CR9238A - PIRROLOPIRAZOLES, POWERFUL INHIBITORS OF CINASA - Google Patents
PIRROLOPIRAZOLES, POWERFUL INHIBITORS OF CINASAInfo
- Publication number
- CR9238A CR9238A CR9238A CR9238A CR9238A CR 9238 A CR9238 A CR 9238A CR 9238 A CR9238 A CR 9238A CR 9238 A CR9238 A CR 9238A CR 9238 A CR9238 A CR 9238A
- Authority
- CR
- Costa Rica
- Prior art keywords
- pirrolopirazoles
- cinasa
- powerful inhibitors
- inhibitors
- compounds
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 101000987297 Homo sapiens Serine/threonine-protein kinase PAK 4 Proteins 0.000 abstract 1
- 102100027940 Serine/threonine-protein kinase PAK 4 Human genes 0.000 abstract 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000003909 protein kinase inhibitor Substances 0.000 abstract 1
- GZTPJDLYPMPRDF-UHFFFAOYSA-N pyrrolo[3,2-c]pyrazole Chemical class N1=NC2=CC=NC2=C1 GZTPJDLYPMPRDF-UHFFFAOYSA-N 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Se proporcionan compuestos de pirrolo-pirazol de formula I, composiciones que incluyen estos compuestos y procedimientos de su uso. Los compuestos preferidos de formula I tienen actividad como inhibidores de proteina cinasa, incluyendo como inhibidores de PAK4.Pyrrolo-pyrazole compounds of formula I, compositions including these compounds and methods of their use are provided. Preferred compounds of formula I have activity as protein kinase inhibitors, including as PAK4 inhibitors.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CR9238A CR9238A (en) | 2007-07-10 | 2007-07-10 | PIRROLOPIRAZOLES, POWERFUL INHIBITORS OF CINASA |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CR9238A CR9238A (en) | 2007-07-10 | 2007-07-10 | PIRROLOPIRAZOLES, POWERFUL INHIBITORS OF CINASA |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR9238A true CR9238A (en) | 2007-08-16 |
Family
ID=44839384
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR9238A CR9238A (en) | 2007-07-10 | 2007-07-10 | PIRROLOPIRAZOLES, POWERFUL INHIBITORS OF CINASA |
Country Status (1)
| Country | Link |
|---|---|
| CR (1) | CR9238A (en) |
-
2007
- 2007-07-10 CR CR9238A patent/CR9238A/en unknown
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