CU20170078A7 - DERIVADOS SUSTITUIDOS DE N-(4-(2-(FENILAMINO)-(1,2,4)-TRIAZOLO (1,5-a) PIRIDIN-7-IL)-FENIL)-2-(FENIL)-PROPANAMIDA ÚTILES PARA EL TRATAMIENTO DEL CÁNCER - Google Patents

DERIVADOS SUSTITUIDOS DE N-(4-(2-(FENILAMINO)-(1,2,4)-TRIAZOLO (1,5-a) PIRIDIN-7-IL)-FENIL)-2-(FENIL)-PROPANAMIDA ÚTILES PARA EL TRATAMIENTO DEL CÁNCER

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Publication number
CU20170078A7
CU20170078A7 CUP2017000078A CU20170078A CU20170078A7 CU 20170078 A7 CU20170078 A7 CU 20170078A7 CU P2017000078 A CUP2017000078 A CU P2017000078A CU 20170078 A CU20170078 A CU 20170078A CU 20170078 A7 CU20170078 A7 CU 20170078A7
Authority
CU
Cuba
Prior art keywords
phenyl
inappropriate cellular
propanamide
triazolo
useful
Prior art date
Application number
CUP2017000078A
Other languages
English (en)
Spanish (es)
Inventor
Ursula Krenz
Dr Hans-Georg Lerchen
Dr Philip Lienau
Dr Ulrich Lücking
Dr Volker Schulze
Dr Gerhard Siemeister
Dr Antje Margret Wengner
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of CU20170078A7 publication Critical patent/CU20170078A7/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
CUP2017000078A 2014-12-09 2015-12-07 DERIVADOS SUSTITUIDOS DE N-(4-(2-(FENILAMINO)-(1,2,4)-TRIAZOLO (1,5-a) PIRIDIN-7-IL)-FENIL)-2-(FENIL)-PROPANAMIDA ÚTILES PARA EL TRATAMIENTO DEL CÁNCER CU20170078A7 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14196859 2014-12-09
PCT/EP2015/078871 WO2016091825A1 (fr) 2014-12-09 2015-12-07 Composés pour le traitement d'un cancer

Publications (1)

Publication Number Publication Date
CU20170078A7 true CU20170078A7 (es) 2017-10-05

Family

ID=52011093

Family Applications (1)

Application Number Title Priority Date Filing Date
CUP2017000078A CU20170078A7 (es) 2014-12-09 2015-12-07 DERIVADOS SUSTITUIDOS DE N-(4-(2-(FENILAMINO)-(1,2,4)-TRIAZOLO (1,5-a) PIRIDIN-7-IL)-FENIL)-2-(FENIL)-PROPANAMIDA ÚTILES PARA EL TRATAMIENTO DEL CÁNCER

Country Status (27)

Country Link
US (1) US20170342064A1 (fr)
EP (1) EP3230285A1 (fr)
JP (1) JP2017537116A (fr)
KR (1) KR20170088872A (fr)
CN (1) CN107001376A (fr)
AR (1) AR102947A1 (fr)
AU (1) AU2015359593A1 (fr)
BR (1) BR112017012317A2 (fr)
CA (1) CA2969902A1 (fr)
CO (1) CO2017005741A2 (fr)
CR (1) CR20170243A (fr)
CU (1) CU20170078A7 (fr)
DO (1) DOP2017000136A (fr)
EA (1) EA201791264A1 (fr)
EC (1) ECSP17036251A (fr)
IL (1) IL252237A0 (fr)
MA (1) MA41136A (fr)
MX (1) MX2017007655A (fr)
NI (1) NI201700072A (fr)
PE (1) PE20170927A1 (fr)
PH (1) PH12017501063A1 (fr)
SG (1) SG11201704684PA (fr)
TN (1) TN2017000241A1 (fr)
TW (1) TW201625565A (fr)
UY (1) UY36421A (fr)
WO (1) WO2016091825A1 (fr)
ZA (1) ZA201704589B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116917467A (zh) * 2021-01-22 2023-10-20 渤健马萨诸塞州股份有限公司 用以增加重组病毒载体滴度的微管去稳定剂添加剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2645031A1 (fr) * 2006-03-07 2007-09-13 Bristol-Myers Squibb Company Composes de promedicament de pyrrolotriazine aniline utiles en tant qu'inhibiteurs de la kinase
UA112096C2 (uk) * 2011-12-12 2016-07-25 Байєр Інтеллектуал Проперті Гмбх Заміщені триазолопіридини та їх застосування як інгібіторів ttk
PE20160156A1 (es) * 2013-06-11 2016-04-20 Bayer Pharma AG Derivados de prodroga de triazolpiridinas sustituidas

Also Published As

Publication number Publication date
BR112017012317A2 (pt) 2018-04-24
MX2017007655A (es) 2017-10-11
UY36421A (es) 2016-06-30
PE20170927A1 (es) 2017-07-13
IL252237A0 (en) 2017-07-31
JP2017537116A (ja) 2017-12-14
CA2969902A1 (fr) 2016-06-16
ZA201704589B (en) 2019-02-27
AU2015359593A1 (en) 2017-06-08
ECSP17036251A (es) 2017-06-30
WO2016091825A1 (fr) 2016-06-16
TW201625565A (zh) 2016-07-16
CO2017005741A2 (es) 2017-08-31
US20170342064A1 (en) 2017-11-30
CR20170243A (es) 2017-07-26
MA41136A (fr) 2017-10-17
EA201791264A1 (ru) 2017-12-29
PH12017501063A1 (en) 2017-12-11
NI201700072A (es) 2017-07-17
KR20170088872A (ko) 2017-08-02
EP3230285A1 (fr) 2017-10-18
SG11201704684PA (en) 2017-07-28
CN107001376A (zh) 2017-08-01
DOP2017000136A (es) 2017-08-31
AR102947A1 (es) 2017-04-05
TN2017000241A1 (en) 2018-10-19

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