CR9853A - Compuestos de exemestano (s)-6-metiloxaalquilo y metodos relacionados con su utilizacion - Google Patents
Compuestos de exemestano (s)-6-metiloxaalquilo y metodos relacionados con su utilizacionInfo
- Publication number
- CR9853A CR9853A CR9853A CR9853A CR9853A CR 9853 A CR9853 A CR 9853A CR 9853 A CR9853 A CR 9853A CR 9853 A CR9853 A CR 9853A CR 9853 A CR9853 A CR 9853A
- Authority
- CR
- Costa Rica
- Prior art keywords
- methylloxyalquil
- methods related
- compounds
- exemestane
- exemestane compounds
- Prior art date
Links
- BFYIZQONLCFLEV-DAELLWKTSA-N Aromasine Chemical class O=C1C=C[C@]2(C)[C@H]3CC[C@](C)(C(CC4)=O)[C@@H]4[C@@H]3CC(=C)C2=C1 BFYIZQONLCFLEV-DAELLWKTSA-N 0.000 title 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000035755 proliferation Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0003—Androstane derivatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Abstract
Los compuestos de cemestano 6-Metiloxaalquilo y composiciones relacionadas, de la forma en que pueden utilizarse, quimioterapeuticamente, para inhibir el desarrrollo y proliferacion de celulas cancerosas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US72220405P | 2005-09-30 | 2005-09-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR9853A true CR9853A (es) | 2008-10-10 |
Family
ID=37906827
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR9853A CR9853A (es) | 2005-09-30 | 2008-03-31 | Compuestos de exemestano (s)-6-metiloxaalquilo y metodos relacionados con su utilizacion |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7846918B2 (es) |
| EP (1) | EP1931385B1 (es) |
| JP (1) | JP5255444B2 (es) |
| KR (1) | KR101484134B1 (es) |
| CN (1) | CN101312743A (es) |
| BR (1) | BRPI0616639A2 (es) |
| CA (1) | CA2624269C (es) |
| CR (1) | CR9853A (es) |
| WO (1) | WO2007041564A2 (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE548375T1 (de) * | 2004-01-16 | 2012-03-15 | Cedarburg Pharmaceuticals Inc | Exemestan und zwischenprodukte davon und verfahren zu dessen herstellung |
| US10174070B2 (en) * | 2005-09-30 | 2019-01-08 | Endece Llc | 6-substituted estradiol derivatives and methods of use |
| US8168621B2 (en) | 2005-09-30 | 2012-05-01 | Endece, Llc | 6-substituted estradiol derivatives and methods of use |
| CA2670773C (en) * | 2006-11-30 | 2013-01-22 | Endece, Llc | 6-alkoxyalkyl estradiol derivatives and methods of use |
| CA2794565C (en) | 2010-04-08 | 2018-08-21 | Emory University | Substituted androst-4-ene diones |
| ES2605960T3 (es) | 2010-09-14 | 2017-03-17 | Endece, Llc | Derivados de desmetil-estradiol 6-sustituido como agonistas del RE-beta |
| AU2012230974B2 (en) * | 2011-03-21 | 2016-05-12 | Endece Llc | 6-substituted estradiol derivatives for use in remyelination of nerve axons |
| US9585894B2 (en) | 2013-07-19 | 2017-03-07 | The Johns Hopkins University | Compositions comprising exemestane and novel methods of use |
| WO2022133265A1 (en) * | 2020-12-17 | 2022-06-23 | University Of Florida Research Foundation, Incorported | Steroidal compound derivatives as therapeutic agents |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8517360D0 (en) | 1985-07-09 | 1985-08-14 | Erba Farmitalia | Substituted androsta-1,4-diene-3,17-diones |
| JPH07215992A (ja) * | 1993-12-07 | 1995-08-15 | Teikoku Hormone Mfg Co Ltd | 6−又は7−置換アンドロスタ−1,4−ジエン誘導体 |
| ATE548375T1 (de) | 2004-01-16 | 2012-03-15 | Cedarburg Pharmaceuticals Inc | Exemestan und zwischenprodukte davon und verfahren zu dessen herstellung |
-
2006
- 2006-10-02 BR BRPI0616639-3A patent/BRPI0616639A2/pt not_active Application Discontinuation
- 2006-10-02 EP EP06825386.3A patent/EP1931385B1/en not_active Not-in-force
- 2006-10-02 CA CA2624269A patent/CA2624269C/en not_active Expired - Fee Related
- 2006-10-02 JP JP2008533773A patent/JP5255444B2/ja not_active Expired - Fee Related
- 2006-10-02 CN CNA2006800431487A patent/CN101312743A/zh active Pending
- 2006-10-02 KR KR20087010296A patent/KR101484134B1/ko not_active Expired - Fee Related
- 2006-10-02 WO PCT/US2006/038583 patent/WO2007041564A2/en not_active Ceased
- 2006-10-02 US US11/541,987 patent/US7846918B2/en not_active Expired - Fee Related
-
2008
- 2008-03-31 CR CR9853A patent/CR9853A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007041564A3 (en) | 2007-07-05 |
| EP1931385A2 (en) | 2008-06-18 |
| KR20080054426A (ko) | 2008-06-17 |
| WO2007041564A2 (en) | 2007-04-12 |
| EP1931385A4 (en) | 2009-06-24 |
| JP2009510125A (ja) | 2009-03-12 |
| CA2624269C (en) | 2016-03-22 |
| CA2624269A1 (en) | 2007-04-12 |
| KR101484134B1 (ko) | 2015-01-21 |
| BRPI0616639A2 (pt) | 2011-06-28 |
| US7846918B2 (en) | 2010-12-07 |
| EP1931385B1 (en) | 2018-02-28 |
| JP5255444B2 (ja) | 2013-08-07 |
| US20070088013A1 (en) | 2007-04-19 |
| CN101312743A (zh) | 2008-11-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal (granting procedure) |