DK0719775T3 - Substituerede derivater af 4-phenylthiazol, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger, der inde - Google Patents

Substituerede derivater af 4-phenylthiazol, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger, der inde

Info

Publication number
DK0719775T3
DK0719775T3 DK95402969T DK95402969T DK0719775T3 DK 0719775 T3 DK0719775 T3 DK 0719775T3 DK 95402969 T DK95402969 T DK 95402969T DK 95402969 T DK95402969 T DK 95402969T DK 0719775 T3 DK0719775 T3 DK 0719775T3
Authority
DK
Denmark
Prior art keywords
phenylthiazole
preparation
pharmaceutical compositions
compositions containing
substituted derivatives
Prior art date
Application number
DK95402969T
Other languages
English (en)
Inventor
Alain Badorc
Marie-Francoise Bordes
Cointet Paul De
Jean-Marc Herbert
Jean-Pierre Maffrand
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Application granted granted Critical
Publication of DK0719775T3 publication Critical patent/DK0719775T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
DK95402969T 1994-12-28 1995-12-28 Substituerede derivater af 4-phenylthiazol, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger, der inde DK0719775T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9415805A FR2728901B1 (fr) 1994-12-28 1994-12-28 Derives de phenyl-4-thiazoles substitues, procede pour leur preparation et compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
DK0719775T3 true DK0719775T3 (da) 2000-10-23

Family

ID=9470360

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95402969T DK0719775T3 (da) 1994-12-28 1995-12-28 Substituerede derivater af 4-phenylthiazol, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger, der inde

Country Status (28)

Country Link
US (1) US5607952A (da)
EP (1) EP0719775B1 (da)
JP (1) JP3027110B2 (da)
KR (1) KR960022515A (da)
CN (1) CN1048726C (da)
AR (1) AR002017A1 (da)
AT (1) ATE194616T1 (da)
AU (1) AU703490B2 (da)
BR (1) BR1100524A (da)
CA (1) CA2166165A1 (da)
CZ (1) CZ346595A3 (da)
DE (1) DE69517936T2 (da)
DK (1) DK0719775T3 (da)
ES (1) ES2148458T3 (da)
FI (1) FI956278A7 (da)
FR (1) FR2728901B1 (da)
GR (1) GR3034582T3 (da)
HU (1) HUT75096A (da)
IL (1) IL116560A (da)
NO (1) NO306114B1 (da)
NZ (1) NZ280720A (da)
PL (1) PL312078A1 (da)
PT (1) PT719775E (da)
RU (1) RU2124515C1 (da)
SI (1) SI0719775T1 (da)
SK (1) SK281247B6 (da)
TW (1) TW418207B (da)
ZA (1) ZA9511029B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5840733A (en) * 1996-07-01 1998-11-24 Redcell, Canada, Inc. Methods and compositions for producing novel conjugates of thrombin inhibitors and endogenous carriers resulting in anti-thrombins with extended lifetimes
US6010911A (en) * 1997-04-30 2000-01-04 Medtronic, Inc. Apparatus for performing a heparin-independent high sensitivity platelet function evaluation technique
FR2764511B1 (fr) * 1997-06-13 2000-09-08 Sanofi Sa Compositions pour le traitement et la prevention de la thrombose arterielle et utilisation d'un inhibiteur du facteur xa seul et/ou en combinaison avec un antiagregant plaquettaire
AU1735200A (en) 1998-11-18 2000-06-05 Du Pont Pharmaceuticals Company Novel isoxazoline fibrinogen receptor antagonists
US6319937B1 (en) 1998-11-18 2001-11-20 Dupont Pharmaceuticals Company Isoxazoline fibrinogen receptor antagonists
FR2797400A1 (fr) * 1999-08-11 2001-02-16 Sanofi Synthelabo Associations a activite anti-thrombotique constituees de l'hydrogenosulfate de clopidogrel et d'un antagoniste des recepteurs gpiib/iiia et les compositions pharmaceutiques les contenant
TWI284639B (en) * 2000-01-24 2007-08-01 Shionogi & Co A compound having thrombopoietin receptor agonistic effect
US20060198836A1 (en) * 2003-07-17 2006-09-07 Smithkline Beecham Corporation Method of treating hit patients with argatroban
US7601746B2 (en) * 2003-08-12 2009-10-13 Shionogi & Co., Ltd. Compounds exhibiting thrombopoietin receptor agonism
CA2533464A1 (en) * 2003-08-12 2005-02-17 F. Hoffmann-La Roche Ag Thiazole derivatives as npy antagonists
CA2566081A1 (en) * 2004-05-13 2005-12-01 Boehringer Ingelheim International Gmbh Use of dipyridamole for treatment of resistance to platelet inhibitors
JP2007538257A (ja) * 2004-05-17 2007-12-27 メドトロニック・インコーポレーテッド ポイント・オブ・ヘパリン測定システム
US7423053B2 (en) * 2004-07-15 2008-09-09 Hoffmann-La Roche Inc. 4-Aminothiazole derivatives
RU2391340C2 (ru) * 2004-08-11 2010-06-10 Киорин Фармасьютикал Ко., Лтд. Новое циклическое производное аминобензойной кислоты
WO2007003960A1 (en) * 2005-06-30 2007-01-11 Prosidion Limited Gpcr agonists
RU2373929C1 (ru) * 2008-11-11 2009-11-27 Государственное образовательное учреждение высшего профессионального образования "БАШКИРСКИЙ ГОСУДАРСТВЕННЫЙ МЕДИЦИНСКИЙ УНИВЕРСИТЕТ Федерального Агентства по здравоохранению и социальному развитию" (ГОУ ВПО БГМУ РОСЗДРАВА) Корректор системы гемостаза, проявляющий ингибирующее действие на адгезивно-агрегационную функцию тромбоцитов для профилактики патологического тромбообразования

