CU20140134A7 - NOVEDOSAS N-PIRIDINIL CYCLIC AMIDAS REPLACED AS QUINASE INHIBITORS - Google Patents
NOVEDOSAS N-PIRIDINIL CYCLIC AMIDAS REPLACED AS QUINASE INHIBITORSInfo
- Publication number
- CU20140134A7 CU20140134A7 CU2014000134A CU20140134A CU20140134A7 CU 20140134 A7 CU20140134 A7 CU 20140134A7 CU 2014000134 A CU2014000134 A CU 2014000134A CU 20140134 A CU20140134 A CU 20140134A CU 20140134 A7 CU20140134 A7 CU 20140134A7
- Authority
- CU
- Cuba
- Prior art keywords
- novedosas
- piridinil
- amidas
- cyclic
- replaced
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona un compuesto de la fórmula (A): (A) como se describe en la presente, y sales, enantiomeros, rotámeros, tautómeros, o racemátos de los mismos farmacéuticamente aceptables. También se proporcionan métodos de tratar una enfermedad o condición mediada por la quinasa PIM utilizando compuestos de la Fórmula I, y composiciones farmacéuticas que comprenden tales compuestos.The present invention provides a compound of the formula (A): (A) as described herein, and pharmaceutically acceptable salts, enantiomers, rotamers, tautomers, or racemates thereof. Methods of treating a disease or condition mediated by PIM kinase using compounds of Formula I, and pharmaceutical compositions comprising such compounds are also provided.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261695533P | 2012-08-31 | 2012-08-31 | |
| PCT/IB2013/054145 WO2013175388A1 (en) | 2012-05-21 | 2013-05-20 | Novel ring-substituted n-pyridinyl amides as kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU20140134A7 true CU20140134A7 (en) | 2015-03-30 |
Family
ID=53365659
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU2014000134A CU20140134A7 (en) | 2012-08-31 | 2014-11-21 | NOVEDOSAS N-PIRIDINIL CYCLIC AMIDAS REPLACED AS QUINASE INHIBITORS |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU20140134A7 (en) |
-
2014
- 2014-11-21 CU CU2014000134A patent/CU20140134A7/en unknown
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