CR20150442A - Cabazitaxel y su uso para el tratamiento de los cánceres de próstata metastásicos - Google Patents
Cabazitaxel y su uso para el tratamiento de los cánceres de próstata metastásicosInfo
- Publication number
- CR20150442A CR20150442A CR20150442A CR20150442A CR20150442A CR 20150442 A CR20150442 A CR 20150442A CR 20150442 A CR20150442 A CR 20150442A CR 20150442 A CR20150442 A CR 20150442A CR 20150442 A CR20150442 A CR 20150442A
- Authority
- CR
- Costa Rica
- Prior art keywords
- treatment
- prostate cancer
- metastastic
- cabazitaxel
- resistant
- Prior art date
Links
- 206010060862 Prostate cancer Diseases 0.000 title 1
- 208000000236 Prostatic Neoplasms Diseases 0.000 title 1
- BMQGVNUXMIRLCK-OAGWZNDDSA-N cabazitaxel Chemical compound O([C@H]1[C@@H]2[C@]3(OC(C)=O)CO[C@@H]3C[C@@H]([C@]2(C(=O)[C@H](OC)C2=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)C=3C=CC=CC=3)C[C@]1(O)C2(C)C)C)OC)C(=O)C1=CC=CC=C1 BMQGVNUXMIRLCK-OAGWZNDDSA-N 0.000 title 1
- 229960001573 cabazitaxel Drugs 0.000 title 1
- 230000001394 metastastic effect Effects 0.000 title 1
- 208000007882 Gastritis Diseases 0.000 abstract 1
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 208000012671 Gastrointestinal haemorrhages Diseases 0.000 abstract 1
- 206010018001 Gastrointestinal perforation Diseases 0.000 abstract 1
- 208000003011 Neutropenic Enterocolitis Diseases 0.000 abstract 1
- 206010062959 Neutropenic colitis Diseases 0.000 abstract 1
- 206010036909 Prostate cancer metastatic Diseases 0.000 abstract 1
- 206010009887 colitis Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000010227 enterocolitis Diseases 0.000 abstract 1
- 208000030304 gastrointestinal bleeding Diseases 0.000 abstract 1
- 230000003054 hormonal effect Effects 0.000 abstract 1
- 210000003405 ileum Anatomy 0.000 abstract 1
- 208000003243 intestinal obstruction Diseases 0.000 abstract 1
- 208000010658 metastatic prostate carcinoma Diseases 0.000 abstract 1
- 229960005205 prednisolone Drugs 0.000 abstract 1
- OIGNJSKKLXVSLS-VWUMJDOOSA-N prednisolone Chemical compound O=C1C=C[C@]2(C)[C@H]3[C@@H](O)C[C@](C)([C@@](CC4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 OIGNJSKKLXVSLS-VWUMJDOOSA-N 0.000 abstract 1
- 229960004618 prednisone Drugs 0.000 abstract 1
- XOFYZVNMUHMLCC-ZPOLXVRWSA-N prednisone Chemical compound O=C1C=C[C@]2(C)[C@H]3C(=O)C[C@](C)([C@@](CC4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 XOFYZVNMUHMLCC-ZPOLXVRWSA-N 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13305243 | 2013-03-04 | ||
| PCT/EP2014/054156 WO2014135524A1 (fr) | 2013-03-04 | 2014-03-04 | Cabazitaxel et son utilisation pour le traitement des cancers de la prostate métastatiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR20150442A true CR20150442A (es) | 2015-10-07 |
Family
ID=47901920
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR20150442A CR20150442A (es) | 2013-03-04 | 2015-08-25 | Cabazitaxel y su uso para el tratamiento de los cánceres de próstata metastásicos |
Country Status (21)
| Country | Link |
|---|---|
| US (2) | US20150374717A1 (fr) |
| EP (1) | EP2964212A1 (fr) |
| JP (1) | JP2016516673A (fr) |
| KR (1) | KR20150123892A (fr) |
| CN (2) | CN105073104A (fr) |
| AU (1) | AU2014224705A1 (fr) |
| BR (1) | BR112015021450A2 (fr) |
| CA (1) | CA2903132A1 (fr) |
| CL (1) | CL2015002454A1 (fr) |
| CR (1) | CR20150442A (fr) |
| EA (1) | EA201591622A1 (fr) |
| HK (1) | HK1215535A1 (fr) |
| IL (1) | IL241015A0 (fr) |
| MA (1) | MA38356A1 (fr) |
