CR11248A - Compuestos anti-virales, composiciones y metodos de uso - Google Patents

Compuestos anti-virales, composiciones y metodos de uso

Info

Publication number
CR11248A
CR11248A CR11248A CR11248A CR11248A CR 11248 A CR11248 A CR 11248A CR 11248 A CR11248 A CR 11248A CR 11248 A CR11248 A CR 11248A CR 11248 A CR11248 A CR 11248A
Authority
CR
Costa Rica
Prior art keywords
compositions
methods
viral compounds
compounds
virus
Prior art date
Application number
CR11248A
Other languages
English (en)
Inventor
Martin Robert Leivers
Jesse Daniel Keicher
Franz Ulrich Schmitz
Roopa Rai
Ryan Lauchli
Sebastian Reinhard Johannes Liehr
Stephanie Anna Chan
Toney Loc Ton
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of CR11248A publication Critical patent/CR11248A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se dan a conocer compuestos de la Formula (I): sales farmaceuticamente aceptables, y solvatos de los mismos, composiciones de los mismos, y metodos para su preparacion y uso para el tratamiento de infecciones virales mediadas cuando menos en parte por un virus de la familia de virus Flaviviridae.
CR11248A 2007-07-13 2010-02-02 Compuestos anti-virales, composiciones y metodos de uso CR11248A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US94975807P 2007-07-13 2007-07-13

Publications (1)

Publication Number Publication Date
CR11248A true CR11248A (es) 2010-10-05

Family

ID=39929680

Family Applications (1)

Application Number Title Priority Date Filing Date
CR11248A CR11248A (es) 2007-07-13 2010-02-02 Compuestos anti-virales, composiciones y metodos de uso

Country Status (13)

Country Link
US (2) US20110044943A1 (es)
EP (1) EP2178877A1 (es)
JP (1) JP2010533183A (es)
KR (1) KR20100056462A (es)
AU (1) AU2008276611A1 (es)
BR (1) BRPI0814300A2 (es)
CA (1) CA2693793A1 (es)
CR (1) CR11248A (es)
EA (1) EA201000051A1 (es)
MA (1) MA31598B1 (es)
TW (1) TW200920372A (es)
WO (1) WO2009011787A1 (es)
ZA (1) ZA201000992B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1838152A2 (en) * 2005-01-21 2007-10-03 Neurogen Corporation Imidazolylmethyl and pyrazolylmethyl heteroaryl derivatives
JP2010519174A (ja) * 2006-09-18 2010-06-03 バーテックス ファーマシューティカルズ インコーポレイテッド c−Metの複素環阻害薬およびその使用方法
UY31685A (es) * 2008-03-04 2009-11-10 Smithkline Beecham Corp Compuestos antivirales, composiciones y metodos para usarlos
KR101220182B1 (ko) 2009-02-25 2013-01-11 에스케이바이오팜 주식회사 치환된 아졸 유도체 화합물, 이를 포함하는 약제학적 조성물 및 이를 이용한 파킨슨씨 병 치료방법
US20110053892A1 (en) * 2009-08-31 2011-03-03 Martin Leivers Imidazo[4,5-d]Pyridazine Compounds For Treating Viral Infections
EP2545964A1 (en) 2011-07-13 2013-01-16 Phenex Pharmaceuticals AG Novel FXR (NR1H4) binding and activity modulating compounds
CA2968836C (en) 2016-06-13 2025-09-02 Gilead Sciences, Inc. FXR MODULATING COMPOUNDS (NR1H4)
NZ748641A (en) 2016-06-13 2020-04-24 Gilead Sciences Inc Fxr (nr1h4) modulating compounds
WO2018165520A1 (en) 2017-03-10 2018-09-13 Vps-3, Inc. Metalloenzyme inhibitor compounds
SI4122464T1 (sl) 2017-03-28 2024-07-31 Gilead Sciences, Inc. Terapevtske kombinacije za zdravljenje bolezni jeter
PT3911647T (pt) 2019-01-15 2024-03-04 Gilead Sciences Inc Composto de isoxazole como agonista de fxr e composições farmacêuticas que o contenham
JP2022519906A (ja) 2019-02-19 2022-03-25 ギリアード サイエンシーズ, インコーポレイテッド Fxrアゴニストの固体形態
AU2020321955A1 (en) 2019-07-30 2022-03-17 Eikonizo Therapapeutics, Inc. HDAC6 inhibitors and uses thereof
TW202345813A (zh) 2022-04-08 2023-12-01 美商艾科尼佐療法股份有限公司 㗁二唑hdac6抑制劑及其用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2161273B1 (en) * 2003-12-22 2015-04-15 K.U.Leuven Research & Development Imidazo[4,5-c]pyridine compounds and methods of antiviral treatment
BRPI0513811A (pt) * 2004-07-27 2008-07-15 Gilead Sciences Inc imidazo [4,5-d] pirimidinas, seus usos e processos de preparação
AU2005286790A1 (en) * 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Bicyclic heterocyclic derivatives and their use as inhibitors of stearoyl-CoA-desaturase (SCD)
NZ556624A (en) * 2004-12-21 2010-06-25 Gilead Sciences Inc 5-((3-(2,4-trifluoromethyphenyl)isoxazol-5-yl)methyl)-2-(2-fluorophenyl)-5H-imidazo[4,5-c]pyridine and method of antiviral treatment
FR2909090B1 (fr) * 2006-11-23 2009-01-09 Sanofi Aventis Sa Derives de 2,5-dihydro-3h-pyrazolo[4,3-c]pyridazin-3-one substitues,leur preparation et leur application en therapeutique.
US20110053892A1 (en) * 2009-08-31 2011-03-03 Martin Leivers Imidazo[4,5-d]Pyridazine Compounds For Treating Viral Infections

Also Published As

Publication number Publication date
TW200920372A (en) 2009-05-16
JP2010533183A (ja) 2010-10-21
WO2009011787A1 (en) 2009-01-22
ZA201000992B (en) 2011-04-28
MA31598B1 (fr) 2010-08-02
US20090074717A1 (en) 2009-03-19
KR20100056462A (ko) 2010-05-27
CA2693793A1 (en) 2009-01-22
AU2008276611A1 (en) 2009-01-22
EP2178877A1 (en) 2010-04-28
BRPI0814300A2 (pt) 2015-02-03
EA201000051A1 (ru) 2010-08-30
US20110044943A1 (en) 2011-02-24

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)