CU20120030A7 - USEFUL OXAZINE DERIVATIVES IN THE TREATMENT OF NEUROLOGICAL DISORDERS - Google Patents
USEFUL OXAZINE DERIVATIVES IN THE TREATMENT OF NEUROLOGICAL DISORDERSInfo
- Publication number
- CU20120030A7 CU20120030A7 CU2012000030A CU20120030A CU20120030A7 CU 20120030 A7 CU20120030 A7 CU 20120030A7 CU 2012000030 A CU2012000030 A CU 2012000030A CU 20120030 A CU20120030 A CU 20120030A CU 20120030 A7 CU20120030 A7 CU 20120030A7
- Authority
- CU
- Cuba
- Prior art keywords
- useful
- treatment
- neurological disorders
- oxazine derivatives
- formula
- Prior art date
Links
- 150000004893 oxazines Chemical class 0.000 title abstract 2
- 208000012902 Nervous system disease Diseases 0.000 title 1
- 208000025966 Neurological disease Diseases 0.000 title 1
- 102100021257 Beta-secretase 1 Human genes 0.000 abstract 1
- 101000894895 Homo sapiens Beta-secretase 1 Proteins 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se dan a conocer derivados de oxazina de la fórmula (I): ESPACIO PARA LA FÓRMULA los cuales tienen una actividad inhibidora de BACE, en donde todas las variables son como se definen en la memoria descriptiva, en forma libre o en forma de sal, sus métodos de preparación, su uso médico y medicamentos que los comprenden.Oxazine derivatives of the formula (I) are disclosed: SPACE FOR THE FORMULA which have a BACE inhibitory activity, where all the variables are as defined in the specification, in free form or in salt form, its methods of preparation, its medical use and medicines that comprise them.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2010/060718 WO2011009943A1 (en) | 2009-07-24 | 2010-07-23 | Oxazine derivatives and their use as bace inhibitors for the treatment of neurological disorders |
| US201161435088P | 2011-01-21 | 2011-01-21 | |
| PCT/CN2011/077119 WO2012006953A1 (en) | 2010-07-13 | 2011-07-13 | Oxazine derivatives and their use in the treatment of neurological disorders |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CU20120030A7 true CU20120030A7 (en) | 2013-05-31 |
| CU24047B1 CU24047B1 (en) | 2014-12-26 |
Family
ID=53365646
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU2012000030A CU24047B1 (en) | 2010-07-23 | 2012-02-23 | USEFUL OXAZINE DERIVATIVES IN THE TREATMENT OF NEUROLOGICAL DISORDERS |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU24047B1 (en) |
-
2012
- 2012-02-23 CU CU2012000030A patent/CU24047B1/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CU24047B1 (en) | 2014-12-26 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ECSP12011692A (en) | DERIVATIVES OF OXAZINE AND ITS USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS | |
| CU20120099A7 (en) | DERIVATIVES OF PIRAZINA AND ITS USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS | |
| CO6491058A2 (en) | DERIVATIVES OF OXAZINE AND ITS USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS | |
| GT201400063A (en) | BENZILINDAZOLS REPLACED FOR USE AS INHIBITORS OF QUINASA BUB1 IN THE TREATMENT OF HYPERPROLIFERATIVE DISEASES | |
| UY34657A (en) | ? MACROCYCLIC DERIVATIVES FOR THE TREATMENT OF DISEASES ?. | |
| CY1116424T1 (en) | ADENINIS PRODUCTION AS RISK RISK | |
| CU20140048A7 (en) | NEW PURINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER AND NEURODEGENERATIVE DISORDERS | |
| GT201400036A (en) | COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF THE QUINASE C - KIT | |
| UY33883A (en) | NEW HETEROCYCLIC DERIVATIVES | |
| UY35827A (en) | TRIAZOLOPIRAZINE DERIVATIVES AS INHIBITORS OF THE BRD4 PROTEIN | |
| PT2935303T (en) | 4'-FLUORO-NUCLEOSIDES, 4'-FLUORO-NUCLEOTIDES AND THEIR ANALOGS FOR THE TREATMENT OF HCV | |
| MX2015003140A (en) | Formulations of enzalutamide. | |
| UY34750A (en) | ? COMPOUNDS FOR HIV TREATMENT, COMPOSITIONS, PREPARATION METHODS, INTERMEDIARIES AND THERAPEUTIC METHODS ?. | |
| CL2016001895A1 (en) | Compounds | |
| MX374399B (en) | COMPOSITIONS AND THEIR USES FOR TREATING AND PREVENTING HUNTINGTON'S DISEASE. | |
| CR20150326A (en) | AUTOTAXIN INHIBITORS | |
| CR20130588A (en) | HALOGENOALQUIL-1,3-OXAZINAS AS INHIBITORS OF THE BACE1 AND / OR BACE 2 | |
| BR112014013843A2 (en) | use of devices for the treatment of neurological diseases | |
| ECSP16008797A (en) | DERIVATIVES OF HETEROBICICLOARIL AS RORC2 INHIBITORS AND METHODS OF USE OF THE SAME | |
| UY35747A (en) | SUBSTITUTED DERIVATIVES OF PHENYLALANINE | |
| DOP2016000170A (en) | COMPOUNDS DERIVED FROM HYDROXIFORMAMIDE AND USES OF THE SAME | |
| CR20160290A (en) | AUTOTAXINE TETRACYCLIC INHIBITORS | |
| CY1114757T1 (en) | OXAZINE PRODUCTS AND THEIR USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS | |
| UY35745A (en) | SUBSTITUTED DERIVATIVES OF PHENYLALANINE | |
| UA112488C2 (en) | THREE (HETERO) ARILPYRAZOLES AND THEIR APPLICATIONS |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant of patent | ||
| FD | Lapse (for not paying fees) |