa filed Critical Tecnimede Sociedade Tecnico Medicinal Sa
Publication of CL2021002911A1 publication Critical patent/CL2021002911A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente divulgación se refiere a una composición farmacéutica de combinación a dosis fijas de liberación inmediata que comprende los principios activos farmacéuticos memantina y donepezilo para el tratamiento de la enfermedad de Alzheimer de moderada a grave.
CL2021002911A 2019-05-31 2021-11-04 Composiciones farmacéuticas de combinación a dosis fijas de liberación inmediata, métodos y usos de las mismas CL2021002911A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PT11555719 2019-05-31

Publications (1)

Publication Number Publication Date
CL2021002911A1 true CL2021002911A1 (es) 2022-07-15

Family

ID=71092565

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2021002911A CL2021002911A1 (es) 2019-05-31 2021-11-04 Composiciones farmacéuticas de combinación a dosis fijas de liberación inmediata, métodos y usos de las mismas

Country Status (15)

Country Link
EP (2) EP4238555A3 (es)
BR (1) BR112021024054A2 (es)
CL (1) CL2021002911A1 (es)
CO (1) CO2021014967A2 (es)
DK (1) DK3843702T3 (es)
FI (1) FI3843702T3 (es)
HR (1) HRP20231200T1 (es)
IL (1) IL288505A (es)
MX (2) MX2021014673A (es)
PE (1) PE20220936A1 (es)
PT (1) PT3843702T (es)
SA (1) SA521430969B1 (es)
SI (1) SI3843702T1 (es)
WO (1) WO2020240505A1 (es)
ZA (2) ZA202110478B (es)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI95572C (fi) 1987-06-22 1996-02-26 Eisai Co Ltd Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi
ES2059602T3 (es) 1989-04-14 1994-11-16 Merz & Co Gmbh & Co Uso de derivados de adamantano para la prevencion y tratamiento de isquemia cerebral.
WO1997046526A1 (en) 1996-06-07 1997-12-11 Eisai Co., Ltd. Stable polymorphs of donepezil (1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl]methylpiperidine) hydrochloride and process for production
PT1509232E (pt) 2002-05-31 2009-01-07 Lundbeck & Co As H Uma combinação de um antagonista de nmda e inibidores da acetilcolina esterase para o tratamento da doença de alzheimer
TW200418446A (en) 2002-10-24 2004-10-01 Merz Pharma Gmbh & Co Kgaa Combination therapy using 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors
JP5025468B2 (ja) * 2004-06-17 2012-09-12 メルツ・ファルマ・ゲゼルシヤフト・ミト・ベシュレンクテル・ハフツング・ウント・コンパニー・コマンデイトゲゼルシヤフト・アウフ・アクティーン メマンチン又はネラメキサンの直接圧縮によって製造された、飲用に適した即効型錠剤
WO2006076562A1 (en) 2005-01-11 2006-07-20 Teva Pharmaceutical Fine Chemicals S.R.L. Process for the preparation of 1-amino-3,5-dimethyladamantane hydrochloride
ATE481096T1 (de) 2005-04-06 2010-10-15 Adamas Pharmaceuticals Inc Verfahren und zusammensetzungen zur behandlung von zns-erkrankungen
CN101166543B (zh) * 2005-04-28 2014-07-16 卫材R&D管理有限公司 含抗痴呆药物的组合物
DE102005060377A1 (de) * 2005-12-16 2007-06-21 Ratiopharm Gmbh Pharmazeutische Zusammensetzung enthaltend Donepezilhydrochlorid, Tablette hieraus und Verfahren zu deren Herstellung
CN105816441A (zh) * 2016-05-31 2016-08-03 北京康立生医药技术开发有限公司 盐酸美金刚多奈哌齐复方制剂
KR101938872B1 (ko) * 2016-09-30 2019-01-16 주식회사 바이오파마티스 도네페질 또는 그의 약학적으로 허용 가능한 염 및 메만틴 또는 그의 약학적으로 허용 가능한 염을 함유하는 치매 및 인지기능 장애 예방 또는 치료용 약학 조성물 및 이의 제조방법
WO2018062941A1 (ko) * 2016-09-30 2018-04-05 주식회사 바이오파마티스 도네페질 또는 그의 약학적으로 허용 가능한 염 및 메만틴 또는 그의 약학적으로 허용 가능한 염을 함유하는 치매 및 인지기능 장애 예방 또는 치료용 약학 조성물 및 이의 제조방법

Also Published As

Publication number Publication date
MX2025002148A (es) 2025-04-02
MX2021014673A (es) 2022-01-11
DK3843702T3 (da) 2023-10-09
HRP20231200T1 (hr) 2024-01-19
BR112021024054A2 (pt) 2022-01-11
EP4238555A2 (en) 2023-09-06
IL288505A (en) 2022-01-01
CO2021014967A2 (es) 2021-11-19
PE20220936A1 (es) 2022-05-31
FI3843702T3 (fi) 2023-10-09
SA521430969B1 (ar) 2023-12-05
ZA202311560B (en) 2024-07-31
EP3843702A1 (en) 2021-07-07
EP4238555A3 (en) 2023-09-20
SI3843702T1 (sl) 2023-12-29
EP3843702B1 (en) 2023-07-05
ZA202110478B (en) 2024-08-28
WO2020240505A1 (en) 2020-12-03
PT3843702T (pt) 2023-10-13

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