CR10404A - Composicion farmaceutica de liberacion sostenida sobre la base de un sistema de liberacion que comprende un polimero acido-soluble y un polimero ph-dependiente - Google Patents

Composicion farmaceutica de liberacion sostenida sobre la base de un sistema de liberacion que comprende un polimero acido-soluble y un polimero ph-dependiente

Info

Publication number
CR10404A
CR10404A CR10404A CR10404A CR10404A CR 10404 A CR10404 A CR 10404A CR 10404 A CR10404 A CR 10404A CR 10404 A CR10404 A CR 10404A CR 10404 A CR10404 A CR 10404A
Authority
CR
Costa Rica
Prior art keywords
liberation
polymer
acid
basis
pharmaceutical composition
Prior art date
Application number
CR10404A
Other languages
English (en)
Inventor
Rajesh Jain
Kour Chand Jindal
Sampath Kumar Devarajan
Original Assignee
Panacea Biotec Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Panacea Biotec Ltd filed Critical Panacea Biotec Ltd
Publication of CR10404A publication Critical patent/CR10404A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se describen composiciones farmaceuticas de liberacion sostenida que comprenden por lo menos un agente activo escasamente soluble, por lo menos un solubilizante, un sistema polimerico controlador de velocidad de liberacion que consiste en un polimero soluble en acido y un polimero dependiente del pH, y opcionalmente otros excipientes farmaceuticamente aceptables; la presente invencion tambien describe un procedimiento para preparar tales composiciones y metodos de uso de las mismas; las composiciones de liberacion sostenida son utiles para proveer concentraciones terapeuticamente efectivas de los agentes activos durante periodos prolongados.
CR10404A 2006-03-27 2008-10-27 Composicion farmaceutica de liberacion sostenida sobre la base de un sistema de liberacion que comprende un polimero acido-soluble y un polimero ph-dependiente CR10404A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN832DE2006 2006-03-27

Publications (1)

Publication Number Publication Date
CR10404A true CR10404A (es) 2008-12-08

Family

ID=38540835

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10404A CR10404A (es) 2006-03-27 2008-10-27 Composicion farmaceutica de liberacion sostenida sobre la base de un sistema de liberacion que comprende un polimero acido-soluble y un polimero ph-dependiente

Country Status (14)

Country Link
US (1) US20100234288A1 (es)
EP (1) EP2004150A1 (es)
JP (1) JP2009531420A (es)
CN (1) CN101410096A (es)
AU (1) AU2007230549A1 (es)
BR (1) BRPI0709222A2 (es)
CA (1) CA2647421A1 (es)
CR (1) CR10404A (es)
EA (1) EA200870379A1 (es)
MA (1) MA30359B1 (es)
MX (1) MX2008012486A (es)
RS (1) RS20080439A (es)
TN (1) TNSN08365A1 (es)
WO (1) WO2007110878A1 (es)

