DK0937714T3 - Fremgangsmåde til fremstilling af en optisk aktiv indolin-2-carboxylsyre eller et derivat deraf - Google Patents

Fremgangsmåde til fremstilling af en optisk aktiv indolin-2-carboxylsyre eller et derivat deraf

Info

Publication number: DK0937714T3
Authority: DK; Denmark
Prior art keywords: indoline; carboxylic acid; derivative; acid; acyl
Prior art date: 1998-02-13

Application number

DK99200383T

Other languages

Danish (da)

English (en)

Inventor

Andreas Joseph Johan Hendrickx

Thijs Kuilman

Original Assignee

Dsm Ip Assets Bv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-02-13

Filing date

1999-02-10

Publication date

2005-02-07

1999-02-10 Application filed by Dsm Ip Assets Bv filed Critical Dsm Ip Assets Bv

2005-02-07 Application granted granted Critical

2005-02-07 Publication of DK0937714T3 publication Critical patent/DK0937714T3/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Indole Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK99200383T 1998-02-13 1999-02-10 Fremgangsmåde til fremstilling af en optisk aktiv indolin-2-carboxylsyre eller et derivat deraf DK0937714T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
NL1008302A NL1008302C2 (nl)	1998-02-13	1998-02-13	Werkwijze voor de bereiding van een optisch actief indoline-2-carbonzuur of derivaat daarvan.

Publications (1)

Publication Number	Publication Date
DK0937714T3 true DK0937714T3 (da)	2005-02-07

Family

ID=19766536

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK99200383T DK0937714T3 (da)	1998-02-13	1999-02-10	Fremgangsmåde til fremstilling af en optisk aktiv indolin-2-carboxylsyre eller et derivat deraf

Country Status (14)

Country	Link
US (1)	US6121460A (2)
EP (1)	EP0937714B1 (2)
JP (1)	JPH11292844A (2)
CN (1)	CN100383119C (2)
AT (1)	ATE278668T1 (2)
CA (1)	CA2261453C (2)
DE (1)	DE69920784T2 (2)
DK (1)	DK0937714T3 (2)
ES (1)	ES2230794T3 (2)
HU (1)	HU222432B1 (2)
IL (1)	IL128462A (2)
IN (1)	IN188422B (2)
NL (1)	NL1008302C2 (2)
PT (1)	PT937714E (2)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2001266678A1 (en) *	2000-06-02	2001-12-17	Eli Lilly And Company	Methods for resolving chiral (2s) and (2r) chromanes
DE60301774T2 (de) *	2003-02-28	2006-07-20	Les Laboratoires Servier	Verfahren zur Synthese von (2S,3aS,7aS)-1-((S)-Alanyl)-octahydro-1H-indol-2-carbonsäurederivaten und Verwendung in der Synthese von Perindopril
ATE307801T1 (de) *	2003-02-28	2005-11-15	Servier Lab	Verfahren zur synthese des (2s,3as,7as)- perhydroindol-2-carbonsäures und seiner estern, verwendung in der synthese von perindopril
KR100710539B1 (ko)	2003-11-26	2007-04-24	에스케이 주식회사	가수분해 효소를 이용한 (ｓ)-인돌린-2-카르복실산 및이의 메틸 에스테르 화합물의 제조방법
EP1833789B1 (en) *	2004-12-28	2011-07-06	DSM IP Assets B.V.	Process for the preparation of enantiomerically enriched indoline-2-carboxylic acid
EP1676838A1 (en) *	2004-12-28	2006-07-05	DSM IP Assets B.V.	Process for the preparation of enantiomerically enriched indoline-2-carboxylic acid
EP1792896A1 (en)	2005-12-01	2007-06-06	KRKA, tovarna zdravil, d.d., Novo mesto	Process for the preparation of perindopril and salts thereof
US20100330625A1 (en) *	2008-02-06	2010-12-30	Mitsubishi Gas Chemical Company, Inc.	Process for production of optically active indoline-2-carboxylic acid or derivative thereof
CN102060745A (zh) *	2010-11-23	2011-05-18	安徽世华化工有限公司	一种(s)-吲哚啉-2-羧酸的制备方法
CN106631977A (zh) *	2016-11-11	2017-05-10	上海雅本化学有限公司	一种s‑吲哚啉‑2‑羧酸合成的优化方法
CN112375028A (zh) *	2020-12-14	2021-02-19	安徽美诺华药物化学有限公司	合成（2s）-二氢吲哚-甲酸的方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4665087A (en) *	1982-02-22	1987-05-12	Ciba-Geigy Corporation	1-(carbamyl, thiocarbamyl, and iminocarbamyl)-indoline derivatives
US4520205A (en) *	1982-06-28	1985-05-28	American Home Products Corporation	Chemical resolution of (+)-2,3-dihydroindole-2-carboxylic acid
JPH0798802B2 (ja) *	1984-07-13	1995-10-25	東レ株式会社	光学活性インドリン―２―カルボン酸の製造法
JPS6130572A (ja) *	1984-07-20	1986-02-12	Dainippon Pharmaceut Co Ltd	（ｒｓ）−１−アセチルインドリン−２−カルボン酸の光学分割法
US5166361A (en) *	1988-09-13	1992-11-24	Sepracor, Inc.	Methods for preparing captopril and its analogues
US5149821A (en) *	1990-10-11	1992-09-22	Pfizer Inc	Process and intermediates for optically active 3-formyltetrahydropyrans
JPH06130572A (ja) *	1992-10-22	1994-05-13	Konica Corp	ハロゲン化銀写真感光材料処理用錠剤状定着剤及び該定着剤を用いた処理方法

