DD268246A5 - Verfahren zur herstellung neuer milbemycin-derivate - Google Patents

Verfahren zur herstellung neuer milbemycin-derivate Download PDF

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Publication number
DD268246A5
DD268246A5 DD88314036A DD31403688A DD268246A5 DD 268246 A5 DD268246 A5 DD 268246A5 DD 88314036 A DD88314036 A DD 88314036A DD 31403688 A DD31403688 A DD 31403688A DD 268246 A5 DD268246 A5 DD 268246A5
Authority
DD
German Democratic Republic
Prior art keywords
group
formula
compounds
hydrogen
halogen
Prior art date
Application number
DD88314036A
Other languages
German (de)
English (en)
Inventor
Jean-Claude Gehret
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ���@����������@��k�� filed Critical ���@����������@��k��
Publication of DD268246A5 publication Critical patent/DD268246A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DD88314036A 1987-03-27 1988-03-25 Verfahren zur herstellung neuer milbemycin-derivate DD268246A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH118087 1987-03-27

Publications (1)

Publication Number Publication Date
DD268246A5 true DD268246A5 (de) 1989-05-24

Family

ID=4204366

Family Applications (1)

Application Number Title Priority Date Filing Date
DD88314036A DD268246A5 (de) 1987-03-27 1988-03-25 Verfahren zur herstellung neuer milbemycin-derivate

Country Status (14)

Country Link
US (1) US4954484A (fr)
EP (1) EP0285561A3 (fr)
JP (1) JPS63250379A (fr)
KR (1) KR880011170A (fr)
AU (1) AU612139B2 (fr)
CA (1) CA1303029C (fr)
DD (1) DD268246A5 (fr)
HU (1) HUT46323A (fr)
IL (1) IL85869A (fr)
NZ (1) NZ224020A (fr)
PH (1) PH26026A (fr)
PT (1) PT87092B (fr)
ZA (1) ZA882141B (fr)
ZW (1) ZW3088A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0285561A3 (fr) * 1987-03-27 1989-10-25 Ciba-Geigy Ag Dérivés de la milbémycine à activité antiparasitaire et insecticide
US5015630A (en) * 1989-01-19 1991-05-14 Merck & Co., Inc. 5-oxime avermectin derivatives
EP0393890B1 (fr) * 1989-04-11 1992-08-12 Pfizer Limited Compositions injectables à base de 25-cyclohexyle avermectine B1
US5240915A (en) * 1991-10-15 1993-08-31 Merck & Co., Inc. Avermectin derivatives
US5461168A (en) * 1992-09-01 1995-10-24 Sankyo Company, Limited Processes for the production of 13-ether derivatives of milbemycins, and intermediates therefor
GB9315108D0 (en) * 1993-07-21 1993-09-01 Pfizer Ltd Antiparasitic agents

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3950360A (en) * 1972-06-08 1976-04-13 Sankyo Company Limited Antibiotic substances
US4093629A (en) * 1977-04-11 1978-06-06 Merck & Co., Inc. Derivatives of antibiotic substance milbemycin and processes therefor
US4173571A (en) * 1977-12-19 1979-11-06 Merck & Co., Inc. 13-Halo and 13-deoxy derivatives of C-076 compounds
US4130519A (en) * 1978-04-03 1978-12-19 Exxon Research & Engineering Co. Stabilized halogenated butyl rubber
US4328335A (en) * 1979-08-13 1982-05-04 Merck & Co., Inc. Process for the interconversion of C-076 compounds
JPS5632481A (en) * 1979-08-23 1981-04-01 Sankyo Co Ltd Antibiotic b-41d, its preparation, and acaricide and anthelminthic agent and repellent containing the same as active constituent
US4582852A (en) * 1983-11-02 1986-04-15 Ciba-Geigy Corporation 14- and 15-hydroxy milbemycin derivatives for controlling plant and animal parasites
DE3519834C2 (de) * 1984-06-05 1993-12-16 American Cyanamid Co Neue antibiotische Wirkstoffe, Verfahren zu ihrer Gewinnung und ihre Anwendung zur Bekämpfung von Infektionen bei Tieren und Pflanzen
EP0165900A3 (fr) * 1984-06-08 1986-05-28 Ciba-Geigy Ag Lactones, leur méthode de préparation et leur utilisation comme herbicide
CH666690A5 (de) * 1984-09-14 1988-08-15 Glaxo Group Ltd Antibiotisch wirkende verbindungen der makrolidgruppe aus streptomyces-mikroorganismen, ihre herstellung und verwendung.
FI860233L (fi) * 1985-01-22 1986-07-23 Ciba Geigy Ag 13 -alkyl-milbemycinderivat foer bekaempning av parasiter hos djur och vaexter.
US4581345A (en) * 1985-04-08 1986-04-08 Merck & Co., Inc. Avermectin 8,9-cyclopropyl compounds, pharmaceutical composition and therapeutic methods of use
IL78621A (en) * 1985-04-30 1991-06-30 American Cyanamid Co Mylbemycin analogs,their preparation and pesticidal compositions containing them
US4778809A (en) * 1985-08-23 1988-10-18 Ciba-Geigy Corporation 5-esters of milbemycins for controlling parasitic pests
IE62125B1 (en) * 1986-03-12 1994-12-14 American Cyanamid Co Macrolide compounds
EP0285561A3 (fr) * 1987-03-27 1989-10-25 Ciba-Geigy Ag Dérivés de la milbémycine à activité antiparasitaire et insecticide

Also Published As

Publication number Publication date
ZW3088A1 (en) 1988-11-16
KR880011170A (ko) 1988-10-27
CA1303029C (fr) 1992-06-09
NZ224020A (en) 1990-10-26
PH26026A (en) 1992-01-29
PT87092B (pt) 1992-07-31
JPS63250379A (ja) 1988-10-18
US4954484A (en) 1990-09-04
AU612139B2 (en) 1991-07-04
EP0285561A3 (fr) 1989-10-25
AU1374888A (en) 1988-09-29
PT87092A (pt) 1988-04-01
ZA882141B (en) 1990-03-28
HUT46323A (en) 1988-10-28
EP0285561A2 (fr) 1988-10-05
IL85869A0 (en) 1988-09-30
IL85869A (en) 1991-12-12

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Legal Events

Date Code Title Description
ENJ Ceased due to non-payment of renewal fee