CU24746B1 - Apirasas humanas, solubilizadas y modificadas útiles para prevenir y tratar el daño tisular - Google Patents

Apirasas humanas, solubilizadas y modificadas útiles para prevenir y tratar el daño tisular

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Publication number
CU24746B1
CU24746B1 CU2021000008A CU20210008A CU24746B1 CU 24746 B1 CU24746 B1 CU 24746B1 CU 2021000008 A CU2021000008 A CU 2021000008A CU 20210008 A CU20210008 A CU 20210008A CU 24746 B1 CU24746 B1 CU 24746B1
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CU
Cuba
Prior art keywords
human
solubilized
apyrases
useful
preventing
Prior art date
Application number
CU2021000008A
Other languages
English (en)
Other versions
CU20210008A7 (es
Inventor
Agostino Cirillo
Hilmar Ebersbach
Boerje Haraldsson
Thomas Huber
Guido Junge
Regina Link
Max Warncke
Chao Zou
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CU20210008A7 publication Critical patent/CU20210008A7/es
Publication of CU24746B1 publication Critical patent/CU24746B1/es

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    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/14Hydrolases (3)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/43Enzymes; Proenzymes; Derivatives thereof
    • A61K38/46Hydrolases (3)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/43Enzymes; Proenzymes; Derivatives thereof
    • A61K38/46Hydrolases (3)
    • A61K38/465Hydrolases (3) acting on ester bonds (3.1), e.g. lipases, ribonucleases
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12YENZYMES
    • C12Y306/00Hydrolases acting on acid anhydrides (3.6)
    • C12Y306/01Hydrolases acting on acid anhydrides (3.6) in phosphorus-containing anhydrides (3.6.1)
    • C12Y306/01005Apyrase (3.6.1.5), i.e. ATP diphosphohydrolase

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Genetics & Genomics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Microbiology (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Vascular Medicine (AREA)
  • Transplantation (AREA)

Abstract

<p>La invención se refiere a una apirasa humana solubilizada, tal como el CD39 humano, que comprende modificaciones en la regiones N terminal, C terminal y central, y conducen a una proteína sorprendentemente activa, segura y fácil de fabricar. En la presente solicitud se proporciona una apirasa humana solubilizada que comprende la secuencia de aminoácidos SEQ ID NO: 229.</p> <p> </p>
CU2021000008A 2018-07-18 2019-07-17 Apirasas humanas, solubilizadas y modificadas útiles para prevenir y tratar el daño tisular CU24746B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP18184269 2018-07-18
PCT/IB2019/056117 WO2020016804A1 (en) 2018-07-18 2019-07-17 Solubilized apyrases, methods and use

Publications (2)

Publication Number Publication Date
CU20210008A7 CU20210008A7 (es) 2021-08-06
CU24746B1 true CU24746B1 (es) 2025-04-04

Family

ID=62985993

Family Applications (1)

Application Number Title Priority Date Filing Date
CU2021000008A CU24746B1 (es) 2018-07-18 2019-07-17 Apirasas humanas, solubilizadas y modificadas útiles para prevenir y tratar el daño tisular

Country Status (27)

Country Link
US (2) US12325870B2 (es)
EP (1) EP3824079A1 (es)
JP (2) JP7425784B2 (es)
KR (1) KR102919646B1 (es)
CN (6) CN119020318A (es)
AR (1) AR115790A1 (es)
AU (1) AU2019306821B2 (es)
BR (1) BR112021000586A2 (es)
CA (1) CA3103684A1 (es)
CL (1) CL2021000129A1 (es)
CO (1) CO2021000210A2 (es)
CR (1) CR20210021A (es)
CU (1) CU24746B1 (es)
EA (1) EA202190057A1 (es)
EC (1) ECSP21002804A (es)
IL (1) IL280191A (es)
JO (1) JOP20210008A1 (es)
MA (1) MA53177A (es)
MX (1) MX2021000542A (es)
MY (1) MY203583A (es)
PE (1) PE20210185A1 (es)
PH (1) PH12021550122A1 (es)
SG (1) SG11202011776RA (es)
TW (1) TWI857965B (es)
UY (1) UY38299A (es)
WO (1) WO2020016804A1 (es)
ZA (1) ZA202007187B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY38299A (es) 2018-07-18 2020-02-28 Novartis Ag Apirasas solubilizadas, métodos y usos
WO2021243173A1 (en) * 2020-05-28 2021-12-02 Charm Sciences, Inc. Methods and assemblies for sample analysis
KR20250044705A (ko) 2022-07-29 2025-04-01 노파르티스 아게 Cd39, 재조합 cd39를 사용하는 급성 기관 손상의 치료
IL318397A (en) 2022-07-29 2025-03-01 Novartis Ag Improved production of CD39 variants
AU2024360371A1 (en) * 2023-10-13 2026-02-26 Danisco Usa Inc. Methods and compositions for aging and mitochondrial health

