DK0952157T3 - 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin - Google Patents

9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin

Info

Publication number
DK0952157T3
DK0952157T3 DK99302289T DK99302289T DK0952157T3 DK 0952157 T3 DK0952157 T3 DK 0952157T3 DK 99302289 T DK99302289 T DK 99302289T DK 99302289 T DK99302289 T DK 99302289T DK 0952157 T3 DK0952157 T3 DK 0952157T3
Authority
DK
Denmark
Prior art keywords
methylerythromycin
keto
oxime
compounds
formula
Prior art date
Application number
DK99302289T
Other languages
English (en)
Inventor
Yong-Jin Wu
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK0952157T3 publication Critical patent/DK0952157T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Communicable Diseases (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Cephalosporin Compounds (AREA)
DK99302289T 1998-04-24 1999-03-25 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin DK0952157T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8292298P 1998-04-24 1998-04-24

Publications (1)

Publication Number Publication Date
DK0952157T3 true DK0952157T3 (da) 2003-10-13

Family

ID=22174315

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99302289T DK0952157T3 (da) 1998-04-24 1999-03-25 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin

Country Status (11)

Country Link
US (1) US6482801B2 (da)
EP (1) EP0952157B1 (da)
JP (1) JP3432448B2 (da)
AT (1) ATE243219T1 (da)
BR (1) BR9902049A (da)
CA (1) CA2270124C (da)
DE (1) DE69908855T2 (da)
DK (1) DK0952157T3 (da)
ES (1) ES2199524T3 (da)
MX (1) MXPA99003849A (da)
PT (1) PT952157E (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU775637B2 (en) * 1999-04-16 2004-08-12 Kosan Biosciences, Inc. Macrolide antiinfective agents
EP2435460B1 (en) * 2009-05-27 2015-01-07 Wockhardt Limited Ketolide compounds having antimicrobial activity

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0559896B1 (en) 1990-11-28 1997-08-27 Taisho Pharmaceutical Co. Ltd 6-o-methylerythromycin a derivative
ES2087737T3 (es) * 1992-04-22 1996-07-16 Taisho Pharmaceutical Co Ltd Un derivado 5-o-desosaminil-eritronoluro a.
FR2732023B1 (fr) * 1995-03-22 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
PT876388E (pt) * 1995-11-08 2004-07-30 Abbott Lab Derivados de eritromicina triciclica
DE69733439T2 (de) 1996-09-04 2006-05-04 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
PA8461401A1 (es) * 1997-10-29 2000-05-24 Pfizer Prod Inc Derivados de eritromicina triciclicos
US6248719B1 (en) * 1998-06-03 2001-06-19 Pfizer Inc Tricyclic 3-keto derivatives of 6-O-methylerthromycin

Also Published As

Publication number Publication date
DE69908855T2 (de) 2004-05-19
ES2199524T3 (es) 2004-02-16
EP0952157A1 (en) 1999-10-27
JP3432448B2 (ja) 2003-08-04
US6482801B2 (en) 2002-11-19
PT952157E (pt) 2003-11-28
JPH11322777A (ja) 1999-11-24
CA2270124C (en) 2002-07-09
ATE243219T1 (de) 2003-07-15
EP0952157B1 (en) 2003-06-18
MXPA99003849A (es) 2003-09-23
BR9902049A (pt) 2000-05-02
US20010016574A1 (en) 2001-08-23
DE69908855D1 (de) 2003-07-24
CA2270124A1 (en) 1999-10-24

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