DK131033B - Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon. - Google Patents

Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon.

Info

Publication number
DK131033B
DK131033B DK247673AA DK247673A DK131033B DK 131033 B DK131033 B DK 131033B DK 247673A A DK247673A A DK 247673AA DK 247673 A DK247673 A DK 247673A DK 131033 B DK131033 B DK 131033B
Authority
DK
Denmark
Prior art keywords
sulfamyl
quinazolinone
tetrahydro
chloro
phenyl
Prior art date
Application number
DK247673AA
Other languages
English (en)
Other versions
DK131033C (da
Inventor
M Carissimi
F Ravenna
Original Assignee
Maggioni & C Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Maggioni & C Spa filed Critical Maggioni & C Spa
Publication of DK131033B publication Critical patent/DK131033B/da
Application granted granted Critical
Publication of DK131033C publication Critical patent/DK131033C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK247673AA 1972-05-05 1973-05-04 Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon. DK131033B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT2392572 1972-05-05

Publications (2)

Publication Number Publication Date
DK131033B true DK131033B (da) 1975-05-20
DK131033C DK131033C (da) 1975-10-06

Family

ID=11210914

Family Applications (1)

Application Number Title Priority Date Filing Date
DK247673AA DK131033B (da) 1972-05-05 1973-05-04 Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon.

Country Status (12)

Country Link
US (1) US3870720A (da)
JP (1) JPS49132221A (da)
AU (1) AU469087B2 (da)
BE (1) BE799087A (da)
CA (1) CA982578A (da)
DE (1) DE2322699C2 (da)
DK (1) DK131033B (da)
FR (1) FR2183806B1 (da)
GB (1) GB1413008A (da)
NL (1) NL7306164A (da)
SE (1) SE400768B (da)
ZA (1) ZA732937B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA200500234A1 (ru) 2002-08-19 2005-08-25 Пфайзер Продактс Инк. Комбинированная терапия гиперпролиферативных болезней
US20060063803A1 (en) * 2004-09-23 2006-03-23 Pfizer Inc 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
ATE547394T1 (de) 2006-12-01 2012-03-15 Bristol Myers Squibb Co N-((3-benzyl)-2,2-(bis-phenyl)-propan-1- aminderivate als cetp-hemmer für die behandlung von atherosklerose und herz-kreislauf- erkrankungen
CN105143203A (zh) 2013-04-17 2015-12-09 辉瑞大药厂 用于治疗心血管疾病的n-哌啶-3-基苯甲酰胺衍生物
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
WO2020150473A2 (en) 2019-01-18 2020-07-23 Dogma Therapeutics, Inc. Pcsk9 inhibitors and methods of use thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2952680A (en) * 1960-09-13 Derivatives of x-quevazolone
US987847A (en) * 1910-04-12 1911-03-28 Rubin W Weeks Harness.
US3440244A (en) * 1958-02-17 1969-04-22 Pfizer & Co C 3,6-disubstituted-7-sulfamyl-1,2,4-benzthiazide-1,1-dioxides
US3072656A (en) * 1960-01-22 1963-01-08 Ciba Geigy Corp 2-cycloaliphatic-6-sulfamyl-7-halo(or trihalomethyl)-1, 2, 3, 4-tetrahydro-4-quinazolones
US3360518A (en) * 1966-01-03 1967-12-26 Wallace & Tiernan Inc Tetrahydro-halo-sulfamyl quinazolinones

Also Published As

Publication number Publication date
BE799087A (fr) 1973-08-31
FR2183806A1 (da) 1973-12-21
AU5516173A (en) 1974-11-07
DE2322699A1 (de) 1974-01-10
DE2322699C2 (de) 1983-10-27
ZA732937B (en) 1974-03-27
FR2183806B1 (da) 1976-05-14
GB1413008A (en) 1975-11-05
SE400768B (sv) 1978-04-10
NL7306164A (da) 1973-11-07
JPS49132221A (da) 1974-12-18
CA982578A (en) 1976-01-27
AU469087B2 (en) 1976-02-05
DK131033C (da) 1975-10-06
US3870720A (en) 1975-03-11

Similar Documents

Publication Publication Date Title
DK138951B (da) Fremgangsmåde til fremstilling af N-phosphonomethyl-glycin.
DK137329B (da) Analogifremgangsmåde til fremstilling af 2-karbalkoksyaminobenzimidazolderivater.
DK131725B (da) Analogifremgangsmåde til fremstilling af 2,4-diaminoquinazoliner eller salte deraf.
DK135454B (da) Analogifremgangsmåde til fremstilling af 2,1,3-benzothiadiazolderivater.
DK132408B (da) Fremgangsmåde til fremstilling af benzo-1,2,4-triazin-di-N-oxider (1,4).
DK134490B (da) Analogifremgangsmåde til fremstilling af 2,6-diaminonebularin-derivater.
DK132500B (da) Analogifremgangsmåde til fremstilling af 2beta, 16beta-diamino-5alfa-androstaner.
DK134604B (da) Fremgangsmåde til fremstilling af indenyl-3-acetoglucuronider.
DK138230B (da) Analogifremgangsmåde til fremstilling af vincanolsalte.
DK137639B (da) Analogifremgangsmåde til fremstilling af 1-aminomethyl-2,2-diaryl-cyclopropancarboxamider.
DK138796B (da) Analogifremgangsmåde til fremstilling af 2-carboxypyrazin-4-oxidderivater.
DK138898B (da) Fremgangsmåde til fremstilling af N-phosphonomethylglycin.
DK131575B (da) Analogifremgangsmåde til fremstilling af 2beta-hydroxy-3alfa-aminosteroider.
DK138645B (da) Analogifremgangsmåde til fremstilling af sulfamoylfenyl-imidazolidiner.
DK135122B (da) Analogifremgangsmåde til fremstilling af 4-aryl-5-aminoalkyl-4-oxazolin-2-onderivater.
DK131864B (da) Fremgangsmåde til fremstilling af pregnan-21-syrederivater.
DK131855B (da) Fremgangsmåde til fremstilling af 3,4-dihydropyridoner.
DK135166B (da) Analogifremgangsmåde til fremstilling af 2-methyl-5-nitro-imidazoler.
DK132410B (da) Analogifremgangsmåde til fremstilling af 2-amino-4H-pyraner.
DK129657B (da) Analogifremgangsmåde til fremstilling af 3-methylpyrazol-5-carboxamider.
DK132329B (da) Fremgangsmåde til fremstilling af cardenolid-3,alfa-/2'-desoxy-glycosider/.
DK132032B (da) Analogifremgangsmåde til fremstilling af 15alfa,16alfa-methylen-4-pregnener.
DK139225B (da) Fremgangsmåde til fremstilling af morphanthridiner.
DK139677B (da) Fremgangsmåde til fremstilling af 7-benzoylindolin-2-oner.
DK134236B (da) Analogifremgangsmåde til fremstilling af 3-cycloalkoxy-16alfa-cyanopregn-5-en-20-oner.

Legal Events

Date Code Title Description
PBP Patent lapsed