CR20150666A - Composición farmacéutica sinergística de dos analgésicos con distinto perfil farmacocinético - Google Patents
Composición farmacéutica sinergística de dos analgésicos con distinto perfil farmacocinéticoInfo
- Publication number
- CR20150666A CR20150666A CR20150666A CR20150666A CR20150666A CR 20150666 A CR20150666 A CR 20150666A CR 20150666 A CR20150666 A CR 20150666A CR 20150666 A CR20150666 A CR 20150666A CR 20150666 A CR20150666 A CR 20150666A
- Authority
- CR
- Costa Rica
- Prior art keywords
- pharmacocinetic
- analgesics
- profile
- different
- pharmaceutical composition
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229940035676 analgesics Drugs 0.000 title 1
- 239000000730 antalgic agent Substances 0.000 title 1
- 230000002195 synergetic effect Effects 0.000 title 1
- 230000000202 analgesic effect Effects 0.000 abstract 2
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 2
- 230000003637 steroidlike Effects 0.000 abstract 2
- ZRVUJXDFFKFLMG-UHFFFAOYSA-N Meloxicam Chemical compound OC=1C2=CC=CC=C2S(=O)(=O)N(C)C=1C(=O)NC1=NC=C(C)S1 ZRVUJXDFFKFLMG-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- CVNFYQCHAWFYQI-ZSCHJXSPSA-N clonixin lysine salt Chemical compound NCCCC[C@H](N)C(O)=O.CC1=C(Cl)C=CC=C1NC1=NC=CC=C1C(O)=O CVNFYQCHAWFYQI-ZSCHJXSPSA-N 0.000 abstract 1
- 229960003763 lysine clonixinate Drugs 0.000 abstract 1
- 229960001929 meloxicam Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/455—Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Dermatology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se refiere a composiciones farmacéuticas que contienen dos principios activos siendo uno de ellos un analgésico antiinflamatorio no esteroideo conocido como meloxicam o una de sus sales farmacéuticamente aceptables y el otro un analgésico antiinflamatorio no esteroideo conocido como clonixinato de lisina.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/MX2013/000070 WO2014193210A1 (es) | 2013-05-27 | 2013-05-27 | Composición farmacéutica sinergística de dos analgésicos con distinto perfil farmacocinético |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR20150666A true CR20150666A (es) | 2016-03-03 |
Family
ID=51989148
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR20150666A CR20150666A (es) | 2013-05-27 | 2015-12-17 | Composición farmacéutica sinergística de dos analgésicos con distinto perfil farmacocinético |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP3025717B1 (es) |
| BR (1) | BR112015024314A2 (es) |
| CR (1) | CR20150666A (es) |
| ES (1) | ES2586607B1 (es) |
| MX (1) | MX351622B (es) |
| WO (1) | WO2014193210A1 (es) |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2262967B1 (es) * | 1974-03-07 | 1977-11-04 | Roemmers Sa Ind Comercial | |
| DE4037554A1 (de) * | 1990-11-26 | 1992-05-27 | Roemmers Sa | Arzneimittel zur topischen anwendung |
| US8512727B2 (en) * | 2003-03-03 | 2013-08-20 | Alkermes Pharma Ireland Limited | Nanoparticulate meloxicam formulations |
| WO2007083985A1 (es) * | 2006-01-19 | 2007-07-26 | Farmacéuticos Rayere, S.A. | Composición farmacéutica sinergística de diclofenaco y clonixinato de lisina |
| US20070281927A1 (en) * | 2006-06-06 | 2007-12-06 | Shanthakumar Tyavanagimatt | Anti-inflammatory and analgesic compositions and related methods |
| WO2007148950A1 (es) * | 2006-06-20 | 2007-12-27 | Farmacéuticos Rayere, S.A. | Composición farmacéutica sinergística de ketorolaco y clonixinato de lisina |
| MX357376B (es) * | 2011-06-22 | 2018-07-06 | Laboratorios Senosiain S A De C V Star | Composicion farmaceutica para uso en inflamacion y dolor. |
-
2013
- 2013-05-27 ES ES201590124A patent/ES2586607B1/es not_active Expired - Fee Related
- 2013-05-27 WO PCT/MX2013/000070 patent/WO2014193210A1/es not_active Ceased
- 2013-05-27 MX MX2014004492A patent/MX351622B/es active IP Right Grant
- 2013-05-27 EP EP13885633.1A patent/EP3025717B1/en not_active Not-in-force
- 2013-05-27 BR BR112015024314A patent/BR112015024314A2/pt not_active Application Discontinuation
-
2015
- 2015-12-17 CR CR20150666A patent/CR20150666A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP3025717A1 (en) | 2016-06-01 |
| EP3025717A4 (en) | 2017-03-15 |
| BR112015024314A2 (pt) | 2017-07-18 |
| MX351622B (es) | 2017-10-17 |
| ES2586607B1 (es) | 2017-07-20 |
| EP3025717B1 (en) | 2018-11-07 |
| MX2014004492A (es) | 2016-03-15 |
| WO2014193210A1 (es) | 2014-12-04 |
| ES2586607A1 (es) | 2016-10-17 |
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