CU23533A3 - INHIBITORS OF THE RNA-DEPENDENT RNA POLYMERASE OF THE HEPATITIS C VIRUS AND COMPOSITIONS AND TREATMENTS USING THEM - Google Patents
INHIBITORS OF THE RNA-DEPENDENT RNA POLYMERASE OF THE HEPATITIS C VIRUS AND COMPOSITIONS AND TREATMENTS USING THEMInfo
- Publication number
- CU23533A3 CU23533A3 CU20070041A CU20070041A CU23533A3 CU 23533 A3 CU23533 A3 CU 23533A3 CU 20070041 A CU20070041 A CU 20070041A CU 20070041 A CU20070041 A CU 20070041A CU 23533 A3 CU23533 A3 CU 23533A3
- Authority
- CU
- Cuba
- Prior art keywords
- hepatitis
- virus
- inhibitors
- rna
- treatments
- Prior art date
Links
- 241000711549 Hepacivirus C Species 0.000 title abstract 5
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 238000011282 treatment Methods 0.000 title abstract 2
- 108060004795 Methyltransferase Proteins 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- 102000004190 Enzymes Human genes 0.000 abstract 1
- 108090000790 Enzymes Proteins 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona compuestos de fórmula (4) y sus sales farmacéuticamente aceptables y solvatos, que son útiles como inhibidores de la enzima polimerasa del virus de la Hepatitis C (HCV) y también son útiles para el tratamiento de infecciones por HCV en mamíferos infectados por HCV. La presente invención también proporciona composiciones farmacéuticas que comprenden compuestos de fórmula (4), sus sales farmacéuticamente aceptables y solvatos. Además, la presente invención proporciona compuestos intermedios y métodos útiles en la preparación de compuestos de fórmula (4).The present invention provides compounds of formula (4) and their pharmaceutically acceptable salts and solvates, which are useful as inhibitors of the Hepatitis C virus (HCV) polymerase enzyme and are also useful for the treatment of HCV infections in infected mammals. by HCV. The present invention also provides pharmaceutical compositions comprising compounds of formula (4), their pharmaceutically acceptable salts and solvates. In addition, the present invention provides intermediate compounds and methods useful in the preparation of compounds of formula (4).
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20070041A CU23533A3 (en) | 2007-02-08 | 2007-02-08 | INHIBITORS OF THE RNA-DEPENDENT RNA POLYMERASE OF THE HEPATITIS C VIRUS AND COMPOSITIONS AND TREATMENTS USING THEM |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20070041A CU23533A3 (en) | 2007-02-08 | 2007-02-08 | INHIBITORS OF THE RNA-DEPENDENT RNA POLYMERASE OF THE HEPATITIS C VIRUS AND COMPOSITIONS AND TREATMENTS USING THEM |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU23533A3 true CU23533A3 (en) | 2010-06-17 |
Family
ID=42633313
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU20070041A CU23533A3 (en) | 2007-02-08 | 2007-02-08 | INHIBITORS OF THE RNA-DEPENDENT RNA POLYMERASE OF THE HEPATITIS C VIRUS AND COMPOSITIONS AND TREATMENTS USING THEM |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU23533A3 (en) |
-
2007
- 2007-02-08 CU CU20070041A patent/CU23533A3/en not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant of patent | ||
| FD | Lapse (for not paying fees) |