DK162220C - Tricykliske pyridazinderivater, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling af derivaterne, og laegemidler, hvori de er til stede - Google Patents

Tricykliske pyridazinderivater, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling af derivaterne, og laegemidler, hvori de er til stede

Info

Publication number: DK162220C
Authority: DK; Denmark
Prior art keywords: derivatives; cholinerge; tricyclic; agonists; receptors
Prior art date: 1986-07-03

Application number

DK340987A

Other languages

English (en)

Other versions

DK340987D0 (da

DK162220B (da

DK340987A (da

Inventor

Kathleen Biziere

Camille Georges Wermuth

Paul Worms

Jean-Jacques Bourguignon

Original Assignee

Sanofi Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-07-03

Filing date

1987-07-02

Publication date

1992-03-02

1987-07-02 Application filed by Sanofi Sa filed Critical Sanofi Sa

1987-07-02 Publication of DK340987D0 publication Critical patent/DK340987D0/da

1988-01-04 Publication of DK340987A publication Critical patent/DK340987A/da

1991-09-30 Publication of DK162220B publication Critical patent/DK162220B/da

1992-03-02 Application granted granted Critical

1992-03-02 Publication of DK162220C publication Critical patent/DK162220C/da

Links

239000000556 agonist Substances 0.000 title 1
229940126601 medicinal product Drugs 0.000 title 1
238000000034 method Methods 0.000 title 1
PBMFSQRYOILNGV-UHFFFAOYSA-N pyridazine Chemical class C1=CC=NN=C1 PBMFSQRYOILNGV-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
- C07D237/36—Benzo-cinnolines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

DK340987A 1986-07-03 1987-07-02 Tricykliske pyridazinderivater, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling af derivaterne, og laegemidler, hvori de er til stede DK162220C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8609681		1986-07-03
FR8609681A FR2601011B1 (fr)	1986-07-03	1986-07-03	Nouveaux derives tricycliques agonistes des recepteurs cholinergiques et medicaments en contenant

Publications (4)

Publication Number	Publication Date
DK340987D0 DK340987D0 (da)	1987-07-02
DK340987A DK340987A (da)	1988-01-04
DK162220B DK162220B (da)	1991-09-30
DK162220C true DK162220C (da)	1992-03-02

Family

ID=9337042

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK340987A DK162220C (da)	1986-07-03	1987-07-02	Tricykliske pyridazinderivater, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling af derivaterne, og laegemidler, hvori de er til stede

Country Status (16)

Country	Link
US (1)	US4977152A (da)
EP (1)	EP0251937B1 (da)
JP (1)	JPH029866A (da)
KR (1)	KR880001614A (da)
AR (1)	AR245123A1 (da)
AT (1)	ATE60589T1 (da)
AU (1)	AU602339B2 (da)
CA (1)	CA1312864C (da)
DE (1)	DE3767794D1 (da)
DK (1)	DK162220C (da)
ES (1)	ES2039256T3 (da)
FR (1)	FR2601011B1 (da)
GR (1)	GR3001646T3 (da)
NZ (1)	NZ220926A (da)
PT (1)	PT85234B (da)
ZA (1)	ZA874846B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2625201B1 (fr) *	1987-12-24	1990-06-15	Sanofi Sa	Nouveaux derives tricycliques agonistes des recepteurs cholinergiques et medicaments en contenant
US4985560A (en) *	1990-01-12	1991-01-15	American Home Products Corporation	Pyridazino(4,5-b)indolizines
US20100210590A1 (en) *	1995-09-27	2010-08-19	Northwestern University	Compositions and treatments for seizure-related disorders
US20030176437A1 (en) *	2001-08-31	2003-09-18	D.M. Watterson	Anti-inflammatory and protein kinase inhibitor compositions and related methods for downregulation of detrimental cellular responses and inhibition of cell death
KR100422589B1 (ko) *	2001-11-20	2004-03-16	(주)경인양행	셀룰로오스 섬유 또는 셀룰로오스 혼방섬유의 염색 방법
ATE523199T1 (de) *	2004-11-02	2011-09-15	Univ Northwestern	Pyridazinverbindungen und verfahren
BRPI0517947A (pt)	2004-11-02	2008-10-21	Univ Northwestern	composto de piridazina, composições e métodos
US20100168120A1 (en) *	2006-04-28	2010-07-01	Neuromedix Inc.	Salts of pyridazine compounds
CA2650711A1 (en) *	2006-04-28	2007-11-08	Northwestern University	Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
JP2009535344A (ja)	2006-04-28	2009-10-01	ノースウェスタンユニバーシティ	神経炎症性疾患の処置のためのピリダジン化合物を含む処方物
US20110052643A1 (en) *	2008-01-07	2011-03-03	Synta Pharmaceuticals Corp.	Compounds for inflammation and immune-related uses