| MX (1) | MX2015011589A (fr) |
| PH (1) | PH12015501900A1 (fr) |
| SG (1) | SG11201506803XA (fr) |
| TN (1) | TN2015000378A1 (fr) |
| TW (2) | TW201438714A (fr) |
| WO (1) | WO2014135524A1 (fr) |
| ZA (1) | ZA201506310B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016113752A2 (fr) * | 2015-01-12 | 2016-07-21 | Emcure Pharmaceuticals Limited | Formulation liquide de cabazitaxel |
| WO2022067185A1 (fr) * | 2020-09-27 | 2022-03-31 | Veru Inc. | Méthodes de traitement du cancer de la prostate à effets secondaires minimes |
| JP2024534805A (ja) * | 2021-08-17 | 2024-09-26 | フォンダツィオーネ ペル リスティトゥート オンコロジコ ディ リチェルカ (イオエッレ) | 共生細菌は前立腺がんにおいてアンドロゲン生合成を介して内分泌抵抗性を促進する |
| KR102685052B1 (ko) * | 2023-02-15 | 2024-07-12 | 사회복지법인 삼성생명공익재단 | 전이성 전립선암의 호르몬 치료 저항성 예측용 신규 바이오마커 및 이의 용도 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2862340T3 (es) * | 2009-10-29 | 2021-10-07 | Sanofi Mature Ip | Nuevo uso antitumoral de cabazitaxel |
-
2014
- 2014-02-27 TW TW103106902A patent/TW201438714A/zh unknown
- 2014-02-27 TW TW107107732A patent/TW201827417A/zh unknown
- 2014-03-04 CA CA2903132A patent/CA2903132A1/fr not_active Abandoned
- 2014-03-04 SG SG11201506803XA patent/SG11201506803XA/en unknown
- 2014-03-04 KR KR1020157026716A patent/KR20150123892A/ko not_active Withdrawn
- 2014-03-04 HK HK16103503.6A patent/HK1215535A1/zh unknown
- 2014-03-04 EA EA201591622A patent/EA201591622A1/ru unknown
- 2014-03-04 MA MA38356A patent/MA38356A1/fr unknown
- 2014-03-04 JP JP2015560660A patent/JP2016516673A/ja not_active Ceased
- 2014-03-04 CN CN201480012665.2A patent/CN105073104A/zh active Pending
- 2014-03-04 EP EP14708014.7A patent/EP2964212A1/fr not_active Withdrawn
- 2014-03-04 BR BR112015021450A patent/BR112015021450A2/pt not_active IP Right Cessation
- 2014-03-04 WO PCT/EP2014/054156 patent/WO2014135524A1/fr not_active Ceased
- 2014-03-04 CN CN201810410731.1A patent/CN108354921A/zh active Pending
- 2014-03-04 AU AU2014224705A patent/AU2014224705A1/en not_active Abandoned
- 2014-03-04 MX MX2015011589A patent/MX2015011589A/es unknown
-
2015
- 2015-08-25 CR CR20150442A patent/CR20150442A/es unknown
- 2015-08-27 ZA ZA2015/06310A patent/ZA201506310B/en unknown
- 2015-08-27 PH PH12015501900A patent/PH12015501900A1/en unknown
- 2015-08-31 TN TN2015000378A patent/TN2015000378A1/en unknown
- 2015-09-01 IL IL241015A patent/IL241015A0/en unknown
- 2015-09-02 CL CL2015002454A patent/CL2015002454A1/es unknown
- 2015-09-03 US US14/844,480 patent/US20150374717A1/en not_active Abandoned
-
2016
- 2016-12-14 US US15/378,728 patent/US20180042941A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20150374717A1 (en) | 2015-12-31 |
| PH12015501900A1 (en) | 2016-01-11 |
| CN108354921A (zh) | 2018-08-03 |
| TW201438714A (zh) | 2014-10-16 |
| KR20150123892A (ko) | 2015-11-04 |
| MX2015011589A (es) | 2016-06-24 |
| HK1215535A1 (zh) | 2016-09-02 |
| ZA201506310B (en) | 2017-02-22 |
| CA2903132A1 (fr) | 2014-09-12 |
| EP2964212A1 (fr) | 2016-01-13 |
| CL2015002454A1 (es) | 2016-02-12 |
| TN2015000378A1 (en) | 2017-01-03 |
| BR112015021450A2 (pt) | 2017-07-18 |
| US20180042941A1 (en) | 2018-02-15 |
| TW201827417A (zh) | 2018-08-01 |
| JP2016516673A (ja) | 2016-06-09 |
| MA38356A1 (fr) | 2017-06-30 |
| WO2014135524A1 (fr) | 2014-09-12 |
| IL241015A0 (en) | 2015-11-30 |
| SG11201506803XA (en) | 2015-09-29 |
| AU2014224705A1 (en) | 2015-09-24 |
| CN105073104A (zh) | 2015-11-18 |
| EA201591622A1 (ru) | 2016-04-29 |
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