CU20100087A7 - SOME DERIVATIVES OF 2-PIRAZINONA AND ITS USE AS INHIBITORS OF ELASTASA DE LOS NEUTRÓFILOS - Google Patents

SOME DERIVATIVES OF 2-PIRAZINONA AND ITS USE AS INHIBITORS OF ELASTASA DE LOS NEUTRÓFILOS

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Publication number
CU20100087A7
CU20100087A7 CU20100087A CU20100087A CU20100087A7 CU 20100087 A7 CU20100087 A7 CU 20100087A7 CU 20100087 A CU20100087 A CU 20100087A CU 20100087 A CU20100087 A CU 20100087A CU 20100087 A7 CU20100087 A7 CU 20100087A7
Authority
CU
Cuba
Prior art keywords
inhibitors
derivatives
pirazinona
neutrófilos
elastasa
Prior art date
Application number
CU20100087A
Other languages
Spanish (es)
Inventor
Antonios Nikitidis
Af Rosenschoeld Magnus Munck
Michael Lundkvist
Hans Loenn
Martin Lindsjoe
David Chapman
John Pavey
Debra Ainge
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to CU20100087A priority Critical patent/CU20100087A7/en
Publication of CU20100087A7 publication Critical patent/CU20100087A7/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención proporciona ciertos nuevos derivados de 6-heteroaril-5-metil-3-oxo-4-[3-(trifluorometil)fenil]-3,4-dihidropirazina-2-carboxamida y sales farmacéuticamente aceptables de los mismos y formas particulares de los mismos; junto con procesos para su preparación, composiciones farmacéuticas que los contienen y su uso en terapia. Los compuestos son inhibidores de la estasa de los neutrófilos humanos.The invention provides certain novel derivatives of 6-heteroaryl-5-methyl-3-oxo-4- [3- (trifluoromethyl) phenyl] -3,4-dihydropyrazine-2-carboxamide and pharmaceutically acceptable salts thereof and particular forms of the same; together with processes for its preparation, pharmaceutical compositions containing them and their use in therapy. The compounds are inhibitors of human neutrophil stase.

CU20100087A 2010-05-05 2010-05-05 SOME DERIVATIVES OF 2-PIRAZINONA AND ITS USE AS INHIBITORS OF ELASTASA DE LOS NEUTRÓFILOS CU20100087A7 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20100087A CU20100087A7 (en) 2010-05-05 2010-05-05 SOME DERIVATIVES OF 2-PIRAZINONA AND ITS USE AS INHIBITORS OF ELASTASA DE LOS NEUTRÓFILOS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20100087A CU20100087A7 (en) 2010-05-05 2010-05-05 SOME DERIVATIVES OF 2-PIRAZINONA AND ITS USE AS INHIBITORS OF ELASTASA DE LOS NEUTRÓFILOS

Publications (1)

Publication Number Publication Date
CU20100087A7 true CU20100087A7 (en) 2011-10-05

Family

ID=45000082

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20100087A CU20100087A7 (en) 2010-05-05 2010-05-05 SOME DERIVATIVES OF 2-PIRAZINONA AND ITS USE AS INHIBITORS OF ELASTASA DE LOS NEUTRÓFILOS

Country Status (1)

Country Link
CU (1) CU20100087A7 (en)

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