CR9645A - COMPLEXES WITH CONTENT OF PERFLUOROALQUILO, PROCEDURES FOR ITS PREPARATION AS WELL AS ITS USE - Google Patents
COMPLEXES WITH CONTENT OF PERFLUOROALQUILO, PROCEDURES FOR ITS PREPARATION AS WELL AS ITS USEInfo
- Publication number
- CR9645A CR9645A CR9645A CR9645A CR9645A CR 9645 A CR9645 A CR 9645A CR 9645 A CR9645 A CR 9645A CR 9645 A CR9645 A CR 9645A CR 9645 A CR9645 A CR 9645A
- Authority
- CR
- Costa Rica
- Prior art keywords
- preparation
- content
- well
- perfluoroalquilo
- complexes
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 238000009825 accumulation Methods 0.000 abstract 1
- 239000008280 blood Substances 0.000 abstract 1
- 210000004369 blood Anatomy 0.000 abstract 1
- 238000003745 diagnosis Methods 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 150000002831 nitrogen free-radicals Chemical class 0.000 abstract 1
- 125000005010 perfluoroalkyl group Chemical group 0.000 abstract 1
- 238000001959 radiotherapy Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Radiology & Medical Imaging (AREA)
- Engineering & Computer Science (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Steroid Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La invencion se refiere a los objetos caracterizados en las reivindicaciones, a saber, complejos metalicos con contenido de perfluoroalquilo con radicales con nitrogeno de la formula general I, a procedimientos para su preparacion y a su uso en el diagnostico por RMN y rayos X, en el radiodiagnostico y la radioterapia, asi como en la linfografia MRT y para la representacion de la acumulacion de sangre por imagenes.The invention relates to the objects characterized in the claims, namely, metal complexes containing perfluoroalkyl content with nitrogen radicals of the general formula I, methods for their preparation and their use in the diagnosis by NMR and X-rays, in the radiodiagnosis and radiotherapy, as well as in MRT lymphography and for the representation of blood accumulation by images.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005033902A DE102005033902B3 (en) | 2005-07-15 | 2005-07-15 | Perfluoroalkyl-containing complexes, processes for their preparation, and their use and pharmaceutical compositions containing them |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR9645A true CR9645A (en) | 2008-05-21 |
Family
ID=37057146
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR9645A CR9645A (en) | 2005-07-15 | 2008-01-08 | COMPLEXES WITH CONTENT OF PERFLUOROALQUILO, PROCEDURES FOR ITS PREPARATION AS WELL AS ITS USE |
Country Status (22)
| Country | Link |
|---|---|
| EP (1) | EP1904463A2 (en) |
| JP (1) | JP2009501174A (en) |
| KR (1) | KR20080043762A (en) |
| CN (1) | CN101223148A (en) |
| AR (1) | AR054865A1 (en) |
| AU (1) | AU2006272025A1 (en) |
| BR (1) | BRPI0613407A2 (en) |
| CA (1) | CA2615443A1 (en) |
| CR (1) | CR9645A (en) |
| DE (1) | DE102005033902B3 (en) |
| DO (1) | DOP2006000167A (en) |
| EC (1) | ECSP088100A (en) |
| GT (1) | GT200600313A (en) |
| IL (1) | IL187926A0 (en) |
| NO (1) | NO20080813L (en) |
| PE (1) | PE20070376A1 (en) |
| RU (1) | RU2008105356A (en) |
| TN (1) | TNSN08016A1 (en) |
| TW (1) | TW200706538A (en) |
| UY (1) | UY29664A1 (en) |
| WO (1) | WO2007009638A2 (en) |
| ZA (1) | ZA200801523B (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102007015598A1 (en) * | 2007-03-29 | 2008-10-02 | Heinrich-Heine-Universität Düsseldorf | Use of fluorochemical compounds for diagnostic purposes using imaging techniques |
| JP5730581B2 (en) | 2008-01-08 | 2015-06-10 | ランセウス メディカル イメージング, インコーポレイテッド | N-alkoxyamide conjugates as contrast agents |
| WO2021067738A1 (en) * | 2019-10-04 | 2021-04-08 | United States Government As Represented By The Department Of Veterans Affairs | Development of imaging and therapeutic glucose analogues for sodium dependent glucose transporters |
