DK1440977T3 - Forbedret fremgangsmåde til fremstilling af diamidderivater af tripeptidet KPV - Google Patents

Forbedret fremgangsmåde til fremstilling af diamidderivater af tripeptidet KPV

Info

Publication number: DK1440977T3
Authority: DK; Denmark
Prior art keywords: optionally; formula; alkyl; proline; compound
Prior art date: 2003-01-24

Application number

DK04300039T

Other languages

English (en)

Inventor

Sylvie Genard

Original Assignee

Oreal

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-01-24

Filing date

2004-01-22

Publication date

2006-11-20

2004-01-22 Application filed by Oreal filed Critical Oreal

2006-11-20 Application granted granted Critical

2006-11-20 Publication of DK1440977T3 publication Critical patent/DK1440977T3/da

Links

150000001470 diamides Chemical class 0.000 title abstract 3
-1 N,N'-diprotected lysine compound Chemical class 0.000 abstract 9
125000000217 alkyl group Chemical group 0.000 abstract 6
125000005842 heteroatom Chemical group 0.000 abstract 4
229910052757 nitrogen Inorganic materials 0.000 abstract 4
229910052760 oxygen Inorganic materials 0.000 abstract 4
125000006239 protecting group Chemical group 0.000 abstract 4
229910052717 sulfur Inorganic materials 0.000 abstract 4
230000008878 coupling Effects 0.000 abstract 3
238000010168 coupling process Methods 0.000 abstract 3
238000005859 coupling reaction Methods 0.000 abstract 3
229910052500 inorganic mineral Inorganic materials 0.000 abstract 3
239000011707 mineral Substances 0.000 abstract 3
125000003710 aryl alkyl group Chemical group 0.000 abstract 2
125000003118 aryl group Chemical group 0.000 abstract 2
230000015572 biosynthetic process Effects 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000000753 cycloalkyl group Chemical group 0.000 abstract 2
125000005843 halogen group Chemical group 0.000 abstract 2
150000007522 mineralic acids Chemical class 0.000 abstract 2
150000007524 organic acids Chemical class 0.000 abstract 2
125000001500 prolyl group Chemical group [H]N1C([H])(C(=O)[*])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
229920006395 saturated elastomer Polymers 0.000 abstract 2
229910052710 silicon Inorganic materials 0.000 abstract 2
238000003786 synthesis reaction Methods 0.000 abstract 2
239000004474 valine Substances 0.000 abstract 2
NGNBDVOYPDDBFK-UHFFFAOYSA-N 2-[2,4-di(pentan-2-yl)phenoxy]acetyl chloride Chemical compound CCCC(C)C1=CC=C(OCC(Cl)=O)C(C(C)CCC)=C1 NGNBDVOYPDDBFK-UHFFFAOYSA-N 0.000 abstract 1
108010016626 Dipeptides Proteins 0.000 abstract 1
KDXKERNSBIXSRK-UHFFFAOYSA-N Lysine Natural products NCCCCC(N)C(O)=O KDXKERNSBIXSRK-UHFFFAOYSA-N 0.000 abstract 1
239000004472 Lysine Substances 0.000 abstract 1
ONIBWKKTOPOVIA-UHFFFAOYSA-N Proline Natural products OC(=O)C1CCCN1 ONIBWKKTOPOVIA-UHFFFAOYSA-N 0.000 abstract 1
230000003213 activating effect Effects 0.000 abstract 1
235000001014 amino acid Nutrition 0.000 abstract 1
150000001413 amino acids Chemical class 0.000 abstract 1
150000008064 anhydrides Chemical class 0.000 abstract 1
210000004899 c-terminal region Anatomy 0.000 abstract 1
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
239000003153 chemical reaction reagent Substances 0.000 abstract 1
150000007530 organic bases Chemical class 0.000 abstract 1
108090000765 processed proteins & peptides Proteins 0.000 abstract 1
239000002904 solvent Substances 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/64—Proteins; Peptides; Derivatives or degradation products thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/005—Preparations for sensitive skin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/007—Preparations for dry skin
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0815—Tripeptides with the first amino acid being basic
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Dermatology (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
Genetics & Genomics (AREA)
Proteomics, Peptides & Aminoacids (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Molecular Biology (AREA)
Birds (AREA)
Epidemiology (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Cosmetics (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Saccharide Compounds (AREA)

DK04300039T 2003-01-24 2004-01-22 Forbedret fremgangsmåde til fremstilling af diamidderivater af tripeptidet KPV DK1440977T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0300808A FR2850383B1 (fr)	2003-01-24	2003-01-24	Procede de synthese ameliore de derives diamides du tripeptide kpv

Publications (1)

Publication Number	Publication Date
DK1440977T3 true DK1440977T3 (da)	2006-11-20

Family

ID=32525006

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK04300039T DK1440977T3 (da)	2003-01-24	2004-01-22	Forbedret fremgangsmåde til fremstilling af diamidderivater af tripeptidet KPV

Country Status (10)

