CU20110012A7 - HETEROARILO DERIVATIVES AS DGAT1 INHIBITORS - Google Patents
HETEROARILO DERIVATIVES AS DGAT1 INHIBITORSInfo
- Publication number
- CU20110012A7 CU20110012A7 CU20110012A CU20110012A CU20110012A7 CU 20110012 A7 CU20110012 A7 CU 20110012A7 CU 20110012 A CU20110012 A CU 20110012A CU 20110012 A CU20110012 A CU 20110012A CU 20110012 A7 CU20110012 A7 CU 20110012A7
- Authority
- CU
- Cuba
- Prior art keywords
- heteroarilo
- derivatives
- treatment
- dgat1 inhibitors
- disorders
- Prior art date
Links
- 229940127193 DGAT1 inhibitor Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 102100036869 Diacylglycerol O-acyltransferase 1 Human genes 0.000 abstract 1
- 101000927974 Homo sapiens Diacylglycerol O-acyltransferase 1 Proteins 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 208000030159 metabolic disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La invención se refiere a los compuestos de la fórmula (I): ESPACIO PARA LA FÓRMULA en donde A es un heteroarilo opcionalmente sustituido, útiles para el tratamiento de los trastornos mediados por acil-transferasa de acil-CoA-diacil-glicerol 1 (DGAT1), por ejemplo, trastornos metabólicos. La invención también proporciona métodos para el tratamiento de estos trastornos, y los compuestos y composiciones etc. para su tratamiento.The invention relates to the compounds of the formula (I): SPACE FOR FORMULA wherein A is an optionally substituted heteroaryl, useful for the treatment of acyl-CoA-diacyl-glycerol-1-acyl-transferase-mediated disorders (DGAT1 ), for example, metabolic disorders. The invention also provides methods for the treatment of these disorders, and the compounds and compositions etc. for your treatment
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20110012A CU20110012A7 (en) | 2011-01-17 | 2011-01-17 | HETEROARILO DERIVATIVES AS DGAT1 INHIBITORS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20110012A CU20110012A7 (en) | 2011-01-17 | 2011-01-17 | HETEROARILO DERIVATIVES AS DGAT1 INHIBITORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU20110012A7 true CU20110012A7 (en) | 2011-12-28 |
Family
ID=45508731
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU20110012A CU20110012A7 (en) | 2011-01-17 | 2011-01-17 | HETEROARILO DERIVATIVES AS DGAT1 INHIBITORS |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU20110012A7 (en) |
-
2011
- 2011-01-17 CU CU20110012A patent/CU20110012A7/en unknown
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