CS295191A3 - 2-/4-piperidinyl/-1h-pyrido/4,3-b/indol-1-ones and derived compounds, intermediates and process for preparing thereof - Google Patents

2-/4-piperidinyl/-1h-pyrido/4,3-b/indol-1-ones and derived compounds, intermediates and process for preparing thereof Download PDF

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Publication number
CS295191A3
CS295191A3 CS912951A CS295191A CS295191A3 CS 295191 A3 CS295191 A3 CS 295191A3 CS 912951 A CS912951 A CS 912951A CS 295191 A CS295191 A CS 295191A CS 295191 A3 CS295191 A3 CS 295191A3
Authority
CS
Czechoslovakia
Prior art keywords
lower alkyl
phenyl
alkyl group
groups
group
Prior art date
Application number
CS912951A
Other languages
Czech (cs)
English (en)
Inventor
Lawrence Leo Martin
Denise M Flanagan
Joseph Francis Payack
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of CS295191A3 publication Critical patent/CS295191A3/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
CS912951A 1990-09-27 1991-09-26 2-/4-piperidinyl/-1h-pyrido/4,3-b/indol-1-ones and derived compounds, intermediates and process for preparing thereof CS295191A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07588870 US5102889B1 (en) 1990-09-27 1990-09-27 2-(4-piperidinyl)-1h-pyrido(4,3-b)indol-1-ones and related compounds

Publications (1)

Publication Number Publication Date
CS295191A3 true CS295191A3 (en) 1992-04-15

Family

ID=24355647

Family Applications (1)

Application Number Title Priority Date Filing Date
CS912951A CS295191A3 (en) 1990-09-27 1991-09-26 2-/4-piperidinyl/-1h-pyrido/4,3-b/indol-1-ones and derived compounds, intermediates and process for preparing thereof

Country Status (22)

Country Link
US (1) US5102889B1 (de)
EP (1) EP0481254B1 (de)
JP (1) JP3241762B2 (de)
KR (1) KR100210338B1 (de)
AT (1) ATE132148T1 (de)
AU (1) AU8475091A (de)
CA (1) CA2052424C (de)
CS (1) CS295191A3 (de)
DE (1) DE69115833T2 (de)
DK (1) DK0481254T3 (de)
ES (1) ES2082078T3 (de)
FI (1) FI914503A7 (de)
GR (1) GR3018746T3 (de)
HU (1) HUT59405A (de)
IE (1) IE72156B1 (de)
IL (3) IL99579A (de)
NO (1) NO913777L (de)
NZ (2) NZ239934A (de)
PT (1) PT99074B (de)
TW (1) TW199159B (de)
YU (1) YU158691A (de)
ZA (1) ZA917691B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4975445A (en) * 1989-12-06 1990-12-04 Warner-Lambert Company Substituted cyclohexenes as central nervous system agents
JP2004502642A (ja) * 2000-02-11 2004-01-29 ブリストル−マイヤーズ　スクイブ　カンパニー カンナビノイドレセプターモジュレーター、それらの製造方法、および呼吸系および非呼吸系疾患の処置のためのカンナビノイドレセプターモジュレーターの使用
KR102570307B1 (ko) * 2016-10-31 2023-08-25 주식회사 이엔에프테크놀로지 식각 조성물
CN109400617A (zh) * 2019-01-09 2019-03-01 湖北大学 一种新型吲哚并吡喃酮骨架化合物及其制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR205452A1 (es) * 1973-12-06 1976-05-07 Endo Lab Metodo para preparar nuevos trans-2, 3, 4, 4a, 5, 9b-hexahidro-5-fenil-1h-pirido(4,3-b) indoles
DE2557341A1 (de) * 1975-12-19 1977-06-30 Hoechst Ag Basisch substituierte indolderivate und verfahren zu ihrer herstellung
US4432978A (en) * 1979-07-30 1984-02-21 Pfizer Inc. Hexahydro-trans-pyridoindole
US4252811A (en) * 1979-07-30 1981-02-24 Pfizer Inc. Hexahydro-trans-pyridoindole neuroleptic agents
FR2619111B1 (fr) * 1987-08-07 1991-01-11 Synthelabo Derives de (piperidinyl-4)methyl-2 tetrahydro-1,2,3,4 9h-pyrido (3,4-b) indole, leur preparation et leur application en therapeutique
NZ226032A (en) * 1987-09-03 1991-12-23 Glaxo Group Ltd 2-(imidazolylmethyl)-pyrido or-azepino(4,3-b)indole-1(2h)-one derivatives; preparatory processes and pharmaceutical compositions
IL91167A (en) * 1988-08-02 1993-06-10 Glaxo Group Ltd Substituted 2-(imidazolymethyl)-pyrido- (and azepino-) indol-1-one derivatives, their preparation and pharmaceutical compositions containing them
GB8904551D0 (en) * 1989-02-28 1989-04-12 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
IL99579A0 (en) 1992-08-18
EP0481254A3 (de) 1992-05-06
NZ248705A (en) 1994-09-27
HU913081D0 (en) 1992-01-28
EP0481254B1 (de) 1995-12-27
ATE132148T1 (de) 1996-01-15
IL113439A (en) 1997-03-18
TW199159B (de) 1993-02-01
DE69115833T2 (de) 1996-06-05
ZA917691B (en) 1992-05-27
NO913777L (no) 1992-03-30
JP3241762B2 (ja) 2001-12-25
IL99579A (en) 1999-04-11
DK0481254T3 (da) 1996-04-29
NZ239934A (en) 1994-09-27
IL113439A0 (en) 1995-07-31
NO913777D0 (no) 1991-09-26
PT99074B (pt) 1999-02-26
CA2052424A1 (en) 1992-03-28
KR100210338B1 (ko) 1999-07-15
CA2052424C (en) 2001-12-25
JPH04282381A (ja) 1992-10-07
IE913388A1 (en) 1992-04-08
KR920006355A (ko) 1992-04-27
FI914503L (fi) 1992-03-28
GR3018746T3 (en) 1996-04-30
FI914503A0 (fi) 1991-09-25
US5102889B1 (en) 1993-05-11
ES2082078T3 (es) 1996-03-16
HUT59405A (en) 1992-05-28
AU8475091A (en) 1992-04-02
FI914503A7 (fi) 1992-03-28
EP0481254A2 (de) 1992-04-22
US5102889A (en) 1992-04-07
DE69115833D1 (de) 1996-02-08
PT99074A (pt) 1992-08-31
YU158691A (sh) 1994-06-10
IE72156B1 (en) 1997-03-26

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