DK0801655T3 - Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika - Google Patents

Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika

Info

Publication number: DK0801655T3
Authority: DK; Denmark
Prior art keywords: pct; antibiotics; basic; derivatives; sec
Prior art date: 1995-02-07

Application number

DK96903955T

Other languages

English (en)

Inventor

Sergio Lociuro

Pierfausto Seneci

Ermenegildo Restelli

Romeo Ciabatti

Original Assignee

Biosearch Italia Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-02-07

Filing date

1996-02-01

Publication date

1999-02-08

1996-02-01 Application filed by Biosearch Italia Spa filed Critical Biosearch Italia Spa

1999-02-08 Application granted granted Critical

1999-02-08 Publication of DK0801655T3 publication Critical patent/DK0801655T3/da

Links

239000003242 anti bacterial agent Substances 0.000 title abstract 2
229940088710 antibiotic agent Drugs 0.000 title abstract 2
VLJNHYLEOZPXFW-BYPYZUCNSA-N L-prolinamide Chemical class NC(=O)[C@@H]1CCCN1 VLJNHYLEOZPXFW-BYPYZUCNSA-N 0.000 title 1
150000001408 amides Chemical class 0.000 abstract 2
241000192125 Firmicutes Species 0.000 abstract 1
101000655610 Planobispora rosea Thiocillin GE2270 Proteins 0.000 abstract 1
239000004599 antimicrobial Substances 0.000 abstract 1
230000003115 biocidal effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Gastroenterology & Hepatology (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Immunology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK96903955T 1995-02-07 1996-02-01 Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika DK0801655T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP95101597		1995-02-07
PCT/EP1996/000407 WO1996024607A1 (en)	1995-02-07	1996-02-01	Basic proline-amide derivatives of ge 2270 and ge 2270-like antibiotics

Publications (1)

Publication Number	Publication Date
DK0801655T3 true DK0801655T3 (da)	1999-02-08

Family

ID=8218961

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96903955T DK0801655T3 (da)	1995-02-07	1996-02-01	Basiske prolinamidderivater af GE 2270 og GE 2270-lignende antibiotika

Country Status (12)

Country	Link
US (1)	US6143739A (da)
EP (1)	EP0801655B1 (da)
JP (1)	JP2825667B2 (da)
KR (1)	KR100381688B1 (da)
AT (1)	ATE165101T1 (da)
AU (1)	AU693995B2 (da)
CA (1)	CA2212372A1 (da)
DE (1)	DE69600244T2 (da)
DK (1)	DK0801655T3 (da)
ES (1)	ES2115424T3 (da)
SI (1)	SI0801655T1 (da)
WO (1)	WO1996024607A1 (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE165101T1 (de) *	1995-02-07	1998-05-15	Biosearch Italia Spa	Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
JP3518606B2 (ja) *	1995-02-07	2004-04-12	バイオサーチ・イタリア・ソチエタ・ペル・アチオニ	Ｇｅ２２７０及びｇｅ２２７０−様抗生物質の塩基性オキサゾリン−アミド誘導体
EP0880541B1 (en) *	1996-02-14	2003-01-15	Biosearch Italia S.p.A.	Derivatives of antibiotic ge2270 factors
CA2371618A1 (en) *	1999-04-28	2000-11-09	Yuji Ishihara	Cyclic amide compounds, their production and use
DK1553967T3 (da) *	2002-06-17	2011-08-29	Naicons S C A R L	Anvendelse af et amidderivat af GE 2270 faktor A3 til behandling af acne
US20060074014A1 (en) *	2002-11-18	2006-04-06	Vicuron Pharmaceuticals Inc.	Dalbavancin compositions for treatment of bacterial infections
EP1565201B1 (en) *	2002-11-18	2018-10-31	Vicuron Pharmaceuticals, Inc.	Methods of administering dalbavancin for treatment of bacterial infections
US7119061B2 (en) *	2002-11-18	2006-10-10	Vicuron Pharmaceuticals, Inc.	Dalbavancin compositions for treatment of bacterial infections
US8288606B2 (en) *	2005-03-08	2012-10-16	Ineos Usa Llc	Propylene polymer catalyst donor component
PE20080103A1 (es) *	2006-05-31	2008-04-03	Novartis Ag	AMINOTIAZOLES COMO MODULADORES DEL FACTOR DE ELONGACION EF-Tu
WO2008082562A2 (en) *	2006-12-20	2008-07-10	Novartis Ag	Aminothiazole macrocycles, their use as antibacterial compounds and processes for their production
CA2708793C (en)	2007-12-12	2016-06-21	Novartis Ag	Aminothiazoles and their uses