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CA2733611A1 (en) * 2008-08-11 2010-02-18 Ratiopharm Gmbh Pharmaceutical compositions with modified release properties comprising 5-chloro-n-({(5s)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
CN101361979B (zh) * 2008-09-19 2011-01-19 天津博科林药品包装技术有限公司 一种固体制剂薄膜包衣剂及其制备方法
WO2010082855A1 (en) * 2009-01-15 2010-07-22 Zaklady Farmaceutyczne Polpharma Sa Pharmaceutical compositions comprising ziprasidone free base or ziprasidone hydrochloride and the method for their preparation
US9138309B2 (en) 2010-02-05 2015-09-22 Allergan, Inc. Porous materials, methods of making and uses
US9205577B2 (en) * 2010-02-05 2015-12-08 Allergan, Inc. Porogen compositions, methods of making and uses
WO2011103718A1 (zh) * 2010-02-26 2011-09-01 上海沪美医药科技有限公司 一种含有喹硫平的控(缓)释制剂及其制备方法和用途
US11202853B2 (en) * 2010-05-11 2021-12-21 Allergan, Inc. Porogen compositions, methods of making and uses
MX2013001637A (es) * 2010-08-10 2014-06-23 Lupin Ltd Composiciones farmaceuticas de liberacion controlada oral de blonanserina.
HUE051133T2 (hu) * 2010-11-01 2021-03-01 Melinta Subsidiary Corp Gyógyászati készítmények
CN102058517A (zh) * 2010-12-31 2011-05-18 泰州万全医药科技有限公司 一种帕潘立酮缓释剂及其制备方法
US20150174247A1 (en) * 2012-06-29 2015-06-25 Maruishi Pharmaceutical Co., Ltd. Oral pharmaceutical preparation of aripiprazole
TWI722988B (zh) * 2015-06-05 2021-04-01 瑩碩生技醫藥股份有限公司 緩釋性醫藥組合物及其製備方法
CN105199115B (zh) * 2015-10-27 2021-01-12 中国林业科学研究院林产化学工业研究所 一种多孔渗水的三维网状结构的可注射水凝胶的制备及其应用
WO2017218772A1 (en) * 2016-06-17 2017-12-21 The Procter & Gamble Company Delayed-release particles
CN108203508A (zh) * 2016-12-16 2018-06-26 中国石油化工股份有限公司 一种改性尼龙6材料及其制备方法
CA3047354A1 (en) 2016-12-20 2018-06-28 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system containing asenapine and polysiloxane or polyisobutylene
RU2762896C2 (ru) 2016-12-20 2021-12-23 Лтс Ломанн Терапи-Систем Аг Трансдермальная терапевтическая система, содержащая азенапин
KR101813835B1 (ko) * 2017-02-17 2017-12-29 이충근 피이지 프리 가용화제 및 이의 제조방법
CN107028903B (zh) * 2017-05-03 2020-03-10 深圳万和制药有限公司 布南色林片剂药物组合物及其制备方法
EP3644973B1 (en) 2017-06-26 2021-03-24 LTS LOHMANN Therapie-Systeme AG Transdermal therapeutic system containing asenapine and silicone acrylic hybrid polymer
MX2020005517A (es) 2017-12-05 2020-11-09 Sunovion Pharmaceuticals Inc Formas cristalinas y metodos de produccion de las mismas.
US10369134B2 (en) 2017-12-05 2019-08-06 Sunovion Pharmaceuticals Inc. Nonracemic mixtures and uses thereof
US11672781B2 (en) 2018-05-07 2023-06-13 Prana Biosciences Inc Metaxalone formulations
CN110958876B (zh) 2018-06-20 2020-12-18 罗曼治疗系统股份公司 含有阿塞那平的透皮治疗系统
CN112533593A (zh) 2018-06-20 2021-03-19 罗曼治疗系统股份公司 含有阿塞那平的透皮治疗系统
EP3897728A1 (en) * 2018-12-18 2021-10-27 DDP Specialty Electronic Materials US, Inc. A sustained release composition comprising a hydroxyalkyl methylcellulose
CN109984999B (zh) * 2019-04-28 2021-12-24 重庆仁泽医药科技有限公司 一种药物组合物及其制备方法和用途
WO2020247627A1 (en) 2019-06-04 2020-12-10 Sunovion Pharmaceuticals Inc. Modified release formulations and uses thereof
CN111568856B (zh) * 2020-06-24 2021-07-06 珠海舒桐医疗科技有限公司 一种阴道凝胶制剂及其制备方法
EP4456887A4 (en) * 2021-12-30 2025-12-17 Neuropro Therapeutics Inc PHARMACEUTICAL COMPOSITION

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US20030180352A1 (en) * 1999-11-23 2003-09-25 Patel Mahesh V. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
KR100694667B1 (ko) * 1999-12-08 2007-03-14 동아제약주식회사 생체내이용률 향상과 개인간 및 개인내 흡수 편차를감소시킨 이트라코나졸 함유 항진균성 제제
ES2333645T3 (es) * 2001-06-22 2010-02-25 Bend Research, Inc. Composiciones farmaceuticas de dispersiones de medicamentos y polimeros neutros.
US20050096365A1 (en) * 2003-11-03 2005-05-05 David Fikstad Pharmaceutical compositions with synchronized solubilizer release

Also Published As

Publication number Publication date
MA30359B1 (fr) 2009-04-01
RS20080439A (sr) 2009-05-06
JP2009531420A (ja) 2009-09-03
BRPI0709222A2 (pt) 2011-07-12
EP2004150A1 (en) 2008-12-24
CN101410096A (zh) 2009-04-15
US20100234288A1 (en) 2010-09-16
AU2007230549A1 (en) 2007-10-04
WO2007110878A1 (en) 2007-10-04
EA200870379A1 (ru) 2009-04-28
TNSN08365A1 (en) 2009-12-29
MX2008012486A (es) 2008-10-10
CA2647421A1 (en) 2007-10-04

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