DK0801655T3 - Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika - Google Patents

Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika

Info

Publication number: DK0801655T3
Authority: DK; Denmark
Prior art keywords: pct; antibiotics; basic; derivatives; sec
Prior art date: 1995-02-07

Application number

DK96903955T

Other languages

English (en)

Inventor

Sergio Lociuro

Pierfausto Seneci

Ermenegildo Restelli

Romeo Ciabatti

Original Assignee

Biosearch Italia Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-02-07

Filing date

1996-02-01

Publication date

1999-02-08

1996-02-01 Application filed by Biosearch Italia Spa filed Critical Biosearch Italia Spa

1999-02-08 Application granted granted Critical

1999-02-08 Publication of DK0801655T3 publication Critical patent/DK0801655T3/da

Links

239000003242 anti bacterial agent Substances 0.000 title abstract 2
229940088710 antibiotic agent Drugs 0.000 title abstract 2
VLJNHYLEOZPXFW-BYPYZUCNSA-N L-prolinamide Chemical class NC(=O)[C@@H]1CCCN1 VLJNHYLEOZPXFW-BYPYZUCNSA-N 0.000 title 1
150000001408 amides Chemical class 0.000 abstract 2
241000192125 Firmicutes Species 0.000 abstract 1
101000655610 Planobispora rosea Thiocillin GE2270 Proteins 0.000 abstract 1
239000004599 antimicrobial Substances 0.000 abstract 1
230000003115 biocidal effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Gastroenterology & Hepatology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)

DK96903955T 1995-02-07 1996-02-01 Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika DK0801655T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP95101597		1995-02-07
PCT/EP1996/000407 WO1996024607A1 (en)	1995-02-07	1996-02-01	Basic proline-amide derivatives of ge 2270 and ge 2270-like antibiotics

Publications (1)

Publication Number	Publication Date
DK0801655T3 true DK0801655T3 (da)	1999-02-08

Family

ID=8218961

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96903955T DK0801655T3 (da)	1995-02-07	1996-02-01	Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika

Country Status (12)

Country	Link
US (1)	US6143739A (da)
EP (1)	EP0801655B1 (da)
JP (1)	JP2825667B2 (da)
KR (1)	KR100381688B1 (da)
AT (1)	ATE165101T1 (da)
AU (1)	AU693995B2 (da)
CA (1)	CA2212372A1 (da)
DE (1)	DE69600244T2 (da)
DK (1)	DK0801655T3 (da)
ES (1)	ES2115424T3 (da)
SI (1)	SI0801655T1 (da)
WO (1)	WO1996024607A1 (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1996024608A1 (en) *	1995-02-07	1996-08-15	Biosearch Italia S.P.A.	Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics
DE69600244T2 (de) *	1995-02-07	1998-10-01	Biosearch Italia Spa	Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
ES2186866T3 (es) *	1996-02-14	2003-05-16	Biosearch Italia Spa	Derivados de factores del antibiotico ge2270.
CA2371618A1 (en) *	1999-04-28	2000-11-09	Yuji Ishihara	Cyclic amide compounds, their production and use
KR20050026401A (ko) *	2002-06-17	2005-03-15	비큐론 파마세티컬스 인코포레이티드	여드름 치료를 위한 ｇｅ 2270 인자 ａ3의 아미드유도체의 용도
US7119061B2 (en) *	2002-11-18	2006-10-10	Vicuron Pharmaceuticals, Inc.	Dalbavancin compositions for treatment of bacterial infections
US20060074014A1 (en) *	2002-11-18	2006-04-06	Vicuron Pharmaceuticals Inc.	Dalbavancin compositions for treatment of bacterial infections
MXPA05005338A (es) *	2002-11-18	2005-12-14	Vicuron Pharm Inc	Metodos para administrar dalbavancin para el tratamiento de infecciones bacterianas.
US8288606B2 (en) *	2005-03-08	2012-10-16	Ineos Usa Llc	Propylene polymer catalyst donor component
AR060977A1 (es) *	2006-05-31	2008-07-23	Novartis Ag	Aminotiazoles y sus usos
BRPI0720542A2 (pt) *	2006-12-20	2014-01-21	Novartis Ag	Compostos antibacterianos e processos para a sua produção
EP2229386B1 (en)	2007-12-12	2015-06-03	Novartis AG	An aminothiazole derivative as antibacterial agent

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5202241A (en) *	1988-09-09	1993-04-13	Gruppo Lepetit S.P.A.	Antibiotic GE 2270
DE69016284T2 (de) *	1989-07-04	1995-05-24	Lepetit Spa	Antibiotikum GE 22270, Faktoren A1,A2,A3 und H.
ES2071143T3 (es) *	1990-03-08	1995-06-16	Lepetit Spa	Factores b1, b2, c1, c2, d1, d2, e y t del antibiotico ge 2270.
IL100572A (en) *	1991-01-03	1997-01-10	Lepetit Spa	Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them
DK0529410T3 (da) *	1991-08-30	1998-05-11	Biosearch Italia Spa	Antibiotikum GE 2270 faktor C2a
WO1996024608A1 (en) *	1995-02-07	1996-08-15	Biosearch Italia S.P.A.	Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics
DE69600244T2 (de) *	1995-02-07	1998-10-01	Biosearch Italia Spa	Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
ES2186866T3 (es) *	1996-02-14	2003-05-16	Biosearch Italia Spa	Derivados de factores del antibiotico ge2270.