Country	Link
EP (1)	EP1440977B1 (da)
JP (1)	JP4050238B2 (da)
AT (1)	ATE334142T1 (da)
CY (1)	CY1105713T1 (da)
DE (1)	DE602004001590T2 (da)
DK (1)	DK1440977T3 (da)
ES (1)	ES2270318T3 (da)
FR (1)	FR2850383B1 (da)
PT (1)	PT1440977E (da)
SI (1)	SI1440977T1 (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN122036841A (zh) *	2026-03-10	2026-05-15	上海中翊日化有限公司	一种环三肽-5的液相合成工艺

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1988000833A2 (en) *	1986-08-08	1988-02-11	Board Of Regents, The University Of Texas System	Antipyretic and anti-inflammatory peptides
WO2002069884A2 (en) *	2000-11-01	2002-09-12	Zengen, Inc.	A sunburn treatment and sunburn prevention method

2003
- 2003-01-24 FR FR0300808A patent/FR2850383B1/fr not_active Expired - Fee Related
2004
- 2004-01-22 DK DK04300039T patent/DK1440977T3/da active
- 2004-01-22 EP EP04300039A patent/EP1440977B1/fr not_active Expired - Lifetime
- 2004-01-22 PT PT04300039T patent/PT1440977E/pt unknown
- 2004-01-22 DE DE602004001590T patent/DE602004001590T2/de not_active Expired - Lifetime
- 2004-01-22 ES ES04300039T patent/ES2270318T3/es not_active Expired - Lifetime
- 2004-01-22 AT AT04300039T patent/ATE334142T1/de not_active IP Right Cessation
- 2004-01-22 SI SI200430088T patent/SI1440977T1/sl unknown
- 2004-01-26 JP JP2004017359A patent/JP4050238B2/ja not_active Expired - Fee Related
2006
- 2006-10-19 CY CY20061101497T patent/CY1105713T1/el unknown

Also Published As

Publication number	Publication date
ES2270318T3 (es)	2007-04-01
CY1105713T1 (el)	2010-12-22
JP4050238B2 (ja)	2008-02-20
DE602004001590T2 (de)	2007-07-19
ATE334142T1 (de)	2006-08-15
DE602004001590D1 (de)	2006-09-07
JP2004231653A (ja)	2004-08-19
PT1440977E (pt)	2006-12-29
SI1440977T1 (sl)	2006-12-31
EP1440977B1 (fr)	2006-07-26
FR2850383B1 (fr)	2005-04-15
FR2850383A1 (fr)	2004-07-30
EP1440977A1 (fr)	2004-07-28

Publication	Publication Date	Title
CA2200192C (en)	2001-01-16	Amidino and guanidino substituted inhibitors of trypsin-like enzymes
US6846806B2 (en)	2005-01-25	Peptide inhibitors of Hepatitis C virus NS3 protein
CA2098166A1 (en)	1993-12-26	Hydroxamic acid derivatives
ATE90107T1 (de)	1993-06-15	Peptide mit collagenase hemmender wirkung.
DE69315079D1 (de)	1997-12-11	Beta-aminoalkyl und beta-n-peptidylaminoalkylborsäure
CA1244041A (en)	1988-11-01	Process for the preparation of cis, endo- octahydrocyclopenta¬b\|pyrrole-2-carboxylate
JPH0144693B2 (da)	1989-09-29
PE20061427A1 (es)	2007-01-11	Metodos para identificar objetivos terapeuticos para el tratamiento de la atrofia vulvovaginal
DE69636987D1 (de)	2007-05-03	Mittel zur förderung von knochenbildung
DK0910575T3 (da)	2003-02-03	Fremgangsmåde til fremstilling af peptider
US5462964A (en)	1995-10-31	Dipeptide boronic acid inhibitors of trypsin-like enzymes
Li et al.	2000	Highly efficient synthesis of sterically hindered peptides containing N-methylated amino acid residues using a novel 1H-benzimidazolium salt
Pearson et al.	2006	Photoswitch inhibitors of α-chymotrypsin—increased substitution and peptidic character in peptidomimetic boronate esters
SI1440977T1 (sl)	2006-12-31	Postopek za izboljsano pripravo diamidnih derivatov tripeptida KPV
EP1160236A2 (en)	2001-12-05	Production of mixed acid anhydride and amine compound
US3095408A (en)	1963-06-25	Processes in peptide synthesis
AU8294401A (en)	2002-02-25	A process for the preparation of alpha' chloroketones
US2617793A (en)	1952-11-11	Method of preparing amides
Awahara et al.	2014	Effect of prime-site sequence of retro-inverso-modified HTLV-1 protease inhibitor
JPS59231061A (ja)	1984-12-25	アミノ酸誘導体及びその製造方法
DE19721290A1 (de)	1997-12-11	Verfahren zur Herstellung von Verbindungen mit ACE-Hemmwirkung
Green et al.	2000	Substrate related O, O-dialkyldipeptidyly ψ carboxybenzylphosphonates, a new type of thrombin inhibitor
ATE473208T1 (de)	2010-07-15	Isodipeptid als syntheseeinheit zur herstellung von peptiden
US2673871A (en)	1954-03-30	Diesterphosphiteamides of aminoacid derivatives
GB872332A (en)	1961-07-05	Derivatives of amino acids and peptides, and synthesis of peptides