CU20140022A7 - DERIVATIVES OF BICYCLIC HETEROCICLES FOR THE TREATMENT OF PULMONARY ARTERIAL HYPERTENSION - Google Patents

DERIVATIVES OF BICYCLIC HETEROCICLES FOR THE TREATMENT OF PULMONARY ARTERIAL HYPERTENSION

Info

Publication number
CU20140022A7
CU20140022A7 CU2014000022A CU20140022A CU20140022A7 CU 20140022 A7 CU20140022 A7 CU 20140022A7 CU 2014000022 A CU2014000022 A CU 2014000022A CU 20140022 A CU20140022 A CU 20140022A CU 20140022 A7 CU20140022 A7 CU 20140022A7
Authority
CU
Cuba
Prior art keywords
derivatives
bicyclic
heterocicles
treatment
arterial hypertension
Prior art date
Application number
CU2014000022A
Other languages
Spanish (es)
Inventor
Ian Bruce
Sylvie Chamon
Stephen Paul Collingwood
Pascal Furet
Vikki Furminger
Sara Lewis
Jon Christopher Loren
Valentina Molteni
Alex Michael Saunders
Duncan Shaw
Lilya Sviridenko
Christopher Thomson
Vince Yeh
Diana Janus
Ryan West
Original Assignee
Irm Llc
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/IB2012/054501 external-priority patent/WO2013030802A1/en
Application filed by Irm Llc, Novartis Ag filed Critical Irm Llc
Publication of CU20140022A7 publication Critical patent/CU20140022A7/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Derivados de heterociclos bicíclicos de la fórmula I útiles en la inhibición de la actividad biológica mediada por el receptor PDGF. en donde A es Y R^1, R^1a, R^2, R^3, R^4, R^5, R^6 y X son como se definen en la presente.Derivatives of bicyclic heterocycles of the formula I useful in inhibiting the biological activity mediated by the PDGF receptor. wherein A is Y R ^ 1, R ^ 1a, R ^ 2, R ^ 3, R ^ 4, R ^ 5, R ^ 6 and X are as defined herein.

CU2014000022A 2012-08-06 2014-02-27 DERIVATIVES OF BICYCLIC HETEROCICLES FOR THE TREATMENT OF PULMONARY ARTERIAL HYPERTENSION CU20140022A7 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261680119P 2012-08-06 2012-08-06
PCT/IB2012/054501 WO2013030802A1 (en) 2011-09-01 2012-08-31 Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension

Publications (1)

Publication Number Publication Date
CU20140022A7 true CU20140022A7 (en) 2014-05-27

Family

ID=52394768

Family Applications (1)

Application Number Title Priority Date Filing Date
CU2014000022A CU20140022A7 (en) 2012-08-06 2014-02-27 DERIVATIVES OF BICYCLIC HETEROCICLES FOR THE TREATMENT OF PULMONARY ARTERIAL HYPERTENSION

Country Status (1)

Country Link
CU (1) CU20140022A7 (en)

Similar Documents

Publication Publication Date Title
CR20140099A (en) DERIVATIVES OF BICYCLIC HETEROCICLES FOR THE TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
DOP2013000027A (en) DERIVATIVES OF TETRAHIDRO-PIRIDO-PIRIMIDINA
UY33943A (en) SCIROCYCLIC DERIVATIVES OF ISOXAZOLINE AS ANTIPARASITARY AGENTS.
UY34051A (en) PIRROLOTRIAZINONA DERIVATIVES AS PI3K INHIBITORS
CO6771441A2 (en) Triazolopyridine compounds as pim kinase inhibitors
UY34657A (en) ? MACROCYCLIC DERIVATIVES FOR THE TREATMENT OF DISEASES ?.
UY34472A (en) MODIFIED DERIVATIVES OF 4-PHENYL-PYRIDINE
CR20140161A (en) BENZILINDAZOLS REPLACED FOR USE AS INHIBITORS OF QUINASA BUB1 IN THE TREATMENT OF HYPERPROLIFERATIVE DISEASES
CO7151548A2 (en) Macrocyclic picolinamides as fungicides
CO7071122A2 (en) 1,3-oxazines as inhibitors of bace1 and / or bace2
ECSP12011692A (en) DERIVATIVES OF OXAZINE AND ITS USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS
CO6311079A2 (en) AMINODIHYDROTIAZINE DERIVATIVES AS INHIBITORS OF THE BACE ENZYME FOR THE TREATMENT OF ALZHEIMER'S DISEASE
UY34602A (en) Derivatives of benzimidazolyl- and imidazopyridinyl-methylamine?
UY34352A (en) 3-PIRIMIDIN-4-IL-OXAZOLIDIN-2-ONAS AS INHIBITORS OF THE MUTANT HDI
CR20140084A (en) DERIVATIVES OF 2-AMINO-4- (PIRIDIN-2-IL) -5,6-DIHIDRO-4H-1,3-OXAZINE AND ITS USE AS BACE-1 AND / OR BACE-2 INHIBITORS
UY34333A (en) ? METHODS AND COMPOSITIONS FOR WEED CONTROL, AND METHODS TO REDUCE THE EXPRESSION OF ENZYME DHPS?
BR112013022813A2 (en) diaminocarbonitrile pyrimidines and substituted diaminocarboxamide, compositions thereof and methods of treating them
UY34201A (en) AZAINDOL COMPOUNDS AND METHODS FOR HIV TREATMENT.
BR112013007850A2 (en) 1,2-dihydro-4-hydroxy-2-oxo-quinoline-3-carboxanilides as ahr activators
EA201591024A1 (en) DIMER CONNECTIONS
UY33976A (en) DERIVATIVES OF PIRAZOLO-PYRIMIDINE.
CR20140564A (en) PIRIMIDINONE DERIVATIVES AS ANTIMALARIAN AGENTS
LT2782602T (en) NUCLEOTIDE DIMS0-150 FOR THE TREATMENT OF LOWER ACTIVE OPERATIVE COLOLIS
UY34043A (en) ISOXAZOLINS AS THERAPEUTIC AGENTS
EP2688901A4 (en) HEMMER OF 17-BETA-HSD1, 17-BETA-HSD3 AND 17BETA-HSD10