DK126785B - Analogifremgangsmåde til fremstilling af 2-[2-(3-hydroxyphenyl)-vinyl eller -ethyl]-imidazoliner eller de tilsvarende 2-tetrahydropyrimidiner eller syreadditionssalte af disse forbindelser. - Google Patents

Analogifremgangsmåde til fremstilling af 2-[2-(3-hydroxyphenyl)-vinyl eller -ethyl]-imidazoliner eller de tilsvarende 2-tetrahydropyrimidiner eller syreadditionssalte af disse forbindelser.

Info

Publication number
DK126785B
DK126785B DK85470AA DK85470A DK126785B DK 126785 B DK126785 B DK 126785B DK 85470A A DK85470A A DK 85470AA DK 85470 A DK85470 A DK 85470A DK 126785 B DK126785 B DK 126785B
Authority
DK
Denmark
Prior art keywords
tetrahydropyrimidines
imidazolines
hydroxyphenyl
vinyl
ethyl
Prior art date
Application number
DK85470AA
Other languages
English (en)
Inventor
J Mcfarland
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK126785B publication Critical patent/DK126785B/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C243/24—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids
    • C07C243/26—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C243/34—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of a carbon skeleton further substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/12—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines
    • C07C259/14—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines having carbon atoms of hydroxamidine groups bound to hydrogen atoms or to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/42—Unsaturated compounds containing hydroxy or O-metal groups
    • C07C59/52—Unsaturated compounds containing hydroxy or O-metal groups a hydroxy or O-metal group being bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/01—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
    • C07C65/03—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups monocyclic and having all hydroxy or O-metal groups bound to the ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D233/22—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D233/24—Radicals substituted by nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK85470AA 1967-08-30 1970-02-20 Analogifremgangsmåde til fremstilling af 2-[2-(3-hydroxyphenyl)-vinyl eller -ethyl]-imidazoliner eller de tilsvarende 2-tetrahydropyrimidiner eller syreadditionssalte af disse forbindelser. DK126785B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US66425867A 1967-08-30 1967-08-30

Publications (1)

Publication Number Publication Date
DK126785B true DK126785B (da) 1973-08-20

Family

ID=24665273

Family Applications (2)

Application Number Title Priority Date Filing Date
DK366168AA DK123710B (da) 1967-08-30 1968-07-29 Analogifremgangsmåde til fremstilling af N,N-dimethyl-3-(3-hydroxyphenyl)-propionamidiner eller -acrylamidiner eller syreadditionssalte deraf.
DK85470AA DK126785B (da) 1967-08-30 1970-02-20 Analogifremgangsmåde til fremstilling af 2-[2-(3-hydroxyphenyl)-vinyl eller -ethyl]-imidazoliner eller de tilsvarende 2-tetrahydropyrimidiner eller syreadditionssalte af disse forbindelser.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK366168AA DK123710B (da) 1967-08-30 1968-07-29 Analogifremgangsmåde til fremstilling af N,N-dimethyl-3-(3-hydroxyphenyl)-propionamidiner eller -acrylamidiner eller syreadditionssalte deraf.

Country Status (11)

Country Link
US (1) US3579510A (da)
JP (1) JPS4813108B1 (da)
BR (1) BR6801003D0 (da)
DE (1) DE1793050C3 (da)
DK (2) DK123710B (da)
FR (2) FR1584069A (da)
GB (1) GB1168361A (da)
IL (1) IL30383A (da)
NL (1) NL162074C (da)
NO (1) NO126440B (da)
SE (1) SE349579B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3930001A (en) * 1971-11-30 1975-12-30 Pfizer 2-(Substituted)-5,6-dihydro-4H-1,4-thiazines used for the control of rice blast
US3890443A (en) * 1973-09-17 1975-06-17 Pfizer 2-(Substituted) thiazolines for the control of rice blast
US4490388A (en) * 1981-02-27 1984-12-25 Torii & Co., Ltd. Amidine compound and anticomplement agent comprising same
DE3211301A1 (de) * 1982-03-26 1983-09-29 Bayer Ag, 5090 Leverkusen Cyclische amidine, verfahren zu ihrer herstellung und die verwendung cyclischer amidine als katalysatoren fuer die haertung von epoxidharzen
WO1995007100A1 (en) * 1993-09-10 1995-03-16 Petrovax L.L.C. Compounds for the prevention and treatment of helminth infections

Also Published As

Publication number Publication date
BR6801003D0 (pt) 1973-07-03
NO126440B (da) 1973-02-05
DE1793050A1 (de) 1971-12-16
DE1793050C3 (de) 1975-09-11
SE349579B (da) 1972-10-02
FR1584069A (da) 1969-12-12
US3579510A (en) 1971-05-18
NL162074B (nl) 1979-11-15
GB1168361A (en) 1969-10-22
NL162074C (nl) 1980-04-15
JPS4813108B1 (da) 1973-04-25
IL30383A0 (en) 1968-09-26
FR7991M (da) 1970-06-08
IL30383A (en) 1973-02-28
DE1793050B2 (de) 1975-01-23
NL6810601A (da) 1969-03-04
DK123710B (da) 1972-07-24

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