CR20220610A - Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas - Google Patents
Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismasInfo
- Publication number
- CR20220610A CR20220610A CR20220610A CR20220610A CR20220610A CR 20220610 A CR20220610 A CR 20220610A CR 20220610 A CR20220610 A CR 20220610A CR 20220610 A CR20220610 A CR 20220610A CR 20220610 A CR20220610 A CR 20220610A
- Authority
- CR
- Costa Rica
- Prior art keywords
- compound
- formula
- mixtures
- fungicidally effective
- compositions
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/22—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/69—Benzenesulfonamido-pyrimidines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
- A01N25/04—Dispersions, emulsions, suspoemulsions, suspension concentrates or gels
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/12—Powders or granules
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/30—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests characterised by the surfactants
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
- A01N25/32—Ingredients for reducing the noxious effect of the active substances to organisms other than pests, e.g. toxicity reducing compositions, self-destructing compositions
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P3/00—Fungicides
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Agronomy & Crop Science (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Toxicology (AREA)
- Microbiology (AREA)
- Mycology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Dispersion Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención proporciona una composición líquida estable que comprende: (a) una cantidad fungicidamente eficaz de un compuesto de Fórmula I, y (b) un vehículo líquido, en el que: (i) la composición comprende (a) una sustancia fungicidamente eficaz y sustancialmente pura cantidad del compuesto de Fórmula I o una cantidad eficaz como fungicida de una mezcla que contiene el compuesto de Fórmula I, donde 95% o más en peso de la mezcla es el compuesto de Fórmula I, y (b) el vehículo líquido, y / o (ii) 95% o más de la cantidad del compuesto de Fórmula I está en forma de polimorfo de Forma I, polimorfo de Forma II, Hidrato, o una mezcla de los mismos. La presente invención también proporciona mezclas y composiciones que comprenden (a) una cantidad fungicidamente eficaz de un compuesto de Fórmula I y (b) al menos un adyuvante seleccionado del grupo que consiste en: (i) poli (óxido de alquileno) alquil éter; (ii) copolímero de óxido de polialquileno de siloxano; (iii) ésteres de ácidos grasos; (iv) vinilpirrolidonas y derivados de las mismas; (v) tensioactivos a base de azúcar, (vi) ligninas, (vii) terpenos; y (viii) cualquier combinación de (i), (ii), (iii), (iv), (v), (vi) y (vii). La presente invención también proporciona métodos de uso de las mezclas y composiciones descritas en este documento y procesos para preparar las mezclas y composiciones descritas en este documento.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063019871P | 2020-05-04 | 2020-05-04 | |
| US202063024031P | 2020-05-13 | 2020-05-13 | |
| PCT/IB2021/053762 WO2021224802A1 (en) | 2020-05-04 | 2021-05-04 | Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR20220610A true CR20220610A (es) | 2023-01-10 |
Family
ID=75888117
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR20220610A CR20220610A (es) | 2020-05-04 | 2021-05-04 | Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20230292746A1 (es) |
| EP (1) | EP4146632A1 (es) |
| JP (2) | JP7826287B2 (es) |
| KR (1) | KR20230069875A (es) |
| CN (1) | CN116113623A (es) |
| AU (1) | AU2021267206A1 (es) |
| BR (1) | BR112022022281A2 (es) |
| CA (1) | CA3177682A1 (es) |
| CL (1) | CL2022003040A1 (es) |
| CO (1) | CO2022017377A2 (es) |
| CR (1) | CR20220610A (es) |
| EC (1) | ECSP22091704A (es) |
| IL (1) | IL297864A (es) |
| MX (1) | MX2022013874A (es) |
| PE (1) | PE20230446A1 (es) |
| PY (1) | PY2135531A (es) |
| TW (1) | TW202208341A (es) |
| UY (1) | UY39197A (es) |
| WO (1) | WO2021224802A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3876717A1 (en) | 2018-11-05 | 2021-09-15 | Adama Makhteshim Ltd. | Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof |
| PY2057637A (es) | 2019-09-23 | 2021-10-05 | Adama Makhteshim Ltd | Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto |
| TW202208355A (zh) | 2020-05-04 | 2022-03-01 | 美商安進公司 | 作為骨髓細胞觸發受體2促效劑之雜環化合物及使用方法 |