1996
- 1996-02-01 DE DE69600244T patent/DE69600244T2/de not_active Expired - Fee Related
- 1996-02-01 JP JP8523951A patent/JP2825667B2/ja not_active Expired - Fee Related
- 1996-02-01 DK DK96903955T patent/DK0801655T3/da active
- 1996-02-01 EP EP96903955A patent/EP0801655B1/en not_active Expired - Lifetime
- 1996-02-01 AU AU47858/96A patent/AU693995B2/en not_active Ceased
- 1996-02-01 WO PCT/EP1996/000407 patent/WO1996024607A1/en not_active Ceased
- 1996-02-01 KR KR1019970705393A patent/KR100381688B1/ko not_active Expired - Fee Related
- 1996-02-01 AT AT96903955T patent/ATE165101T1/de not_active IP Right Cessation
- 1996-02-01 US US08/875,707 patent/US6143739A/en not_active Expired - Fee Related
- 1996-02-01 ES ES96903955T patent/ES2115424T3/es not_active Expired - Lifetime
- 1996-02-01 CA CA002212372A patent/CA2212372A1/en not_active Abandoned
- 1996-02-01 SI SI9630006T patent/SI0801655T1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
JPH10504040A (ja)	1998-04-14
EP0801655B1 (en)	1998-04-15
SI0801655T1 (en)	1998-08-31
ES2115424T3 (es)	1998-06-16
AU693995B2 (en)	1998-07-09
KR19980701996A (ko)	1998-06-25
ATE165101T1 (de)	1998-05-15
WO1996024607A1 (en)	1996-08-15
CA2212372A1 (en)	1996-08-15
US6143739A (en)	2000-11-07
JP2825667B2 (ja)	1998-11-18
AU4785896A (en)	1996-08-27
KR100381688B1 (ko)	2003-12-11
DE69600244T2 (de)	1998-10-01
EP0801655A1 (en)	1997-10-22
DE69600244D1 (de)	1998-05-20

Publication	Publication Date	Title
NO996269L (no)	2000-02-16	Kinolin-indol antimikrobielle midler, samt anvendelse og blandinger derav
DK41193D0 (da)	1993-04-07	Ionkanalaabnere
MY119820A (en)	2005-07-29	Guanidine mimics as factor xa inhibitors
BR9611175B1 (pt)	2009-01-13	compostos e composiÇÕes farmacÊuticas.
BG103945A (bg)	2000-07-31	Производни на 4"-заместен-9-деоксо-9а-аза-9а- хомоеритромицин а
DE69729583D1 (de)	2004-07-22	N-(amidinophenyl)-n'-(subst.)-3h-2,4-benzodiazepin-3-on derivative als faktor xa inhibitoren
ES2153975T3 (es)	2001-03-16	Derivados de pirimidona con actividad antifungica.
TR199701654T1 (xx)	1998-05-21	4-Fenilaminotiyazol t�revleri.
TR200000059T2 (tr)	2000-06-21	Piridin türevleri
TR200200579T2 (tr)	2002-12-23	Amino-tirazolpiridin türevleri.
BG103947A (en)	2000-07-31	Derivatives of 9-oxymerythromycin
YU11997A (sh)	1999-09-27	Laktamski derivati i njihove farmaceutske kompozicije
NO20005400L (no)	2000-10-26	Kinoloner anvendt som MRS-inhibitorer og baktericider
MX9803650A (es)	1998-11-30	Agentes antimicrobianos de benzoxazina.
AU3973697A (en)	1998-03-06	Isoxazoline derivatives useful as antimicrobials
DK0801655T3 (da)	1999-02-08	Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika
GT199900208A (es)	2001-05-31	Antibiòticos cetòlidos carbamato y carbazato.
DK0808326T3 (da)	2001-10-01	Basiske oxazolinamidderivater af GE2270 og GE2270-lignende antibiotika
BR9609847A (pt)	1999-03-09	Derivados de N-(4-Benzila-substituída)-2-aminolactam
ATE219085T1 (de)	2002-06-15	2-beta-substituierte-6-alkylidenpenizillansäure derivate als beta-laktamase inhibitoren
DE69513837D1 (de)	2000-01-13	Cyklopeptolide
PL323305A1 (en)	1998-03-16	Applications of allyl amines
TR200001122T2 (tr)	2000-08-21	Farmasötikler olarak bifenil türevleri.
PL324884A1 (en)	1998-06-22	Application of prostane derivatives and their compositions with antibiotics in treating bacterial infections
TW349092B (en)	1999-01-01	Substituted indole derivatives