CU23568B7 - PYRIMIDINES REPLACED WITH SULFOXIMINE AS CDK AND / OR VEGF INHIBITORS, THEIR PREPARATION AND THEIR USES AS A MEDICINAL PRODUCT - Google Patents

PYRIMIDINES REPLACED WITH SULFOXIMINE AS CDK AND / OR VEGF INHIBITORS, THEIR PREPARATION AND THEIR USES AS A MEDICINAL PRODUCT

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Publication number
CU23568B7
CU23568B7 CU20060085A CU20060085A CU23568B7 CU 23568 B7 CU23568 B7 CU 23568B7 CU 20060085 A CU20060085 A CU 20060085A CU 20060085 A CU20060085 A CU 20060085A CU 23568 B7 CU23568 B7 CU 23568B7
Authority
CU
Cuba
Prior art keywords
preparation
sulfoximine
cdk
medicinal product
vegf inhibitors
Prior art date
Application number
CU20060085A
Other languages
Spanish (es)
Inventor
Rolf Jautelat
Ulrich Luecking
Martin Krueger
Gerhard Siemeister
Original Assignee
Bayer Schering Pharma Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Aktiengesellschaft filed Critical Bayer Schering Pharma Aktiengesellschaft
Priority to CU20060085A priority Critical patent/CU23568B7/en
Publication of CU23568B7 publication Critical patent/CU23568B7/en

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Abstract

La presente invención se refiere a derivados de pirimidina de la fórmula general (I), en donde Q, R1, R2, R3, R4, R5, X y m tienen los significados contenidos en la descripción, como inhibidores de las quinasas dependientes de ciclinas y tirosina quinasas de los receptores de VEGF, su preparación, y sus usos como medicamento para el tratamiento de diversas enfermedades.The present invention relates to pyrimidine derivatives of the general formula (I), wherein Q, R1, R2, R3, R4, R5, X and m have the meanings contained in the description, as inhibitors of cyclin-dependent kinases and tyrosine kinases of VEGF receptors, their preparation, and their uses as a medicine for the treatment of various diseases.

CU20060085A 2006-04-13 2006-04-13 PYRIMIDINES REPLACED WITH SULFOXIMINE AS CDK AND / OR VEGF INHIBITORS, THEIR PREPARATION AND THEIR USES AS A MEDICINAL PRODUCT CU23568B7 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20060085A CU23568B7 (en) 2006-04-13 2006-04-13 PYRIMIDINES REPLACED WITH SULFOXIMINE AS CDK AND / OR VEGF INHIBITORS, THEIR PREPARATION AND THEIR USES AS A MEDICINAL PRODUCT

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20060085A CU23568B7 (en) 2006-04-13 2006-04-13 PYRIMIDINES REPLACED WITH SULFOXIMINE AS CDK AND / OR VEGF INHIBITORS, THEIR PREPARATION AND THEIR USES AS A MEDICINAL PRODUCT

Publications (1)

Publication Number Publication Date
CU23568B7 true CU23568B7 (en) 2010-09-30

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
CU20060085A CU23568B7 (en) 2006-04-13 2006-04-13 PYRIMIDINES REPLACED WITH SULFOXIMINE AS CDK AND / OR VEGF INHIBITORS, THEIR PREPARATION AND THEIR USES AS A MEDICINAL PRODUCT

Country Status (1)

Country Link
CU (1) CU23568B7 (en)

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