CN1243748C - 醇的甲氨酰化方法 - Google Patents

醇的甲氨酰化方法 Download PDF

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Publication number
CN1243748C
CN1243748C CNB028042816A CN02804281A CN1243748C CN 1243748 C CN1243748 C CN 1243748C CN B028042816 A CNB028042816 A CN B028042816A CN 02804281 A CN02804281 A CN 02804281A CN 1243748 C CN1243748 C CN 1243748C
Authority
CN
China
Prior art keywords
alcohol
cyanate
reaction
capravirine
methanesulfonic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CNB028042816A
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English (en)
Chinese (zh)
Other versions
CN1489584A (zh
Inventor
詹姆斯·E·埃利斯
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Warner Lambert Co LLC
Original Assignee
Warner Lambert Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co LLC filed Critical Warner Lambert Co LLC
Publication of CN1489584A publication Critical patent/CN1489584A/zh
Application granted granted Critical
Publication of CN1243748C publication Critical patent/CN1243748C/zh
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
CNB028042816A 2001-01-31 2002-01-11 醇的甲氨酰化方法 Expired - Fee Related CN1243748C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26550201P 2001-01-31 2001-01-31
US60/265,502 2001-01-31

Publications (2)

Publication Number Publication Date
CN1489584A CN1489584A (zh) 2004-04-14
CN1243748C true CN1243748C (zh) 2006-03-01

Family

ID=23010706

Family Applications (1)

Application Number Title Priority Date Filing Date
CNB028042816A Expired - Fee Related CN1243748C (zh) 2001-01-31 2002-01-11 醇的甲氨酰化方法

Country Status (18)

Country Link
US (1) US6613908B2 (cs)
EP (1) EP1377568A1 (cs)
JP (1) JP2004518687A (cs)
KR (1) KR100567706B1 (cs)
CN (1) CN1243748C (cs)
AR (1) AR032419A1 (cs)
BR (1) BR0206806A (cs)
CA (1) CA2433364A1 (cs)
CZ (1) CZ20032001A3 (cs)
HU (1) HUP0303028A3 (cs)
IL (1) IL156363A0 (cs)
MX (1) MXPA03005403A (cs)
PL (1) PL363321A1 (cs)
RU (1) RU2256657C2 (cs)
TW (1) TWI228507B (cs)
WO (1) WO2002060893A1 (cs)
YU (1) YU52303A (cs)
ZA (1) ZA200304687B (cs)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL1628685T3 (pl) 2003-04-25 2011-05-31 Gilead Sciences Inc Przeciwwirusowe analogi fosfonianowe
EP1656387A2 (en) * 2003-07-30 2006-05-17 Gilead Sciences, Inc. Nucleobase phosphonate analogs for antiviral treatment
WO2005016912A1 (en) * 2003-08-19 2005-02-24 Pfizer Inc. An efficient microbial preparation of capravirine metabolites m4 and m5
US20050080268A1 (en) * 2003-10-08 2005-04-14 Yong-Moon Choi Process of preparing O-carbamoyl compounds in the presence of active amine group
DK1778702T3 (da) * 2004-07-16 2011-10-17 Gilead Sciences Inc Antivirale forbindelser
EP1778251B1 (en) 2004-07-27 2011-04-13 Gilead Sciences, Inc. Nucleoside phosphonate conjugates as anti hiv agents
TW200738742A (en) * 2005-07-14 2007-10-16 Gilead Sciences Inc Antiviral compounds
TWI389908B (zh) * 2005-07-14 2013-03-21 Gilead Sciences Inc 抗病毒化合物類
US20080076740A1 (en) * 2005-07-27 2008-03-27 Gilead Sciences, Inc. Antiviral compounds
WO2008005542A2 (en) * 2006-07-07 2008-01-10 Gilead Sciences, Inc., Antiviral phosphinate compounds
AU2009268681B2 (en) * 2008-07-08 2014-10-02 Gilead Sciences, Inc. Salts of HIV inhibitor compounds
US8810796B2 (en) 2009-04-21 2014-08-19 Michigan Aerospace Corporation Light processing system and method
EP3661937B1 (en) 2017-08-01 2021-07-28 Gilead Sciences, Inc. Crystalline forms of ethyl ((s)-((((2r,5r)-5-(6-amino-9h-purin-9-yl)-4-fluoro-2,5-dihydrofuran-2-yl)oxy)methyl)(phenoxy)phosphoryl)-l-alaninate (gs-9131) for treating viral infections

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2611695A1 (de) * 1976-03-19 1977-09-29 Hoechst Ag Herbizide mittel
DE69532245T2 (de) 1994-09-26 2004-09-16 Shionogi & Co., Ltd. Imidazolderivat

Also Published As

Publication number Publication date
HUP0303028A3 (en) 2005-10-28
RU2003123791A (ru) 2005-02-27
CN1489584A (zh) 2004-04-14
PL363321A1 (en) 2004-11-15
CZ20032001A3 (en) 2004-06-16
IL156363A0 (en) 2004-01-04
HUP0303028A2 (hu) 2003-12-29
BR0206806A (pt) 2004-02-03
US6613908B2 (en) 2003-09-02
US20020103378A1 (en) 2002-08-01
AR032419A1 (es) 2003-11-05
KR100567706B1 (ko) 2006-04-05
WO2002060893A1 (en) 2002-08-08
KR20030069227A (ko) 2003-08-25
RU2256657C2 (ru) 2005-07-20
MXPA03005403A (es) 2003-09-25
HK1060573A1 (en) 2004-08-13
YU52303A (sh) 2006-05-25
EP1377568A1 (en) 2004-01-07
CA2433364A1 (en) 2002-08-08
TWI228507B (en) 2005-03-01
ZA200304687B (en) 2004-08-10
JP2004518687A (ja) 2004-06-24

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