DK0596891T3 - Aminoalkylsubstituerede 2-amino-5-mercaptothiadiazoler, deres fremstilling og anvendelse - Google Patents

Aminoalkylsubstituerede 2-amino-5-mercaptothiadiazoler, deres fremstilling og anvendelse

Info

Publication number: DK0596891T3
Authority: DK; Denmark
Prior art keywords: pct; aminoalkyl; amino; substituted; preparation
Prior art date: 1991-06-15

Application number

DK92910040T

Other languages

English (en)

Inventor

Beatrice Rendenbach-Mueller

Hans-Juergen Teschendorf

Liliane Unger

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-06-15

Filing date

1992-05-08

Publication date

1998-10-26

1992-05-08 Application filed by Basf Ag filed Critical Basf Ag

1998-10-26 Application granted granted Critical

1998-10-26 Publication of DK0596891T3 publication Critical patent/DK0596891T3/da

Links

GOISVZSJABSIHS-UHFFFAOYSA-N 2-amino-3h-thiadiazole-5-thiol Chemical class NN1NC=C(S)S1 GOISVZSJABSIHS-UHFFFAOYSA-N 0.000 title 1
GDGIVSREGUOIJZ-UHFFFAOYSA-N 5-amino-3h-1,3,4-thiadiazole-2-thione Chemical class NC1=NN=C(S)S1 GDGIVSREGUOIJZ-UHFFFAOYSA-N 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
201000010099 disease Diseases 0.000 abstract 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Psychiatry (AREA)
Psychology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DK92910040T 1991-06-15 1992-05-08 Aminoalkylsubstituerede 2-amino-5-mercaptothiadiazoler, deres fremstilling og anvendelse DK0596891T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE4119758A DE4119758A1 (de)	1991-06-15	1991-06-15	Aminoalkylsubstituierte 2-amino-5-mercaptothiadiazole, ihre herstellung und verwendung
PCT/EP1992/001003 WO1992022542A1 (de)	1991-06-15	1992-05-08	Aminoalkylsubstituierte 2-amino-5-mercaptothiadiazole, ihre herstellung und verwendung

Publications (1)

Publication Number	Publication Date
DK0596891T3 true DK0596891T3 (da)	1998-10-26

Family

ID=6434012

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK92910040T DK0596891T3 (da)	1991-06-15	1992-05-08	Aminoalkylsubstituerede 2-amino-5-mercaptothiadiazoler, deres fremstilling og anvendelse

Country Status (9)

Country	Link
US (1)	US5401743A (da)
EP (1)	EP0596891B1 (da)
JP (1)	JP3199736B2 (da)
AT (1)	ATE169619T1 (da)
CA (1)	CA2111442A1 (da)
DE (2)	DE4119758A1 (da)
DK (1)	DK0596891T3 (da)
ES (1)	ES2118817T3 (da)
WO (1)	WO1992022542A1 (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4425145A1 (de) *	1994-07-15	1996-01-18	Basf Ag	Verwendung von Thiazol- und Thiadiazolverbindungen
US6191152B1 (en)	1997-01-14	2001-02-20	Egis Gyógyszergyar Rt.	2-(1,2,4-triazole-1-yl)-1,3,4-thiadiazole derivatives having an effect on the C.N.S. and the heart
DE19728996A1 (de)	1997-07-07	1999-01-14	Basf Ag	Triazolverbindungen und deren Verwendung
US20030087917A1 (en) *	2000-03-27	2003-05-08	Dorothea Strack	Use of dopamine-d3 receptor ligands for the treatment of diseases of the central nervous system
EP4092013A1 (en)	2017-06-20	2022-11-23	Imbria Pharmaceuticals, Inc.	Compositions and methods for increasing efficiency of cardiac metabolism
WO2020081361A1 (en)	2018-10-17	2020-04-23	Imbria Pharmaceuticals, Inc.	Methods of treating rheumatic diseases using trimetazidine-based compounds
WO2020243120A1 (en)	2019-05-31	2020-12-03	Imbria Pharmaceuticals, Inc.	Methods of treating fibrosis using compounds that promote glucose oxidation
US11530184B2 (en)	2020-06-30	2022-12-20	Imbria Pharmaceuticals, Inc.	Crystal forms of 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate
US11780811B2 (en)	2020-06-30	2023-10-10	Imbria Pharmaceuticals, Inc.	Methods of synthesizing 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate
US11883396B2 (en)	2021-05-03	2024-01-30	Imbria Pharmaceuticals, Inc.	Methods of treating kidney conditions using modified forms of trimetazidine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US1053085A (en)	1909-05-08	1913-02-11	Edward S Cole	Recording device.
US4074049A (en)	1976-11-19	1978-02-14	The Dow Chemical Company	Antithrombotic 1,3,4-thiadiazole
JPS62153276A (ja) *	1985-12-26	1987-07-08	Yamanouchi Pharmaceut Co Ltd	含窒素５員複素環化合物及びその製造法

