DK0653422T3 - Fremgangsmåde til fremstilling af 2-substituerede 5-chlorimidazol-4-carbaldehyder - Google Patents
Fremgangsmåde til fremstilling af 2-substituerede 5-chlorimidazol-4-carbaldehyderInfo
- Publication number
- DK0653422T3 DK0653422T3 DK94117951.7T DK94117951T DK0653422T3 DK 0653422 T3 DK0653422 T3 DK 0653422T3 DK 94117951 T DK94117951 T DK 94117951T DK 0653422 T3 DK0653422 T3 DK 0653422T3
- Authority
- DK
- Denmark
- Prior art keywords
- substituted
- carbaldehydes
- chloroimidazole
- preparation
- ester
- Prior art date
Links
- -1 2-substituted 5-chloroimidazole-4-carbaldehydes Chemical class 0.000 title abstract 5
- 238000000034 method Methods 0.000 title abstract 2
- AHIMYRXIOVKJGA-UHFFFAOYSA-N 5-(aminomethylidene)-1h-imidazol-4-one Chemical class NC=C1NC=NC1=O AHIMYRXIOVKJGA-UHFFFAOYSA-N 0.000 abstract 1
- OHVWCRAXBOZMMG-UHFFFAOYSA-N 5-chloro-1h-imidazole-4-carbaldehyde Chemical class ClC=1N=CNC=1C=O OHVWCRAXBOZMMG-UHFFFAOYSA-N 0.000 abstract 1
- DHMQDGOQFOQNFH-UHFFFAOYSA-N Glycine Natural products NCC(O)=O DHMQDGOQFOQNFH-UHFFFAOYSA-N 0.000 abstract 1
- 239000004471 Glycine Substances 0.000 abstract 1
- DHKHKXVYLBGOIT-UHFFFAOYSA-N acetaldehyde Diethyl Acetal Natural products CCOC(C)OCC DHKHKXVYLBGOIT-UHFFFAOYSA-N 0.000 abstract 1
- 230000036772 blood pressure Effects 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 238000005660 chlorination reaction Methods 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- ZHNUHDYFZUAESO-UHFFFAOYSA-N formamide Substances NC=O ZHNUHDYFZUAESO-UHFFFAOYSA-N 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/96—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/68—Halogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Epoxy Resins (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Photoreceptors In Electrophotography (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH341093 | 1993-11-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0653422T3 true DK0653422T3 (da) | 1998-05-11 |
Family
ID=4255388
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK94117951.7T DK0653422T3 (da) | 1993-11-15 | 1994-11-14 | Fremgangsmåde til fremstilling af 2-substituerede 5-chlorimidazol-4-carbaldehyder |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US5486617A (da) |
| EP (1) | EP0653422B1 (da) |
| JP (1) | JP3924795B2 (da) |
| KR (1) | KR100343825B1 (da) |
| AT (1) | ATE163411T1 (da) |
| CA (1) | CA2135541C (da) |
| DE (1) | DE59405299D1 (da) |
| DK (1) | DK0653422T3 (da) |
| ES (1) | ES2115134T3 (da) |
| HU (1) | HU223139B1 (da) |
| RU (1) | RU94040184A (da) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2175420C (en) * | 1995-05-17 | 2007-04-10 | Gareth Griffiths | Process for the preparation of optionally 2-substituted 5-chloroimidazole-4-carbaldehydes |
| JP4103149B2 (ja) | 1996-01-05 | 2008-06-18 | ロンザ リミテッド | ２−置換５−クロロイミダゾール−４−カルブアルデヒドの製造方法 |
| US20040126337A1 (en) * | 2002-12-30 | 2004-07-01 | Singleton Laura C. | Sunscreen compositions |
| ATE485278T1 (de) * | 2005-04-15 | 2010-11-15 | Dishman Pharmaceuticals And Ch | Herstellung von 2-substituierten 4-chlor-5- formylimidazolen durch vilsmeier-reaktion des kondensationsprodukts von glycin und einem imidoester mit einem formamid in gegenwart eines triflat- (trifluormethansulfonat-) katalysators |
| CN101838242B (zh) * | 2010-05-16 | 2015-07-15 | 浙江工业大学 | 2-正丁基-4-氯-5-甲酰基咪唑的合成方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL53783A (en) * | 1977-02-03 | 1982-08-31 | American Cyanamid Co | Imidazo(1,5-d)-as-triazine-4 (3h)-(thi)one derivatives,their preparation and pharmaceutical compositions containing them |
| JPS5671074A (en) * | 1979-11-12 | 1981-06-13 | Takeda Chem Ind Ltd | 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative |
-
1994
- 1994-11-10 CA CA002135541A patent/CA2135541C/en not_active Expired - Fee Related
- 1994-11-11 RU RU94040184/04A patent/RU94040184A/ru unknown
- 1994-11-11 JP JP27817194A patent/JP3924795B2/ja not_active Expired - Fee Related
- 1994-11-14 DE DE59405299T patent/DE59405299D1/de not_active Expired - Lifetime
- 1994-11-14 HU HU9403263A patent/HU223139B1/hu not_active IP Right Cessation
- 1994-11-14 US US08/340,377 patent/US5486617A/en not_active Expired - Lifetime
- 1994-11-14 EP EP94117951A patent/EP0653422B1/de not_active Expired - Lifetime
- 1994-11-14 ES ES94117951T patent/ES2115134T3/es not_active Expired - Lifetime
- 1994-11-14 DK DK94117951.7T patent/DK0653422T3/da active
- 1994-11-14 AT AT94117951T patent/ATE163411T1/de active
- 1994-11-15 KR KR1019940029964A patent/KR100343825B1/ko not_active Expired - Fee Related
-
1995
- 1995-06-19 US US08/492,444 patent/US5536841A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| JPH07188180A (ja) | 1995-07-25 |
| US5486617A (en) | 1996-01-23 |
| US5536841A (en) | 1996-07-16 |
| CA2135541A1 (en) | 1995-05-16 |
| ES2115134T3 (es) | 1998-06-16 |
| HU9403263D0 (en) | 1995-01-30 |
| DE59405299D1 (de) | 1998-04-02 |
| CA2135541C (en) | 2006-01-10 |
| EP0653422A1 (de) | 1995-05-17 |
| HUT70047A (en) | 1995-09-28 |
| RU94040184A (ru) | 1996-10-10 |
| EP0653422B1 (de) | 1998-02-25 |
| KR950014076A (ko) | 1995-06-15 |
| HU223139B1 (hu) | 2004-03-29 |
| KR100343825B1 (ko) | 2002-11-23 |
| JP3924795B2 (ja) | 2007-06-06 |
| ATE163411T1 (de) | 1998-03-15 |
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