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5202241A (en) *	1988-09-09	1993-04-13	Gruppo Lepetit S.P.A.	Antibiotic GE 2270
ES2066914T3 (es) *	1989-07-04	1995-03-16	Lepetit Spa	Factores a1, a2, a3 y h del antibiotico ge 2270.
DK0451486T3 (da) *	1990-03-08	1995-05-08	Lepetit Spa	Antibiotikum GE 2270 faktorer B1, B2, C1, C2, D1, D2, E og T
IL100572A (en) *	1991-01-03	1997-01-10	Lepetit Spa	Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them
DE69224497T2 (de) *	1991-08-30	1998-07-02	Biosearch Italia Spa	Faktor C2a des Antibiotikums CE 2270
ATE165101T1 (de) *	1995-02-07	1998-05-15	Biosearch Italia Spa	Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
JP3518606B2 (ja) *	1995-02-07	2004-04-12	バイオサーチ・イタリア・ソチエタ・ペル・アチオニ	Ｇｅ２２７０及びｇｅ２２７０−様抗生物質の塩基性オキサゾリン−アミド誘導体
EP0880541B1 (en) *	1996-02-14	2003-01-15	Biosearch Italia S.p.A.	Derivatives of antibiotic ge2270 factors

1996
- 1996-02-01 AT AT96903955T patent/ATE165101T1/de not_active IP Right Cessation
- 1996-02-01 KR KR1019970705393A patent/KR100381688B1/ko not_active Expired - Fee Related
- 1996-02-01 AU AU47858/96A patent/AU693995B2/en not_active Ceased
- 1996-02-01 ES ES96903955T patent/ES2115424T3/es not_active Expired - Lifetime
- 1996-02-01 DK DK96903955T patent/DK0801655T3/da active
- 1996-02-01 US US08/875,707 patent/US6143739A/en not_active Expired - Fee Related
- 1996-02-01 SI SI9630006T patent/SI0801655T1/xx not_active IP Right Cessation
- 1996-02-01 JP JP8523951A patent/JP2825667B2/ja not_active Expired - Fee Related
- 1996-02-01 CA CA002212372A patent/CA2212372A1/en not_active Abandoned
- 1996-02-01 DE DE69600244T patent/DE69600244T2/de not_active Expired - Fee Related
- 1996-02-01 EP EP96903955A patent/EP0801655B1/en not_active Expired - Lifetime
- 1996-02-01 WO PCT/EP1996/000407 patent/WO1996024607A1/en not_active Ceased

Also Published As

Publication number	Publication date
ATE165101T1 (de)	1998-05-15
KR100381688B1 (ko)	2003-12-11
JP2825667B2 (ja)	1998-11-18
ES2115424T3 (es)	1998-06-16
DE69600244T2 (de)	1998-10-01
EP0801655B1 (en)	1998-04-15
SI0801655T1 (en)	1998-08-31
AU4785896A (en)	1996-08-27
US6143739A (en)	2000-11-07
JPH10504040A (ja)	1998-04-14
DE69600244D1 (de)	1998-05-20
EP0801655A1 (en)	1997-10-22
AU693995B2 (en)	1998-07-09
CA2212372A1 (en)	1996-08-15
WO1996024607A1 (en)	1996-08-15
KR19980701996A (ko)	1998-06-25

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