| PE20230609A1 (es) | 2020-05-04 | 2023-04-13 | Amgen Inc | Compuestos heterociclicos como agonistas del receptor de activacion expresado en las celulas mieloides 2 y metodos de uso |
| UY40172A (es) * | 2022-03-03 | 2023-10-13 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas |
| AU2023318916A1 (en) | 2022-08-03 | 2025-02-20 | Adama Makhteshim Ltd. | 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1h)-one for fungicide-resistant fungus |
| IL308593A (en) * | 2023-11-15 | 2025-06-01 | Adama Makhteshim Ltd | Reducing environmental impact of fungicidal enhancement |
| WO2026038217A1 (en) | 2024-08-15 | 2026-02-19 | Adama Makhteshim Ltd. | Mixtures and compositions comprising flumetylsulforim and methods of use thereof |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2614303T3 (es) * | 2003-11-17 | 2017-05-30 | Syngenta Participations Ag | Concentrados emulsionables que contienen adyuvantes |
| PH12012502138B1 (en) | 2010-04-26 | 2019-09-25 | Adama Makhteshim Ltd | N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives |
| JP6315702B2 (ja) * | 2012-02-27 | 2018-04-25 | ハンツマン・コーポレーシヨン・オーストラリア・ピーテイワイ・リミテツド | 農薬乳化性濃厚調剤 |
| AU2013370494B2 (en) * | 2012-12-31 | 2017-08-17 | Adama Makhteshim Ltd. | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides |
| EP3021668B1 (en) * | 2013-07-18 | 2018-09-12 | Basf Se | Emulsifiable concentrate comprising pesticide, alkyl lactate, fatty amide and acetophenone |
| CA2935594C (en) | 2013-12-31 | 2022-05-03 | Nakyen Choy | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
| NZ722419A (en) * | 2013-12-31 | 2018-01-26 | Adama Makhteshim Ltd | Synergistic fungicidal mixtures and compositions for fungal control |
| MA41272A (fr) | 2014-12-23 | 2017-10-31 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences |
| UY36964A (es) * | 2015-10-27 | 2017-05-31 | Bayer Cropscience Ag | Combinaciones de principios activos que comprenden un derivado de (tio) carboxamida y un compuesto funguicida |
| JP2017122055A (ja) | 2016-01-05 | 2017-07-13 | 日本農薬株式会社 | フルオロピリミジン化合物を含有する有害生物防除剤組成物及びその使用方法 |
| JP6922271B2 (ja) | 2016-03-11 | 2021-08-18 | 住友化学株式会社 | 植物病害防除組成物及び植物病害防除方法 |
| JP6922272B2 (ja) * | 2016-03-11 | 2021-08-18 | 住友化学株式会社 | 植物病害防除組成物及び植物病害防除方法 |
| EP3655396A1 (en) * | 2017-07-17 | 2020-05-27 | Adama Makhteshim Ltd. | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| EP3876717A1 (en) * | 2018-11-05 | 2021-09-15 | Adama Makhteshim Ltd. | Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof |
-
2021
- 2021-05-04 EP EP21724789.9A patent/EP4146632A1/en active Pending
- 2021-05-04 KR KR1020227042365A patent/KR20230069875A/ko active Pending
- 2021-05-04 CN CN202180043243.1A patent/CN116113623A/zh active Pending
- 2021-05-04 WO PCT/IB2021/053762 patent/WO2021224802A1/en not_active Ceased
- 2021-05-04 BR BR112022022281A patent/BR112022022281A2/pt unknown
- 2021-05-04 JP JP2023509880A patent/JP7826287B2/ja active Active
- 2021-05-04 AU AU2021267206A patent/AU2021267206A1/en active Pending
- 2021-05-04 UY UY0001039197A patent/UY39197A/es unknown
- 2021-05-04 PE PE2022002560A patent/PE20230446A1/es unknown
- 2021-05-04 IL IL297864A patent/IL297864A/en unknown
- 2021-05-04 CA CA3177682A patent/CA3177682A1/en active Pending
- 2021-05-04 TW TW110116082A patent/TW202208341A/zh unknown
- 2021-05-04 US US17/997,903 patent/US20230292746A1/en active Pending
- 2021-05-04 PY PY202102135531A patent/PY2135531A/es unknown
- 2021-05-04 CR CR20220610A patent/CR20220610A/es unknown
- 2021-05-04 MX MX2022013874A patent/MX2022013874A/es unknown
-
2022
- 2022-11-03 CL CL2022003040A patent/CL2022003040A1/es unknown
- 2022-12-01 EC ECSENADI202291704A patent/ECSP22091704A/es unknown
- 2022-12-02 CO CONC2022/0017377A patent/CO2022017377A2/es unknown
-
2025
- 2025-11-25 JP JP2025203016A patent/JP2026048693A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| MX2022013874A (es) | 2022-11-30 |
| CO2022017377A2 (es) | 2022-12-20 |
| CA3177682A1 (en) | 2021-11-11 |
| EP4146632A1 (en) | 2023-03-15 |
| PE20230446A1 (es) | 2023-03-08 |
| BR112022022281A2 (pt) | 2023-01-03 |
| UY39197A (es) | 2021-11-30 |
| CN116113623A (zh) | 2023-05-12 |
| KR20230069875A (ko) | 2023-05-19 |
| ECSP22091704A (es) | 2023-02-28 |
| IL297864A (en) | 2023-01-01 |
| AU2021267206A1 (en) | 2022-12-08 |
| PY2135531A (es) | 2022-02-01 |
| TW202208341A (zh) | 2022-03-01 |
| CL2022003040A1 (es) | 2023-07-07 |
| WO2021224802A1 (en) | 2021-11-11 |
| JP2023523655A (ja) | 2023-06-06 |
| JP7826287B2 (ja) | 2026-03-09 |
| JP2026048693A (ja) | 2026-03-17 |
| US20230292746A1 (en) | 2023-09-21 |
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