CU20100047A7 - DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3 - Google Patents

DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3

Info

Publication number
CU20100047A7
CU20100047A7 CU20100047A CU20100047A CU20100047A7 CU 20100047 A7 CU20100047 A7 CU 20100047A7 CU 20100047 A CU20100047 A CU 20100047A CU 20100047 A CU20100047 A CU 20100047A CU 20100047 A7 CU20100047 A7 CU 20100047A7
Authority
CU
Cuba
Prior art keywords
histamine
isoindolinona
azaciclilisoquinolinona
antagonists
derivatives
Prior art date
Application number
CU20100047A
Other languages
Spanish (es)
Inventor
Dahul Zhou
Albert Jean Robichaud
Jonathan Laird Gross
Original Assignee
Wyeth Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Llc filed Critical Wyeth Llc
Priority to CU20100047A priority Critical patent/CU20100047A7/en
Publication of CU20100047A7 publication Critical patent/CU20100047A7/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención proporciona un compuesto de fórmula I y su uso para el tratamiento de un trastorno del sistema nervioso central relacionado con, o que se ve afectado por, el receptor de la histamina-3.The present invention provides a compound of formula I and its use for the treatment of a central nervous system disorder related to, or that is affected by, the histamine-3 receptor.

CU20100047A 2010-03-12 2010-03-12 DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3 CU20100047A7 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20100047A CU20100047A7 (en) 2010-03-12 2010-03-12 DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20100047A CU20100047A7 (en) 2010-03-12 2010-03-12 DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3

Publications (1)

Publication Number Publication Date
CU20100047A7 true CU20100047A7 (en) 2011-10-05

Family

ID=45000065

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20100047A CU20100047A7 (en) 2010-03-12 2010-03-12 DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3

Country Status (1)

Country Link
CU (1) CU20100047A7 (en)

Similar Documents

Publication Publication Date Title
CO6300955A2 (en) DERIVATIVES OF ISOQUINOLINILO AND ISOINDOLINILO AS ANTAGONISTS OF HISTAMINE -3
DOP2010000078A (en) DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3
CR20150296A (en) NEWS DERIVED FROM BENCIMIDAZOL AS ANTAGONISTS OF EP4
CL2016000341A1 (en) Methods to treat myositis by sporadic inclusion bodies
CR20150425A (en) AZABENCIMIDAZOL COMPOUNDS AS INHIBITORS OF THE ISOZIMAS PDE4, FOR THE TREATMENT OF THE CENTRAL NERVOUS SYSTEM AND OTHER DISORDERS
CR20140161A (en) BENZILINDAZOLS REPLACED FOR USE AS INHIBITORS OF QUINASA BUB1 IN THE TREATMENT OF HYPERPROLIFERATIVE DISEASES
CR20140166A (en) COMPOUNDS OF (ITS) ARILCICLOPROPILAMINE AS INHIBITORS OF LSD1
CR20210079A (en) SULFAMOILARYLAMIDES AND THEIR USE AS MEDICINES FOR THE TREATMENT OF HEPATITIS B
PE20150669A1 (en) BENZAMIDE DERIVATIVES FOR INHIBITION OF THE ACTIVITY OF ABL1, ABL2 AND BCR-ABL1
UY35906A (en) NEWS DERIVED FROM BENCIMIDAZOL AS LIGANDOS OF EP4
ECSP14002542A (en) NOVEL 2HINDAZOLES AS EP2 RECEPTOR ANTAGONISTS
PA8790101A1 (en) DERIVATIVES OF AMINOALQUILAZOL AS ANTAGONISTS OF HISTAMINE-3
CL2016000325A1 (en) Track antagonists to treat sleep disorders due to phase change
DOP2015000176A (en) AZETIDINYLOXYPHENYLPIRROLIDINE COMPOUNDS
PA8781601A1 (en) "DERIVATIVES OF AZACICLILBENZAMIDE AS ANTAGONISTS OF HISTAMINE-3
BR112016012552A8 (en) chromone derivative as a dopamine d3 receptor antagonist, its use and pharmaceutical composition
ECSP088176A (en) DERIVATIVES OF AZINIL-3-SULFONYLINDAZOL AS LIGANDS DE5-HYDROXYTHYRIPTAMINE-6
CR9734A (en) DERIVATIVES OF 3-SULFONYLINDAZOL REPLACED AS 5-HYDROXYTHYRIPTAMINE-6 LIGANDS
UY31646A1 (en) USE OF SUBSTITUTED PHENYLIMIDAZOLIDINS TO PRODUCE MEDICINES FOR THE TREATMENT OF METABOLIC SYNDROME
ECSP088930A (en) DERIVATIVES OF BENZOXAZOL AND BENZOTIAZOL AS LIGANDOS OF
ECSP088789A (en) DERIVATIVES OF SULFONIL-3-HETEROCICLILINDAZOL AS 5-HYDROXYTHYRIPTAMINE-6 LIGANDS
CU20100047A7 (en) DERIVATIVES OF AZACICLILISOQUINOLINONA E-ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3
CU20100045A7 (en) DERIVATIVES OF ISOQUINOLINILO AND ISOINDOLINILO AS ANTAGONISTS OF HISTAMINE-3
SV2010003508A (en) DERIVATIVES OF AZACICLILISOQUINOLINONA E- ISOINDOLINONA AS ANTAGONISTS OF HISTAMINE-3
UY32191A (en) IMINOPIRIDINE DERIVATIVES AND USE OF THE SAME