DK0614888T3 - Tetrahydrocyclopentab indol-methanaminer og beslægtede forbindelser, en fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler. - Google Patents
Tetrahydrocyclopentab indol-methanaminer og beslægtede forbindelser, en fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler.Info
- Publication number
- DK0614888T3 DK0614888T3 DK94102993.6T DK94102993T DK0614888T3 DK 0614888 T3 DK0614888 T3 DK 0614888T3 DK 94102993 T DK94102993 T DK 94102993T DK 0614888 T3 DK0614888 T3 DK 0614888T3
- Authority
- DK
- Denmark
- Prior art keywords
- tetrahydrocyclopentab
- methanamines
- indole
- drugs
- preparation
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- RNAODKZCUVVPEN-UHFFFAOYSA-N 1h-indol-2-ylmethanamine Chemical class C1=CC=C2NC(CN)=CC2=C1 RNAODKZCUVVPEN-UHFFFAOYSA-N 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 208000024827 Alzheimer disease Diseases 0.000 abstract 1
- 229940122041 Cholinesterase inhibitor Drugs 0.000 abstract 1
- 208000020401 Depressive disease Diseases 0.000 abstract 1
- 229940123685 Monoamine oxidase inhibitor Drugs 0.000 abstract 1
- 239000000544 cholinesterase inhibitor Substances 0.000 abstract 1
- 230000007074 memory dysfunction Effects 0.000 abstract 1
- 239000002899 monoamine oxidase inhibitor Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/58—[b]- or [c]-condensed
- C07D209/62—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles
- C07D209/64—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles with an oxygen atom in position 1
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/028,110 US5350762A (en) | 1993-03-08 | 1993-03-08 | Tetrahydrocyclopent[B]indole methanamines and related compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0614888T3 true DK0614888T3 (da) | 1997-11-03 |
Family
ID=21841633
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK94102993.6T DK0614888T3 (da) | 1993-03-08 | 1994-02-28 | Tetrahydrocyclopentab indol-methanaminer og beslægtede forbindelser, en fremgangsmåde til deres fremstilling og deres anvendelse som lægemidler. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US5350762A (da) |
| EP (1) | EP0614888B1 (da) |
| JP (1) | JP2749259B2 (da) |
| AT (1) | ATE152709T1 (da) |
| CA (1) | CA2117164A1 (da) |
| DE (1) | DE69403015T2 (da) |
| DK (1) | DK0614888T3 (da) |
| ES (1) | ES2101373T3 (da) |
| GR (1) | GR3024187T3 (da) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5756743A (en) | 1996-04-10 | 1998-05-26 | Hoechst Marion Roussel Inc. | Spiro cyclopent b!indole-piperidines! |
| US5665880A (en) * | 1996-10-31 | 1997-09-09 | Hoechst Marion Roussel, Inc. | Method of preparation of physostigmine carbamate derivatives from eseretholes |
| DE69738275T2 (de) | 1996-12-18 | 2008-08-28 | Teva Pharmaceutical Industries Ltd. | Aminoindanderivate |
| US6251938B1 (en) | 1996-12-18 | 2001-06-26 | Teva Pharmaceutical Industries, Ltd., | Phenylethylamine derivatives |
| US5677457A (en) * | 1996-12-19 | 1997-10-14 | Hoechst Marion Roussel, Inc. | Method of preparation of physostigmine carbamate derivatives from eseroline ethers |
| IT1317926B1 (it) * | 2000-11-03 | 2003-07-15 | Sigma Tau Ind Farmaceuti | Derivati triciclici dell'indolo ad attivita' antiangiogenica. |
| CN103142570A (zh) | 2005-12-09 | 2013-06-12 | 耶路撒冷希伯来大学伊森姆研究发展公司 | 低剂量Ladostigil 用于神经保护的用途 |
| TW200744576A (en) | 2006-02-24 | 2007-12-16 | Teva Pharma | Propargylated aminoindans, processes for preparation, and uses thereof |
| MY147588A (en) * | 2006-08-07 | 2012-12-31 | Actelion Pharmaceuticals Ltd | (3-amino-1,2,3,4-tetrahydro-9h-carbazol-9-yl)-acetic acid derivatives |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE757404A (da) * | 1969-10-13 | 1971-04-13 | Sandoz Sa | |
| BE793493A (fr) * | 1971-12-30 | 1973-06-29 | Hoffmann La Roche | Composes tricycliques |
| US4009181A (en) * | 1973-01-22 | 1977-02-22 | Hoffmann-La Roche Inc. | Cyclopenta[b]indole-2-carboxylic acids and derivatives thereof |
| JPS5111760A (da) * | 1974-06-18 | 1976-01-30 | Ayerst Mckenna & Harrison | |
| JPS5283736A (en) * | 1976-01-01 | 1977-07-12 | Ayerst Mckenna & Harrison | Tricyclic alkylamine derivatives |
| US4235903A (en) * | 1979-08-06 | 1980-11-25 | American Home Products Corporation | 1-Hydroxyalkanamine tetrahydrocarbazoles and cyclopent[b]indoles, compositions and method of use |
| US5100891A (en) * | 1991-01-18 | 1992-03-31 | Hoechst-Roussel Pharmaceuticals Inc. | Substituted 1,2,3,4-tetrahydrocyclopent[b]indoles, 1,2,3,3a,4,8a-hexahydrocyclopent[B]indoles and related compounds |
-
1993
- 1993-03-08 US US08/028,110 patent/US5350762A/en not_active Expired - Fee Related
-
1994
- 1994-02-28 DE DE69403015T patent/DE69403015T2/de not_active Expired - Fee Related
- 1994-02-28 ES ES94102993T patent/ES2101373T3/es not_active Expired - Lifetime
- 1994-02-28 DK DK94102993.6T patent/DK0614888T3/da active
- 1994-02-28 AT AT94102993T patent/ATE152709T1/de not_active IP Right Cessation
- 1994-02-28 EP EP94102993A patent/EP0614888B1/en not_active Expired - Lifetime
- 1994-03-07 CA CA002117164A patent/CA2117164A1/en not_active Abandoned
- 1994-03-08 JP JP6037031A patent/JP2749259B2/ja not_active Expired - Fee Related
-
1997
- 1997-07-22 GR GR970401832T patent/GR3024187T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPH06321898A (ja) | 1994-11-22 |
| DE69403015T2 (de) | 1997-10-09 |
| EP0614888A1 (en) | 1994-09-14 |
| DE69403015D1 (de) | 1997-06-12 |
| ES2101373T3 (es) | 1997-07-01 |
| US5350762A (en) | 1994-09-27 |
| CA2117164A1 (en) | 1994-09-09 |
| EP0614888B1 (en) | 1997-05-07 |
| ATE152709T1 (de) | 1997-05-15 |
| GR3024187T3 (en) | 1997-10-31 |
| JP2749259B2 (ja) | 1998-05-13 |
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