CR7203A - 5-SUBSTITUTES-2-ARILPIRIDINAS AS MODULATORS OF CORTICOTROPINE RELEASE FACTOR 1 - Google Patents
5-SUBSTITUTES-2-ARILPIRIDINAS AS MODULATORS OF CORTICOTROPINE RELEASE FACTOR 1Info
- Publication number
- CR7203A CR7203A CR7203A CR7203A CR7203A CR 7203 A CR7203 A CR 7203A CR 7203 A CR7203 A CR 7203A CR 7203 A CR7203 A CR 7203A CR 7203 A CR7203 A CR 7203A
- Authority
- CR
- Costa Rica
- Prior art keywords
- modulators
- arilpiridinas
- substitutes
- disorders
- release factor
- Prior art date
Links
- IDLFZVILOHSSID-OVLDLUHVSA-N corticotropin Chemical compound C([C@@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C(C)C)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC=1C=CC=CC=1)C(O)=O)NC(=O)[C@@H](N)CO)C1=CC=C(O)C=C1 IDLFZVILOHSSID-OVLDLUHVSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 208000019901 Anxiety disease Diseases 0.000 abstract 1
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
- 108010056643 Corticotropin-Releasing Hormone Receptors Proteins 0.000 abstract 1
- 208000030814 Eating disease Diseases 0.000 abstract 1
- 208000019454 Feeding and Eating disease Diseases 0.000 abstract 1
- 206010043268 Tension Diseases 0.000 abstract 1
- 230000036506 anxiety Effects 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 235000014632 disordered eating Nutrition 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 210000001428 peripheral nervous system Anatomy 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Estos compuestos pueden actuar como moduladores selectivos de receptores de CRF. Los compuestos de 5-sustituidas-2-arilpiridinas proporcionados son utiles en el tratamiento de varios trastornos de sistema nervioso central y periferico, de manera particular, tension nerviosa, ansiedad, depresion, trastornos cardiovasculares, y trastornos de alimentacion. Se proporciona un metodo de tratamiento de estos trastornos y tambien como composiciones farmaceuticas envasadas.These compounds can act as selective modulators of CRF receptors. The 5-substituted-2-arylpyridine compounds provided are useful in the treatment of various disorders of the central and peripheral nervous system, in particular, nervous tension, anxiety, depression, cardiovascular disorders, and eating disorders. A method of treatment of these disorders and also as packaged pharmaceutical compositions is provided.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CR7203A CR7203A (en) | 2003-12-15 | 2003-12-15 | 5-SUBSTITUTES-2-ARILPIRIDINAS AS MODULATORS OF CORTICOTROPINE RELEASE FACTOR 1 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CR7203A CR7203A (en) | 2003-12-15 | 2003-12-15 | 5-SUBSTITUTES-2-ARILPIRIDINAS AS MODULATORS OF CORTICOTROPINE RELEASE FACTOR 1 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR7203A true CR7203A (en) | 2004-02-23 |
Family
ID=44839148
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR7203A CR7203A (en) | 2003-12-15 | 2003-12-15 | 5-SUBSTITUTES-2-ARILPIRIDINAS AS MODULATORS OF CORTICOTROPINE RELEASE FACTOR 1 |
Country Status (1)
| Country | Link |
|---|---|
| CR (1) | CR7203A (en) |
-
2003
- 2003-12-15 CR CR7203A patent/CR7203A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal (granting procedure) |