CR20120032A - Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituida-n1 - Google Patents

Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituida-n1

Info

Publication number
CR20120032A
CR20120032A CR20120032A CR20120032A CR20120032A CR 20120032 A CR20120032 A CR 20120032A CR 20120032 A CR20120032 A CR 20120032A CR 20120032 A CR20120032 A CR 20120032A CR 20120032 A CR20120032 A CR 20120032A
Authority
CR
Costa Rica
Prior art keywords
fluoro
derivatives
substituida
oxopirimidinona
carboxamida
Prior art date
Application number
CR20120032A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR20120032(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of CR20120032A publication Critical patent/CR20120032A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente descripción se relaciona con el campo de las 5-fluoro-2-oxopirimidinona-1-(2H)-carboxamidas substituidas-N1 y sus derivados y el uso de estos compuestos como fungicidas.
CR20120032A 2009-08-07 2012-01-18 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituida-n1 CR20120032A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
CR20120032A true CR20120032A (es) 2012-03-22

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20120032A CR20120032A (es) 2009-08-07 2012-01-18 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituida-n1

Country Status (26)

Country Link
US (2) US8552020B2 (es)
EP (1) EP2461686B1 (es)
JP (1) JP5735510B2 (es)
KR (1) KR101792284B1 (es)
CN (1) CN102497781B (es)
BR (1) BR112012002757B1 (es)
CA (1) CA2769656C (es)
CL (1) CL2012000312A1 (es)
CO (1) CO6491115A2 (es)
CR (1) CR20120032A (es)
DK (1) DK2461686T3 (es)
EA (1) EA020910B1 (es)
EC (1) ECSP12011652A (es)
ES (1) ES2552097T3 (es)
HU (1) HUE027390T2 (es)
IL (1) IL217950A (es)
IN (1) IN2012DN00369A (es)
MX (1) MX2012001617A (es)
NI (1) NI201200021A (es)
NZ (1) NZ597483A (es)
PE (1) PE20120692A1 (es)
PL (1) PL2461686T3 (es)
PT (1) PT2461686E (es)
UA (1) UA107671C2 (es)
WO (1) WO2011017545A1 (es)
ZA (1) ZA201200813B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2461688B1 (en) 2009-08-07 2016-03-16 Dow AgroSciences LLC Pesticidal compositions
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
MX2012001622A (es) * 2009-08-07 2012-04-11 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona.
JP6336480B2 (ja) * 2012-12-28 2018-06-06 アダマ・マクテシム・リミテッド １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体
MX2015008444A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.
AU2013370493B2 (en) * 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
KR102309245B1 (ko) 2012-12-31 2021-10-06 아다마 마켓심 리미티드 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
FI3096619T3 (fi) 2013-12-31 2025-09-03 Adama Makhteshim Ltd Synergistisiä sienituhoaineseoksia sienten torjuntaan viljakasveissa
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
US12414559B2 (en) 2018-11-05 2025-09-16 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
WO2021059160A1 (en) 2019-09-23 2021-04-01 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
US20230045196A1 (en) * 2019-12-10 2023-02-09 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of peanut plants by phytopathogenic microorganisms

Family Cites Families (24)

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US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (es) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
JPS60123486A (ja) * 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンｓおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
DE58908159D1 (de) 1988-03-09 1994-09-15 Ciba Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
DE69618959T2 (de) * 1995-07-05 2002-08-29 E.I. Du Pont De Nemours And Co., Wilmington Pyrimidone und ihre verwendug als fungizide
US6262058B1 (en) 1996-03-11 2001-07-17 Syngenta Crop Protection, Inc. Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
US20080269238A1 (en) * 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
ES2549379T3 (es) * 2008-01-22 2015-10-27 Dow Agrosciences Llc Derivados de 4-amino5-fluoropirimidina como fungicidas
PL2317851T3 (pl) * 2008-08-01 2014-06-30 Dow Agrosciences Llc Zastosowanie 5-fluorocytozyny jako fungicydu
DK2389375T3 (en) * 2009-01-23 2015-08-24 Euro Celtique Sa Hydroxamsyrederivater
MX2012001622A (es) * 2009-08-07 2012-04-11 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona.
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Also Published As

Publication number Publication date
US9000002B2 (en) 2015-04-07
EP2461686B1 (en) 2015-10-07
US20140011824A1 (en) 2014-01-09
NI201200021A (es) 2012-05-22
JP5735510B2 (ja) 2015-06-17
CL2012000312A1 (es) 2012-10-05
ECSP12011652A (es) 2012-03-30
IN2012DN00369A (es) 2015-08-21
WO2011017545A1 (en) 2011-02-10
US8552020B2 (en) 2013-10-08
CA2769656C (en) 2018-05-15
KR101792284B1 (ko) 2017-10-31
BR112012002757B1 (pt) 2020-10-06
DK2461686T3 (en) 2016-01-18
BR112012002757A2 (pt) 2019-12-17
KR20120052281A (ko) 2012-05-23
IL217950A0 (en) 2012-03-29
UA107671C2 (en) 2015-02-10
PE20120692A1 (es) 2012-06-08
ES2552097T3 (es) 2015-11-25
CN102497781A (zh) 2012-06-13
CO6491115A2 (es) 2012-07-31
NZ597483A (en) 2014-02-28
CN102497781B (zh) 2014-12-10
EA020910B1 (ru) 2015-02-27
ZA201200813B (en) 2013-05-29
HK1171915A1 (en) 2013-04-12
PT2461686E (pt) 2015-11-18
EP2461686A4 (en) 2013-02-13
JP2013501727A (ja) 2013-01-17
AU2010279409A1 (en) 2012-02-02
HUE027390T2 (en) 2016-10-28
MX2012001617A (es) 2012-04-11
PL2461686T3 (pl) 2016-04-29
IL217950A (en) 2015-04-30
EP2461686A1 (en) 2012-06-13
EA201270256A1 (ru) 2012-07-30
US20110034492A1 (en) 2011-02-10
CA2769656A1 (en) 2011-02-10

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