CR10164A - Uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de obesidad - Google Patents

Uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de obesidad

Info

Publication number
CR10164A
CR10164A CR10164A CR10164A CR10164A CR 10164 A CR10164 A CR 10164A CR 10164 A CR10164 A CR 10164A CR 10164 A CR10164 A CR 10164A CR 10164 A CR10164 A CR 10164A
Authority
CR
Costa Rica
Prior art keywords
benzo
heterociclic
fusion
sulfamide derivatives
obesity treatment
Prior art date
Application number
CR10164A
Other languages
English (en)
Inventor
L Smith-Swintosky Virginia
B Reitz Allen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CR10164A publication Critical patent/CR10164A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Pyrane Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención es un método para el tratamiento de obesidad, para promover la pérdida de peso y/o suprimir el apetito que comprende la administración a un sujeto que lo necesita de una cantidad terapéuticamente efectiva de uno o más derivados de sulfamida heterocíclica benzo-fusionada novedosos de fórmula (i) como se definen aquí.
CR10164A 2005-12-19 2008-07-21 Uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de obesidad CR10164A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75149905P 2005-12-19 2005-12-19
US11/611,938 US8492431B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of obesity

Publications (1)

Publication Number Publication Date
CR10164A true CR10164A (es) 2009-01-14

Family

ID=37992995

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10164A CR10164A (es) 2005-12-19 2008-07-21 Uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de obesidad

Country Status (30)

Country Link
US (1) US8492431B2 (es)
EP (1) EP1968574B9 (es)
JP (1) JP5190378B2 (es)
KR (1) KR101363308B1 (es)
CN (1) CN101365442B (es)
AR (1) AR058389A1 (es)
AT (1) ATE519484T1 (es)
AU (1) AU2006331637B2 (es)
BR (1) BRPI0620019A2 (es)
CA (1) CA2634093C (es)
CR (1) CR10164A (es)
CY (1) CY1112357T1 (es)
DK (1) DK1968574T3 (es)
EA (1) EA016560B1 (es)
ES (1) ES2369761T3 (es)
HR (1) HRP20110726T2 (es)
IL (1) IL192107A (es)
ME (1) ME01344B (es)
MY (1) MY145823A (es)
NO (1) NO20083006L (es)
NZ (1) NZ568960A (es)
PE (1) PE20070813A1 (es)
PL (1) PL1968574T3 (es)
PT (1) PT1968574E (es)
RS (1) RS52044B (es)
SI (1) SI1968574T1 (es)
SV (1) SV2008002952A (es)
UY (1) UY30033A1 (es)
WO (1) WO2007075833A2 (es)
ZA (1) ZA200806279B (es)

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US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US8492431B2 (en) 2005-12-19 2013-07-23 Janssen Pharmaceutica, N.V. Use of benzo-fused heterocycle sulfamide derivatives for the treatment of obesity
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EA018567B1 (ru) 2008-06-23 2013-08-30 Янссен Фармацевтика Нв Кристаллическая форма (2s)-(-)-n-(6-хлор-2,3-дигидробензо[1,4]диоксин-2-илметил)сульфамида
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
JP2014528953A (ja) 2011-09-29 2014-10-30 ヤンセン ファーマシューティカ エヌ．ベー． スルファミド誘導体の調製プロセス
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EA018567B1 (ru) * 2008-06-23 2013-08-30 Янссен Фармацевтика Нв Кристаллическая форма (2s)-(-)-n-(6-хлор-2,3-дигидробензо[1,4]диоксин-2-илметил)сульфамида

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