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2510997A1 (fr) *	1981-08-10	1983-02-11	Sanofi Sa	Nouveaux derives de la methyl-4 phenyl-6 pyridazine, procede pour leur preparation et medicaments actifs sur le systeme nerveux central en contenant
FR2619818B1 (fr) *	1987-09-01	1990-01-12	Sanofi Sa	Imidazo (1,2-b) pyridazines, procede pour leur preparation et compositions pharmaceutiques les contenant

1986
- 1986-07-03 FR FR8609681A patent/FR2601011B1/fr not_active Expired
1987
- 1987-07-02 PT PT85234A patent/PT85234B/pt not_active IP Right Cessation
- 1987-07-02 AU AU75049/87A patent/AU602339B2/en not_active Ceased
- 1987-07-02 CA CA000541127A patent/CA1312864C/en not_active Expired - Fee Related
- 1987-07-02 AR AR87308037A patent/AR245123A1/es active
- 1987-07-02 DK DK340987A patent/DK162220C/da not_active IP Right Cessation
- 1987-07-02 NZ NZ220926A patent/NZ220926A/xx unknown
- 1987-07-03 JP JP62166746A patent/JPH029866A/ja active Pending
- 1987-07-03 KR KR1019870007113A patent/KR880001614A/ko not_active Ceased
- 1987-07-03 AT AT87401562T patent/ATE60589T1/de not_active IP Right Cessation
- 1987-07-03 ES ES198787401562T patent/ES2039256T3/es not_active Expired - Lifetime
- 1987-07-03 DE DE8787401562T patent/DE3767794D1/de not_active Expired - Fee Related
- 1987-07-03 ZA ZA874846A patent/ZA874846B/xx unknown
- 1987-07-03 EP EP87401562A patent/EP0251937B1/fr not_active Expired - Lifetime
1990
- 1990-01-25 US US07/471,680 patent/US4977152A/en not_active Expired - Fee Related
1991
- 1991-03-21 GR GR91400356T patent/GR3001646T3/el unknown

Also Published As

Publication number	Publication date
PT85234A (fr)	1987-08-01
AU602339B2 (en)	1990-10-11
PT85234B (pt)	1990-04-30
AU7504987A (en)	1988-01-07
EP0251937B1 (fr)	1991-01-30
CA1312864C (en)	1993-01-19
ZA874846B (en)	1988-03-30
KR880001614A (ko)	1988-04-25
DK340987D0 (da)	1987-07-02
JPH029866A (ja)	1990-01-12
NZ220926A (en)	1989-11-28
AR245123A1 (es)	1993-12-30
DK162220B (da)	1991-09-30
GR3001646T3 (en)	1992-11-23
FR2601011A1 (fr)	1988-01-08
FR2601011B1 (fr)	1988-10-28
ES2039256T3 (es)	1993-09-16
DE3767794D1 (de)	1991-03-07
US4977152A (en)	1990-12-11
DK340987A (da)	1988-01-04
ATE60589T1 (de)	1991-02-15
EP0251937A1 (fr)	1988-01-07

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Legal Events

Date	Code	Title	Description
1995-04-03	PBP	Patent lapsed