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6447771B1 (en) 1999-03-19 2002-09-10 Hyseq, Inc. Methods and materials relating to novel CD39-like polypeptides
AU772460B2 (en) 1998-10-16 2004-04-29 Immunex Corporation Inhibitors of platelet activation and recruitment
US20020002277A1 (en) * 1998-10-16 2002-01-03 Maliszewski Charles Richard Inhibitors of platelet activation and recruitment
US6867177B2 (en) 1999-08-13 2005-03-15 The Trustees Of Columbia University In The City Of New York CD39/ECTO-adpase as a treatment for thrombotic and ischemic disorders
US7247300B1 (en) 2002-11-07 2007-07-24 Apt Therapeutics, Inc. Therapeutic use of soluble CD39L3
CA2578908C (en) 2005-03-17 2020-05-26 National Research Council Of Canada Expression vectors for enhanced transient gene expression and mammalian cells expressing them
WO2008002157A1 (en) 2006-06-27 2008-01-03 Agresearch Limited Apyrases and uses thereof
WO2011088231A1 (en) 2010-01-13 2011-07-21 Apt Therapeutics, Inc. Apyrase therapy for bleeding conditions
US8771683B2 (en) * 2010-01-13 2014-07-08 Apt Therapeutics, Inc. Therapeutic apyrase constructs, apyrase agents, and production methods
EP3604331A1 (en) 2013-12-20 2020-02-05 Novartis AG Novel eukaryotic cells and methods for recombinantly expressing a product of interest
AU2014369177B2 (en) 2013-12-20 2017-04-20 Novartis Ag Novel eukaryotic cells and methods for recombinantly expressing a product of interest
UY38299A (es) * 2018-07-18 2020-02-28 Novartis Ag Apirasas solubilizadas, métodos y usos

Also Published As

Publication number Publication date
MY203583A (en) 2024-07-05
JP7425784B2 (ja) 2024-01-31
CR20210021A (es) 2021-03-23
PE20210185A1 (es) 2021-02-02
CN112424346A (zh) 2021-02-26
MA53177A (fr) 2021-05-26
AU2019306821A1 (en) 2020-12-24
SG11202011776RA (en) 2021-02-25
CA3103684A1 (en) 2020-01-23
CN119020320A (zh) 2024-11-26
AU2019306821B2 (en) 2022-09-29
EP3824079A1 (en) 2021-05-26
MX2021000542A (es) 2021-03-29
JOP20210008A1 (ar) 2021-01-12
ECSP21002804A (es) 2021-04-29
AR115790A1 (es) 2021-02-24
CN112424346B (zh) 2024-08-06
CL2021000129A1 (es) 2021-08-20
CO2021000210A2 (es) 2021-01-18
US12325870B2 (en) 2025-06-10
WO2020016804A1 (en) 2020-01-23
US20220356455A1 (en) 2022-11-10
TWI857965B (zh) 2024-10-11
US20250179447A1 (en) 2025-06-05
UY38299A (es) 2020-02-28
IL280191A (en) 2021-03-01
CN119162148A (zh) 2024-12-20
KR20210035806A (ko) 2021-04-01
PH12021550122A1 (en) 2021-09-27
ZA202007187B (en) 2022-06-29
BR112021000586A2 (pt) 2021-04-06
JP2024023297A (ja) 2024-02-21
CU20210008A7 (es) 2021-08-06
TW202016299A (zh) 2020-05-01
EA202190057A1 (ru) 2021-08-24
CN119020319A (zh) 2024-11-26
KR102919646B1 (ko) 2026-01-29
JP2021529550A (ja) 2021-11-04
CN119020321A (zh) 2024-11-26
CN119020318A (zh) 2024-11-26

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