DK105157C - Fremgangsmåde til fremstilling af Δ<1,4>-16-α-metylsteroider. - Google Patents

Fremgangsmåde til fremstilling af Δ<1,4>-16-α-metylsteroider.

Info

Publication number
DK105157C
DK105157C DK83062AA DK83062A DK105157C DK 105157 C DK105157 C DK 105157C DK 83062A A DK83062A A DK 83062AA DK 83062 A DK83062 A DK 83062A DK 105157 C DK105157 C DK 105157C
Authority
DK
Denmark
Prior art keywords
preparation
methyl steroids
steroids
methyl
Prior art date
Application number
DK83062AA
Other languages
English (en)
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Application granted granted Critical
Publication of DK105157C publication Critical patent/DK105157C/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/822—Microorganisms using bacteria or actinomycetales
    • Y10S435/832—Bacillus
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/822—Microorganisms using bacteria or actinomycetales
    • Y10S435/843—Corynebacterium
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
DK83062AA 1961-02-22 1962-02-22 Fremgangsmåde til fremstilling af Δ<1,4>-16-α-metylsteroider. DK105157C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DESCH29274A DE1169444B (de) 1961-02-22 1961-02-22 Verfahren zur Herstellung von ?-16ª‡-Methylsteroiden

Publications (1)

Publication Number Publication Date
DK105157C true DK105157C (da) 1966-08-29

Family

ID=7431375

Family Applications (1)

Application Number Title Priority Date Filing Date
DK83062AA DK105157C (da) 1961-02-22 1962-02-22 Fremgangsmåde til fremstilling af Δ<1,4>-16-α-metylsteroider.

Country Status (11)

Country Link
US (1) US3232839A (da)
BE (1) BE614196A (da)
BR (1) BR6236628D0 (da)
CH (1) CH416608A (da)
DE (1) DE1169444B (da)
DK (1) DK105157C (da)
FI (1) FI42958B (da)
FR (1) FR1916M (da)
GB (1) GB990384A (da)
NO (1) NO122590B (da)
SE (1) SE303283B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3426128A (en) * 1961-02-22 1969-02-04 Schering Ag Delta**1,4-16alpha-methyl steroids
GB1105013A (en) * 1964-12-01 1968-03-06 Organon Labor Ltd 17ª‡-alkyl steroids and a process for making them
CH513843A (fr) * 1969-04-23 1971-10-15 Lark Spa Procédé d'oxhydrilation microbiologique en position 11B
JPS5549078B2 (da) * 1972-12-27 1980-12-10
DE2712861C2 (de) * 1977-03-21 1986-02-27 Schering AG, 1000 Berlin und 4709 Bergkamen 17-Acetoxy-6-chlor-15&beta;-hydroxy-1&alpha;,2&alpha;-methylen-4,6-pregnadien-3,20-dion, Verfahren zu seiner Herstellung und dieses enthaltende Arzneimittel
DE2715853A1 (de) * 1977-04-06 1978-10-19 Schering Ag Wasserloesliche kortikoide
DE2920726A1 (de) * 1979-05-18 1980-11-27 Schering Ag Neue kortikoide, ihre herstellung und verwendung
FR2747680B1 (fr) * 1996-04-18 1998-07-03 Roussel Uclaf Nouveaux steroides, leur application a titre de medicaments, leur procede de preparation, les intermediaires de ce procede et les compositions pharmaceutiques les renfermant
US20130211069A1 (en) 2010-07-20 2013-08-15 Taro Pharmaceutical Industries Ltd. Process for the preparation of 17-desoxy-corticosteroids
CN107793460A (zh) * 2016-08-30 2018-03-13 天津太平洋制药有限公司 一种氟可龙的制备方法
CA3042428A1 (en) 2016-11-08 2018-05-17 Regeneron Pharmaceuticals, Inc. Steroids and protein-conjugates thereof
KR20250008984A (ko) 2017-05-18 2025-01-16 리제너론 파마슈티칼스 인코포레이티드 사이클로덱스트린 단백질 약물 접합체
CA3247730A1 (en) 2017-11-07 2025-10-30 Regeneron Pharmaceuticals, Inc. Hydrophilic linkers for antibody drug conjugates
MA50259A1 (fr) 2018-01-08 2021-07-29 Regeneron Pharma Stéroïdes et leurs conjugués-anticorps
WO2019217591A1 (en) 2018-05-09 2019-11-14 Regeneron Pharmaceuticals, Inc. Anti-msr1 antibodies and methods of use thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2876219A (en) * 1958-06-09 1959-03-03 Upjohn Co 6-fluoro-9alpha-halo-11-oxygenated-4-pregnenes and 6-fluoro-9alpha-halo-11-oxygenated-1,4-pregnadienes

Also Published As

Publication number Publication date
BE614196A (fr) 1962-08-21
BR6236628D0 (pt) 1973-05-31
FR1916M (fr) 1963-07-15
NO122590B (da) 1971-07-19
CH416608A (de) 1966-07-15
FI42958B (da) 1970-09-02
DE1169444B (de) 1964-05-06
US3232839A (en) 1966-02-01
GB990384A (en) 1965-04-28
SE303283B (da) 1968-08-26

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