DK1144408T3 - Substituerede N-(piperidin-4-yl)-4H-3,1-benzo(thia/oxa)zin-2-aminer, fremstilling deraf og terapeutisk anvendelse deraf - Google Patents

Substituerede N-(piperidin-4-yl)-4H-3,1-benzo(thia/oxa)zin-2-aminer, fremstilling deraf og terapeutisk anvendelse deraf

Info

Publication number
DK1144408T3
DK1144408T3 DK00900639T DK00900639T DK1144408T3 DK 1144408 T3 DK1144408 T3 DK 1144408T3 DK 00900639 T DK00900639 T DK 00900639T DK 00900639 T DK00900639 T DK 00900639T DK 1144408 T3 DK1144408 T3 DK 1144408T3
Authority
DK
Denmark
Prior art keywords
carbon atoms
branched
benzo
preparation
therapeutic use
Prior art date
Application number
DK00900639T
Other languages
English (en)
Inventor
Jean-Pierre Rieu
Jean-Francois Patoiseau
Gareth John
Bruno Legrand
Yvan Verscheure
Original Assignee
Pf Medicament
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pf Medicament filed Critical Pf Medicament
Application granted granted Critical
Publication of DK1144408T3 publication Critical patent/DK1144408T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
DK00900639T 1999-01-22 2000-01-21 Substituerede N-(piperidin-4-yl)-4H-3,1-benzo(thia/oxa)zin-2-aminer, fremstilling deraf og terapeutisk anvendelse deraf DK1144408T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9900706A FR2788775B1 (fr) 1999-01-22 1999-01-22 Nouvelles n-alcoyl-n-[1-(omega-(arylalcoyloxy)alcoyl] piperidin-4-yl]-4h-3,1-benzo(thia/oxa)zines-2-amines substituees, leur preparation et leur application en therapeutique
PCT/FR2000/000137 WO2000043391A1 (fr) 1999-01-22 2000-01-21 1-(piperidin-4-yl)-3-(aryl)-isothiourees substituees, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
DK1144408T3 true DK1144408T3 (da) 2003-02-03

Family

ID=9541133

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00900639T DK1144408T3 (da) 1999-01-22 2000-01-21 Substituerede N-(piperidin-4-yl)-4H-3,1-benzo(thia/oxa)zin-2-aminer, fremstilling deraf og terapeutisk anvendelse deraf

Country Status (15)

Country Link
US (1) US6531469B1 (da)
EP (1) EP1144408B1 (da)
JP (1) JP2002535329A (da)
CN (1) CN1129599C (da)
AT (1) ATE224892T1 (da)
AU (1) AU767132B2 (da)
BR (1) BR0007674A (da)
CA (1) CA2359103A1 (da)
DE (1) DE60000500T2 (da)
DK (1) DK1144408T3 (da)
ES (1) ES2182770T3 (da)
FR (1) FR2788775B1 (da)
PT (1) PT1144408E (da)
WO (1) WO2000043391A1 (da)
ZA (1) ZA200105921B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR900701170A (ko) * 1988-09-29 1990-12-01 클러런스 제이 모이에 육류보존법 및 육류보존 물질
EP0982300A3 (en) * 1998-07-29 2000-03-08 Societe Civile Bioprojet Non-imidazole alkylamines as histamine H3 - receptor ligands and their therapeutic applications
FR2821356A1 (fr) * 2001-02-23 2002-08-30 Cerep Nouveaux derives d'arylcarbamates et d'arylurees, preparations et utilisations
FR3001151B1 (fr) 2013-01-21 2016-04-08 Pf Medicament Association d'un bloqueur de courant sodique lent et d'un inhibiteur du courant if sinusal et les compositions pharmarceutiques la contenant
DK2970123T4 (da) * 2013-03-14 2026-01-26 Amgen Inc Krystallinsk dihydrochloridhydratsalt af omecamtiv mecarbil og fremgangsmåde til fremstilling heraf
CN114349745B (zh) * 2022-01-14 2023-12-08 黑龙江中医药大学 一种用于治疗心肌缺血的药物及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2737207B1 (fr) * 1995-07-26 1997-10-17 Pf Medicament Nouvelles n-heterocyclyl-1-aryloxyalcoyl-4-piperidinamines substituees, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
AU3058100A (en) 2000-08-07
BR0007674A (pt) 2001-11-20
PT1144408E (pt) 2003-02-28
DE60000500D1 (de) 2002-10-31
FR2788775A1 (fr) 2000-07-28
DE60000500T2 (de) 2003-07-31
CA2359103A1 (fr) 2000-07-27
AU767132B2 (en) 2003-10-30
WO2000043391A1 (fr) 2000-07-27
CN1129599C (zh) 2003-12-03
FR2788775B1 (fr) 2001-04-13
ATE224892T1 (de) 2002-10-15
ZA200105921B (en) 2002-05-08
ES2182770T3 (es) 2003-03-16
US6531469B1 (en) 2003-03-11
EP1144408B1 (fr) 2002-09-25
EP1144408A1 (fr) 2001-10-17
CN1344267A (zh) 2002-04-10
JP2002535329A (ja) 2002-10-22

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