DK1423385T3 - Mellemprodukter til fremstilling af neuraminidaseinhibitorkonjugater - Google Patents

Mellemprodukter til fremstilling af neuraminidaseinhibitorkonjugater

Info

Publication number
DK1423385T3
DK1423385T3 DK02759906T DK02759906T DK1423385T3 DK 1423385 T3 DK1423385 T3 DK 1423385T3 DK 02759906 T DK02759906 T DK 02759906T DK 02759906 T DK02759906 T DK 02759906T DK 1423385 T3 DK1423385 T3 DK 1423385T3
Authority
DK
Denmark
Prior art keywords
sub
preparation
intermediates
neuraminidase inhibitor
inhibitor conjugates
Prior art date
Application number
DK02759906T
Other languages
English (en)
Inventor
Brian David Judkins
Simon John Fawcett Macdonald
Derek Anthony Demaine
Graham George Adam Inglis
Julie Nicole Hamblin
Original Assignee
Biota Scient Management
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biota Scient Management filed Critical Biota Scient Management
Application granted granted Critical
Publication of DK1423385T3 publication Critical patent/DK1423385T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/06Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrane Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK02759906T 2001-09-07 2002-08-30 Mellemprodukter til fremstilling af neuraminidaseinhibitorkonjugater DK1423385T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AUPR757401 2001-09-07
PCT/AU2002/001187 WO2003022841A1 (en) 2001-09-07 2002-08-30 Intermediates for preparing neuraminidase inhibitor conjugates

Publications (1)

Publication Number Publication Date
DK1423385T3 true DK1423385T3 (da) 2008-11-03

Family

ID=3831510

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02759906T DK1423385T3 (da) 2001-09-07 2002-08-30 Mellemprodukter til fremstilling af neuraminidaseinhibitorkonjugater

Country Status (12)

Country Link
US (1) US7230114B2 (da)
EP (1) EP1423385B1 (da)
JP (1) JP4463553B2 (da)
AT (1) ATE399779T1 (da)
BR (1) BR0212261A (da)
CA (1) CA2456239C (da)
DE (1) DE60227386D1 (da)
DK (1) DK1423385T3 (da)
ES (1) ES2307776T3 (da)
MX (1) MXPA04002141A (da)
PT (1) PT1423385E (da)
WO (1) WO2003022841A1 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104418876B (zh) * 2013-09-09 2019-05-17 中国科学院上海有机化学研究所 扎那米韦和拉那米韦的中间体及其合成方法
CN113461631B (zh) * 2021-06-29 2022-10-14 上海应用技术大学 一种1,3,4-恶二唑类神经氨酸酶抑制剂及其制备方法与应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9516276D0 (en) 1995-08-08 1995-10-11 Biota Scient Management Chemical compounds
CA2245680C (en) * 1996-03-01 2005-09-27 Biota Scientific Management Pty. Ltd. Method of detection of influenza virus and compounds for use therein
CN1126752C (zh) * 1996-08-13 2003-11-05 三共株式会社 神经氨酸化合物
AUPR001000A0 (en) * 2000-09-08 2000-10-05 Biota Scientific Management Pty Ltd Novel chemical compounds and their use

Also Published As

Publication number Publication date
CA2456239A1 (en) 2003-03-20
BR0212261A (pt) 2004-10-19
PT1423385E (pt) 2008-09-24
WO2003022841A1 (en) 2003-03-20
EP1423385A1 (en) 2004-06-02
EP1423385B1 (en) 2008-07-02
ATE399779T1 (de) 2008-07-15
JP4463553B2 (ja) 2010-05-19
JP2005501921A (ja) 2005-01-20
US20050032853A1 (en) 2005-02-10
US7230114B2 (en) 2007-06-12
CA2456239C (en) 2010-11-30
EP1423385A4 (en) 2004-12-01
MXPA04002141A (es) 2004-07-23
ES2307776T3 (es) 2008-12-01
DE60227386D1 (de) 2008-08-14

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