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB542363A (en) * 1940-07-03 1942-01-06 Joseph Arthur Musgrave Woodcoc Improvements in or relating to the manufacture of graphite electrodes
DK157135C (da) * 1982-04-07 1990-04-02 Pfizer Analogifremgangsmaade til fremstilling af 1,2,4-triazol-forbindelser eller farmaceutisk acceptable syreadditionssalte deraf
DE3839758A1 (de) * 1988-10-24 1990-04-26 Bayer Ag Substituierte 2-aminothiazole
US5231091A (en) * 1988-12-19 1993-07-27 American Cyanamid Company Bis-arylphosphate ester antagonists of platelet activating factor
FR2656610B1 (fr) * 1989-12-29 1992-05-07 Sanofi Sa Derives d'amino-2 phenyl-4 thiazole, leur procede de preparation et leur application therapeutique.
AU2915892A (en) * 1991-11-14 1993-06-15 Glaxo Group Limited Piperidine acetic acid derivatives as inhibitors of fibrinogen-dependent blood platelet aggregation
US5405848A (en) * 1993-12-22 1995-04-11 Ortho Pharmaceutical Corporation Substituted thiazolylaminotetrahydropyridopyrimidines derivatives useful as platelet aggregation inhibitors

Also Published As

Publication number Publication date
JPH08231542A (ja) 1996-09-10
NO306114B1 (no) 1999-09-20
HU9503801D0 (en) 1996-02-28
SI0719775T1 (en) 2000-12-31
PT719775E (pt) 2000-12-29
AR002017A1 (es) 1998-01-07
IL116560A (en) 2001-03-19
ES2148458T3 (es) 2000-10-16
CZ346595A3 (en) 1996-08-14
JP3027110B2 (ja) 2000-03-27
NZ280720A (en) 1997-10-24
AU4070995A (en) 1996-07-04
NO955320D0 (no) 1995-12-27
NO955320L (no) 1996-07-01
TW418207B (en) 2001-01-11
US5607952A (en) 1997-03-04
RU2124515C1 (ru) 1999-01-10
FI956278A0 (fi) 1995-12-27
SK163395A3 (en) 1996-09-04
DE69517936T2 (de) 2001-04-19
SK281247B6 (sk) 2001-01-18
FR2728901A1 (fr) 1996-07-05
EP0719775A1 (fr) 1996-07-03
GR3034582T3 (en) 2001-01-31
BR1100524A (pt) 2000-03-14
CA2166165A1 (en) 1996-06-29
PL312078A1 (en) 1996-07-08
CN1133289A (zh) 1996-10-16
FI956278L (fi) 1996-06-29
ATE194616T1 (de) 2000-07-15
EP0719775B1 (fr) 2000-07-12
DE69517936D1 (de) 2000-08-17
AU703490B2 (en) 1999-03-25
FI956278A7 (fi) 1996-06-29
IL116560A0 (en) 1996-03-31
KR960022515A (ko) 1996-07-18
FR2728901B1 (fr) 1997-03-28
CN1048726C (zh) 2000-01-26
ZA9511029B (en) 1997-06-30
HUT75096A (en) 1997-04-28

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