| EP4059925A1 (en) | 2021-03-15 | 2022-09-21 | Bayer Aktiengesellschaft | New contrast agent for use in magnetic resonance imaging |
| CN114181164A (en) * | 2021-12-13 | 2022-03-15 | 武汉大学中南医院 | Synthesis method and application of MRI contrast agent based on Fe (II) specificity |
| EP4335840A1 (en) | 2022-09-09 | 2024-03-13 | Bayer Aktiengesellschaft | New contrast agents for use in diagnostic imaging |
| EP4335462A1 (en) | 2022-09-09 | 2024-03-13 | Bayer AG | Contrast agents for use in diagnostic computed tomography imaging |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4317588C2 (en) * | 1993-05-24 | 1998-04-16 | Schering Ag | Macrocyclic metal complexes containing fluorine, process for their preparation and their use |
| DE19603033A1 (en) * | 1996-01-19 | 1997-07-24 | Schering Ag | Perfluoroalkyl-containing metal complexes, processes for their preparation and their use in NMR diagnostics |
| DE19744003B4 (en) * | 1997-09-26 | 2004-07-08 | Schering Ag | Contrast agent for infarct and necrosis imaging |
| DE19744004C1 (en) * | 1997-09-26 | 1999-07-22 | Schering Ag | Lipophilic metal complexes for necrosis and infarct imaging |
| DE19914101C1 (en) * | 1999-03-22 | 2000-10-12 | Schering Ag | Perfluoroalkylamides, their preparation and their use in diagnostics |
| DE10040858C2 (en) * | 2000-08-11 | 2003-12-18 | Schering Ag | Perfluoroalkyl-containing complexes with polar residues, process for their preparation and their use |
-
2005
- 2005-07-15 DE DE102005033902A patent/DE102005033902B3/en not_active Expired - Fee Related
-
2006
- 2006-07-11 CN CNA2006800258905A patent/CN101223148A/en active Pending
- 2006-07-11 UY UY29664A patent/UY29664A1/en not_active Application Discontinuation
- 2006-07-11 JP JP2008520780A patent/JP2009501174A/en not_active Withdrawn
- 2006-07-11 EP EP06791535A patent/EP1904463A2/en not_active Withdrawn
- 2006-07-11 KR KR1020087001084A patent/KR20080043762A/en not_active Withdrawn
- 2006-07-11 RU RU2008105356/04A patent/RU2008105356A/en not_active Application Discontinuation
- 2006-07-11 WO PCT/EP2006/006777 patent/WO2007009638A2/en not_active Ceased
- 2006-07-11 CA CA002615443A patent/CA2615443A1/en not_active Abandoned
- 2006-07-11 AU AU2006272025A patent/AU2006272025A1/en not_active Abandoned
- 2006-07-11 BR BRPI0613407-6A patent/BRPI0613407A2/en not_active Application Discontinuation
- 2006-07-13 DO DO2006000167A patent/DOP2006000167A/en unknown
- 2006-07-14 PE PE2006000844A patent/PE20070376A1/en not_active Application Discontinuation
- 2006-07-14 GT GT200600313A patent/GT200600313A/en unknown
- 2006-07-14 AR ARP060103020A patent/AR054865A1/en unknown
- 2006-07-14 TW TW095125755A patent/TW200706538A/en unknown
-
2007
- 2007-12-06 IL IL187926A patent/IL187926A0/en unknown
-
2008
- 2008-01-08 CR CR9645A patent/CR9645A/en unknown
- 2008-01-11 EC EC2008008100A patent/ECSP088100A/en unknown
- 2008-01-14 TN TNP2008000016A patent/TNSN08016A1/en unknown
- 2008-02-14 NO NO20080813A patent/NO20080813L/en not_active Application Discontinuation
- 2008-02-14 ZA ZA200801523A patent/ZA200801523B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UY29664A1 (en) | 2007-02-28 |
| AU2006272025A1 (en) | 2007-01-25 |
| NO20080813L (en) | 2008-04-09 |
| IL187926A0 (en) | 2008-03-20 |
| EP1904463A2 (en) | 2008-04-02 |
| ECSP088100A (en) | 2008-05-30 |
| ZA200801523B (en) | 2008-11-26 |
| GT200600313A (en) | 2007-04-23 |
| PE20070376A1 (en) | 2007-04-20 |
| BRPI0613407A2 (en) | 2011-01-11 |
| TNSN08016A1 (en) | 2009-07-14 |
| CA2615443A1 (en) | 2007-01-25 |
| TW200706538A (en) | 2007-02-16 |
| KR20080043762A (en) | 2008-05-19 |
| RU2008105356A (en) | 2009-08-20 |
| AR054865A1 (en) | 2007-07-25 |
| WO2007009638A2 (en) | 2007-01-25 |
| DE102005033902B3 (en) | 2007-04-05 |
| CN101223148A (en) | 2008-07-16 |
| DOP2006000167A (en) | 2007-02-28 |
| JP2009501174A (en) | 2009-01-15 |
| WO2007009638A3 (en) | 2007-04-26 |
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