CU20160019A7 - POLYMORPH OF INHIBITORS OF TIROSINA KINASA DEL BAZO (SYK), METHODS OF PREPRATION AND COMPOSITIONS - Google Patents
POLYMORPH OF INHIBITORS OF TIROSINA KINASA DEL BAZO (SYK), METHODS OF PREPRATION AND COMPOSITIONSInfo
- Publication number
- CU20160019A7 CU20160019A7 CUP2016000019A CU20160019A CU20160019A7 CU 20160019 A7 CU20160019 A7 CU 20160019A7 CU P2016000019 A CUP2016000019 A CU P2016000019A CU 20160019 A CU20160019 A CU 20160019A CU 20160019 A7 CU20160019 A7 CU 20160019A7
- Authority
- CU
- Cuba
- Prior art keywords
- polymorph
- compositions
- syk
- methods
- tirosina
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- OUYCCCASQSFEME-QMMMGPOBSA-N L-tyrosine Chemical compound OC(=O)[C@@H](N)CC1=CC=C(O)C=C1 OUYCCCASQSFEME-QMMMGPOBSA-N 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- OUYCCCASQSFEME-UHFFFAOYSA-N tyrosine Natural products OC(=O)C(N)CC1=CC=C(O)C=C1 OUYCCCASQSFEME-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000004022 Protein-Tyrosine Kinases Human genes 0.000 abstract 1
- 108090000412 Protein-Tyrosine Kinases Proteins 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000004968 inflammatory condition Effects 0.000 abstract 1
- 210000000952 spleen Anatomy 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente divulgación se refiere a polimorfos y composiciones farmaceúticas de polimorfo de compuestos que inhiben la activdad de tirosina quinasa del bazo (Syk, por sus siglas en inglés). la divulgación también se refiere a métodos para preparar tales polimorfos y composiciones farmaceúticas de polimorfo, y el uso de tales polimorfos y composiciones farmaceúticas en el tratamiento de sujetos con diversas enfermedades, que incluyen cácncer y condiciones inflamatorias.The present disclosure relates to polymorphs and pharmaceutical compositions of polymorph of compounds that inhibit the tyrosine kinase activity of the spleen (Syk). The disclosure also relates to methods for preparing such polymorphs and pharmaceutical polymorph compositions, and the use of such polymorphs and pharmaceutical compositions in the treatment of subjects with various diseases, including cancer and inflammatory conditions.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201313618660A | 2013-07-30 | 2013-07-30 | |
| PCT/US2014/048733 WO2015017460A1 (en) | 2013-07-30 | 2014-07-29 | Polymorph of syk inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU20160019A7 true CU20160019A7 (en) | 2016-07-29 |
Family
ID=56565036
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CUP2016000019A CU20160019A7 (en) | 2013-07-30 | 2016-02-01 | POLYMORPH OF INHIBITORS OF TIROSINA KINASA DEL BAZO (SYK), METHODS OF PREPRATION AND COMPOSITIONS |
| CUP2016000018A CU20160018A7 (en) | 2013-07-30 | 2016-02-01 | PHARMACEUTICAL COMPOSITIONS OF COMPOUNDS THAT INHIBIT THE ACTIVITY OF TYROSINE KINASE AND ITS PREPARATION METHODS |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CUP2016000018A CU20160018A7 (en) | 2013-07-30 | 2016-02-01 | PHARMACEUTICAL COMPOSITIONS OF COMPOUNDS THAT INHIBIT THE ACTIVITY OF TYROSINE KINASE AND ITS PREPARATION METHODS |
Country Status (1)
| Country | Link |
|---|---|
| CU (2) | CU20160019A7 (en) |
-
2016
- 2016-02-01 CU CUP2016000019A patent/CU20160019A7/en unknown
- 2016-02-01 CU CUP2016000018A patent/CU20160018A7/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CU20160018A7 (en) | 2016-11-29 |
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