CS189391A3 - Dialkoxypiridylbenzimidazole derivatives, process of their preparation and their pharmaceutical use - Google Patents

Dialkoxypiridylbenzimidazole derivatives, process of their preparation and their pharmaceutical use

Info

Publication number
CS189391A3
CS189391A3 CS911893A CS189391A CS189391A3 CS 189391 A3 CS189391 A3 CS 189391A3 CS 911893 A CS911893 A CS 911893A CS 189391 A CS189391 A CS 189391A CS 189391 A3 CS189391 A3 CS 189391A3
Authority
CS
Czechoslovakia
Prior art keywords
dialkoxypiridylbenzimidazole
derivatives
preparation
pharmaceutical use
pharmaceutical
Prior art date
Application number
CS911893A
Other languages
English (en)
Inventor
Arne Elof Brandstrom
Per Lennart Lindberg
Gunnel Elisabeth Senden
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE9002206A external-priority patent/SE9002206D0/xx
Priority claimed from SE9002207A external-priority patent/SE9002207D0/xx
Application filed by Astra Ab filed Critical Astra Ab
Publication of CS189391A3 publication Critical patent/CS189391A3/cs
Publication of CZ279434B6 publication Critical patent/CZ279434B6/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS911893A 1990-06-20 1991-06-20 Dialkoxypyridylbenzimidazolové deriváty, způsob jejich výroby a farmaceutický prostředek, který j e obsahuje a použití dialkoxypyridylbenzimidazolo vých derivátů k výrobě léčiva. CZ279434B6 (cs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9002206A SE9002206D0 (sv) 1990-06-20 1990-06-20 New compounds
SE9002207A SE9002207D0 (sv) 1990-06-20 1990-06-20 New compounds i

Publications (2)

Publication Number Publication Date
CS189391A3 true CS189391A3 (en) 1992-06-17
CZ279434B6 CZ279434B6 (cs) 1995-04-12

Family

ID=26660803

Country Status (29)

Country Link
US (1) US5430042A (cs)
EP (1) EP0593463B1 (cs)
JP (1) JP3049367B2 (cs)
CN (1) CN1058213A (cs)
AP (1) AP253A (cs)
AT (1) ATE184602T1 (cs)
AU (1) AU649456B2 (cs)
BG (1) BG97198A (cs)
CA (1) CA2083606C (cs)
CZ (1) CZ279434B6 (cs)
DE (1) DE69131627T2 (cs)
EG (1) EG19752A (cs)
ES (1) ES2140391T3 (cs)
FI (1) FI925767A7 (cs)
HU (1) HUT62882A (cs)
IE (1) IE912026A1 (cs)
IL (1) IL98472A (cs)
IS (1) IS3720A7 (cs)
LV (1) LV10269B (cs)
MA (1) MA22198A1 (cs)
NO (1) NO924650L (cs)
NZ (1) NZ238545A (cs)
OA (1) OA09683A (cs)
PL (2) PL166209B1 (cs)
PT (1) PT98036A (cs)
RO (1) RO110497B1 (cs)
TN (1) TNSN91050A1 (cs)
WO (1) WO1991019712A1 (cs)
YU (1) YU104091A (cs)

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SE9500422D0 (sv) * 1995-02-06 1995-02-06 Astra Ab New oral pharmaceutical dosage forms
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US6645988B2 (en) * 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
US6699885B2 (en) * 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
SE9600070D0 (sv) * 1996-01-08 1996-01-08 Astra Ab New oral pharmaceutical dosage forms
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US8993599B2 (en) * 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
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WO2005082337A2 (en) * 2004-02-18 2005-09-09 Allergan, Inc. Compositions comprising prodrugs of proton pump inhibitors
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US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
US8541026B2 (en) 2004-09-24 2013-09-24 Abbvie Inc. Sustained release formulations of opioid and nonopioid analgesics
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US20080103169A1 (en) 2006-10-27 2008-05-01 The Curators Of The University Of Missouri Compositions comprising acid labile proton pump inhibiting agents, at least one other pharmaceutically active agent and methods of using same
US20080194307A1 (en) * 2007-02-13 2008-08-14 Jeff Sanger Sports-based game of chance
JP2011512416A (ja) 2008-02-20 2011-04-21 ザ・キュレイターズ・オブ・ザ・ユニバーシティー・オブ・ミズーリ オメプラゾール及びランソプラゾールの組合せと緩衝剤を含んでなる組成物とそれを使用する方法
KR20110079641A (ko) 2008-09-09 2011-07-07 아스트라제네카 아베 제약 조성물을 이를 필요로 하는 환자에게 전달하는 방법
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WO2011080502A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
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Also Published As

Publication number Publication date
NO924650D0 (no) 1992-12-02
FI925767A0 (fi) 1992-12-18
EP0593463A1 (en) 1994-04-27
AP253A (en) 1993-05-03
CZ279434B6 (cs) 1995-04-12
PT98036A (pt) 1992-03-31
MA22198A1 (fr) 1992-04-01
DE69131627T2 (de) 2000-04-27
PL297295A1 (cs) 1992-07-13
JP3049367B2 (ja) 2000-06-05
OA09683A (en) 1993-05-15
IL98472A (en) 1995-08-31
AU8061791A (en) 1992-01-07
NZ238545A (en) 1993-08-26
ATE184602T1 (de) 1999-10-15
EG19752A (en) 1996-01-31
PL166209B1 (pl) 1995-04-28
BG97198A (bg) 1993-12-24
EP0593463B1 (en) 1999-09-15
PL297294A1 (cs) 1992-07-13
DE69131627D1 (de) 1999-10-21
RO110497B1 (ro) 1996-01-30
IL98472A0 (en) 1992-07-15
CN1058213A (zh) 1992-01-29
CA2083606A1 (en) 1991-12-21
LV10269B (en) 1995-10-20
NO924650L (no) 1992-12-02
JPH05507714A (ja) 1993-11-04
CA2083606C (en) 2001-08-21
ES2140391T3 (es) 2000-03-01
AU649456B2 (en) 1994-05-26
FI925767A7 (fi) 1992-12-18
HU9204034D0 (en) 1993-03-29
YU104091A (sh) 1994-01-20
TNSN91050A1 (fr) 1992-10-25
PL165898B1 (pl) 1995-02-28
AP9100286A0 (en) 1991-07-31
LV10269A (lv) 1994-10-20
IE912026A1 (en) 1992-01-01
WO1991019712A1 (en) 1991-12-26
US5430042A (en) 1995-07-04
HUT62882A (en) 1993-06-28
IS3720A7 (is) 1991-12-21

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