1998
- 1998-02-13 NL NL1008302A patent/NL1008302C2/nl not_active IP Right Cessation
1999
- 1999-02-10 ES ES99200383T patent/ES2230794T3/es not_active Expired - Lifetime
- 1999-02-10 AT AT99200383T patent/ATE278668T1/de not_active IP Right Cessation
- 1999-02-10 IL IL12846299A patent/IL128462A/xx not_active IP Right Cessation
- 1999-02-10 PT PT99200383T patent/PT937714E/pt unknown
- 1999-02-10 DE DE69920784T patent/DE69920784T2/de not_active Expired - Lifetime
- 1999-02-10 EP EP99200383A patent/EP0937714B1/en not_active Expired - Lifetime
- 1999-02-10 DK DK99200383T patent/DK0937714T3/da active
- 1999-02-11 CA CA002261453A patent/CA2261453C/en not_active Expired - Fee Related
- 1999-02-12 HU HU9900344A patent/HU222432B1/hu not_active IP Right Cessation
- 1999-02-12 IN IN179MA1999 patent/IN188422B/en unknown
- 1999-02-12 US US09/249,025 patent/US6121460A/en not_active Expired - Fee Related
- 1999-02-12 CN CNB991018923A patent/CN100383119C/zh not_active Expired - Fee Related
- 1999-02-15 JP JP11036063A patent/JPH11292844A/ja active Pending

Also Published As

Publication number	Publication date
CN100383119C (zh)	2008-04-23
IL128462A (en)	2003-07-31
DE69920784D1 (de)	2004-11-11
EP0937714A1 (en)	1999-08-25
IL128462A0 (en)	2000-01-31
CN1228423A (zh)	1999-09-15
HUP9900344A2 (hu)	1999-10-28
DE69920784T2 (de)	2005-11-03
HU222432B1 (hu)	2003-07-28
NL1008302C2 (nl)	1999-08-16
ATE278668T1 (de)	2004-10-15
PT937714E (pt)	2005-02-28
CA2261453C (en)	2009-05-12
IN188422B (2)	2002-09-21
EP0937714B1 (en)	2004-10-06
ES2230794T3 (es)	2005-05-01
JPH11292844A (ja)	1999-10-26
US6121460A (en)	2000-09-19
HU9900344D0 (en)	1999-04-28
CA2261453A1 (en)	1999-08-13
HUP9900344A3 (en)	2000-03-28

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