CU20100148A7 - 3H- [1,2,3] TRIAZOLO [4,5-D] PIRIMIDINE COMPOUNDS, THEIR USE AS INHIBITORS OF MTOR QUINASA AND PI3 QUINASA AND THEIR SYNTHESIS - Google Patents
3H- [1,2,3] TRIAZOLO [4,5-D] PIRIMIDINE COMPOUNDS, THEIR USE AS INHIBITORS OF MTOR QUINASA AND PI3 QUINASA AND THEIR SYNTHESISInfo
- Publication number
- CU20100148A7 CU20100148A7 CU20100148A CU20100148A CU20100148A7 CU 20100148 A7 CU20100148 A7 CU 20100148A7 CU 20100148 A CU20100148 A CU 20100148A CU 20100148 A CU20100148 A CU 20100148A CU 20100148 A7 CU20100148 A7 CU 20100148A7
- Authority
- CU
- Cuba
- Prior art keywords
- quinasa
- triazolo
- compounds
- mtor
- inhibitors
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 101150097381 Mtor gene Proteins 0.000 title 1
- 102100023085 Serine/threonine-protein kinase mTOR Human genes 0.000 title 1
- 230000015572 biosynthetic process Effects 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
- GIIGHSIIKVOWKZ-UHFFFAOYSA-N 2h-triazolo[4,5-d]pyrimidine Chemical class N1=CN=CC2=NNN=C21 GIIGHSIIKVOWKZ-UHFFFAOYSA-N 0.000 abstract 1
- 239000000470 constituent Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La invención se refiere a compuestos de 3H-[1,2,3]triazolo[4,5-d]pirimidina de fórmula 1: o a una sal farmacéuticamente aceptable de los mismos, en la que las variables constituyentes son como se definen en el presente documento, a composiciones que comprenden los compuestos y a procedimientos para fabricar y usar los compuestos.The invention relates to 3H- [1,2,3] triazolo [4,5-d] pyrimidine compounds of formula 1: or a pharmaceutically acceptable salt thereof, in which the constituent variables are as defined in the herein, to compositions comprising the compounds and to methods for manufacturing and using the compounds.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20100148A CU20100148A7 (en) | 2010-07-15 | 2010-07-15 | 3H- [1,2,3] TRIAZOLO [4,5-D] PIRIMIDINE COMPOUNDS, THEIR USE AS INHIBITORS OF MTOR QUINASA AND PI3 QUINASA AND THEIR SYNTHESIS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20100148A CU20100148A7 (en) | 2010-07-15 | 2010-07-15 | 3H- [1,2,3] TRIAZOLO [4,5-D] PIRIMIDINE COMPOUNDS, THEIR USE AS INHIBITORS OF MTOR QUINASA AND PI3 QUINASA AND THEIR SYNTHESIS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU20100148A7 true CU20100148A7 (en) | 2011-10-31 |
Family
ID=45000116
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU20100148A CU20100148A7 (en) | 2010-07-15 | 2010-07-15 | 3H- [1,2,3] TRIAZOLO [4,5-D] PIRIMIDINE COMPOUNDS, THEIR USE AS INHIBITORS OF MTOR QUINASA AND PI3 QUINASA AND THEIR SYNTHESIS |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU20100148A7 (en) |
-
2010
- 2010-07-15 CU CU20100148A patent/CU20100148A7/en unknown
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