CU23666B7 - AMINOHETEROARILO COMPOUNDS REPLACED WITH PIRAZOL AS INHIBITORS OF PROTEIN QUINASA - Google Patents
AMINOHETEROARILO COMPOUNDS REPLACED WITH PIRAZOL AS INHIBITORS OF PROTEIN QUINASAInfo
- Publication number
- CU23666B7 CU23666B7 CU20070046A CU20070046A CU23666B7 CU 23666 B7 CU23666 B7 CU 23666B7 CU 20070046 A CU20070046 A CU 20070046A CU 20070046 A CU20070046 A CU 20070046A CU 23666 B7 CU23666 B7 CU 23666B7
- Authority
- CU
- Cuba
- Prior art keywords
- inhibitors
- aminoheteroarilo
- pirazol
- compounds replaced
- compounds
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 239000003112 inhibitor Substances 0.000 title 1
- 102000004169 proteins and genes Human genes 0.000 title 1
- 108090000623 proteins and genes Proteins 0.000 title 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000008022 Proto-Oncogene Proteins c-met Human genes 0.000 abstract 1
- 108010089836 Proto-Oncogene Proteins c-met Proteins 0.000 abstract 1
- 230000002159 abnormal effect Effects 0.000 abstract 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 230000010261 cell growth Effects 0.000 abstract 1
- 208000037824 growth disorder Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 239000003909 protein kinase inhibitor Substances 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se proporcionan compuestos de fórmula 1 ESPACIO PARA FÓRMULA así como procedimientos para su síntesis y uso. Los compuestos preferidos son potentes inhibidores de la proteína quinasa c-Met, y son útiles en el tratamiento de trastornos del crecimiento celular anormal, tales como cánceres.Compounds of formula 1 SPACE FOR FORMULA are provided as well as procedures for their synthesis and use. Preferred compounds are potent c-Met protein kinase inhibitors, and are useful in the treatment of abnormal cell growth disorders, such as cancers.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20070046A CU23666B7 (en) | 2007-02-20 | 2007-02-20 | AMINOHETEROARILO COMPOUNDS REPLACED WITH PIRAZOL AS INHIBITORS OF PROTEIN QUINASA |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20070046A CU23666B7 (en) | 2007-02-20 | 2007-02-20 | AMINOHETEROARILO COMPOUNDS REPLACED WITH PIRAZOL AS INHIBITORS OF PROTEIN QUINASA |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU23666B7 true CU23666B7 (en) | 2011-05-27 |
Family
ID=44306267
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU20070046A CU23666B7 (en) | 2007-02-20 | 2007-02-20 | AMINOHETEROARILO COMPOUNDS REPLACED WITH PIRAZOL AS INHIBITORS OF PROTEIN QUINASA |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU23666B7 (en) |
-
2007
- 2007-02-20 CU CU20070046A patent/CU23666B7/en active IP Right Grant
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant of patent |