1991
- 1991-06-15 DE DE4119758A patent/DE4119758A1/de not_active Withdrawn
1992
- 1992-05-08 WO PCT/EP1992/001003 patent/WO1992022542A1/de not_active Ceased
- 1992-05-08 JP JP50949592A patent/JP3199736B2/ja not_active Expired - Fee Related
- 1992-05-08 DK DK92910040T patent/DK0596891T3/da active
- 1992-05-08 DE DE59209455T patent/DE59209455D1/de not_active Expired - Fee Related
- 1992-05-08 EP EP92910040A patent/EP0596891B1/de not_active Expired - Lifetime
- 1992-05-08 ES ES92910040T patent/ES2118817T3/es not_active Expired - Lifetime
- 1992-05-08 CA CA002111442A patent/CA2111442A1/en not_active Abandoned
- 1992-05-08 AT AT92910040T patent/ATE169619T1/de not_active IP Right Cessation
- 1992-05-08 US US08/162,117 patent/US5401743A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US5401743A (en)	1995-03-28
WO1992022542A1 (de)	1992-12-23
CA2111442A1 (en)	1992-12-23
JPH06507887A (ja)	1994-09-08
DE4119758A1 (de)	1992-12-17
JP3199736B2 (ja)	2001-08-20
DE59209455D1 (de)	1998-09-17
ES2118817T3 (es)	1998-10-01
EP0596891A1 (de)	1994-05-18
ATE169619T1 (de)	1998-08-15
EP0596891B1 (de)	1998-08-12

Publication	Publication Date	Title
NO306346B1 (no)	1999-10-25	N-substituerte azabicykloalkanderivater, anvendelse derav og farmasöytisk preparat
DK0668869T3 (da)	1998-10-07	2-[3-(4-amidinophenyl)]-propionsyrederivater, deres fremstilling og anvendelse
BR9706986A (pt)	1999-07-20	5-Amino-1,2,4-tiadiazóis acilados
DK0596891T3 (da)	1998-10-26	Aminoalkylsubstituerede 2-amino-5-mercaptothiadiazoler, deres fremstilling og anvendelse
ATE108437T1 (de)	1994-07-15	Substituierte diaminophthalimide und analoga.
NO972559D0 (no)	1997-06-05	Nye dipeptid-p-amidinobenzylamider med N-terminale sulfonyl- eller aminosulfonylrester
NO306400B1 (no)	1999-11-01	N-substituerte azabicykloheptan-derivater, anvendelse derav og farmasöytisk preparat
DK0589903T3 (da)	1999-06-07	Aminoalkylsubstituerede 5-mercaptothiazoler, deres fremstilling og anvendelse
DK0589908T3 (da)	1998-10-26	Aminoalkylsubsituerede thiazolin-2-oner, deres fremstilling og deres anvendelse
FI923679A0 (fi)	1992-08-17	Ny b-fenylisoserinderivat, dess framstaellning och anvaendning.
DK0592453T3 (da)	1999-08-23	Aminoalkylsubstituerede 2-amino-1,3,4-thiadiazoler, deres fremstilling og deres anvendelse
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ATE92069T1 (de)	1993-08-15	4-substituierte 10-cyanmethylenpyrrolo(4,3-e>benzo-azepine.
NO952292D0 (no)	1995-06-09	Nye triazolokinazoliner, deres fremstilling og anvendelse
ES2093280T3 (es)	1996-12-16	Derivados de leucotrieno-b 4?, procedimiento de obtencion y farmacos.
NO952291D0 (no)	1995-06-09	Nye triazolopyrimidoner, deres fremstilling og deres anvendelse